Efficient bioconjugation of 5-fluoro-5-deoxy-ribose (FDR) to RGD peptides for positron emission tomography (PET) imaging of αvβ3 integrin receptor

Translating the concept of peptidelabeling with 5-deoxy-5-[18F]fluororibose into preclinical practice: 18F-labeling of Siglec-9 peptide for PET imaging of inflammation

(2013) Xiang-Guo Li et al.   CHEMICAL COMMUNICATIONS

Carbohydrate-Based Molecules for Molecular Imaging in Nuclear Medicine

(2013) Goreti Ribeiro Morais et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

RGD-based PET tracers for imaging receptor integrin αvβ3expression

(2013) Hancheng Cai et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

[18F]-5-Fluoro-5-deoxyribose, an efficient peptide bioconjugation ligand for positron emission tomography (PET) imaging

(2012) Xiang-Guo Li et al.   CHEMICAL COMMUNICATIONS

Labeling Strategies of Peptides with 18F for Positron Emission Tomography

(2012) D. E. Olberg et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Oxime formation for fluorine-18 labeling of peptides and proteins for positron emission tomography (PET) imaging: A review

(2012) Xiang-Guo Li et al.   JOURNAL OF FLUORINE CHEMISTRY

Biodistribution and Radiation Dosimetry of the Integrin Marker 18F-RGD-K5 Determined from Whole-Body PET/CT in Monkeys and Humans

(2012) M. Doss et al.   JOURNAL OF NUCLEAR MEDICINE

One-step 18F-labeling of peptides for positron emission tomography imaging using the SiFA methodology

(2012) Carmen Wängler et al.   Nature Protocols

Quantitative Analysis and Comparison Study of [18F]AlF-NOTA-PRGD2, [18F]FPPRGD2 and [68Ga]Ga-NOTA-PRGD2 Using a Reference Tissue Model

(2012) Ning Guo et al.   PLoS One

Linear Trifluoroethylamine RGD Peptidomimetics: Stereoselective Synthesis and Integrin αvβ3 Affinity

(2012) Matteo Zanda et al.   SYNLETT

Integrin Targeted Delivery of Chemotherapeutics

(2012) Kai Chen et al.   Theranostics

Rapid and Simple One-Step F-18 Labeling of Peptides

(2011) Orit Jacobson et al.   BIOCONJUGATE CHEMISTRY

Comparison Study of [18F]FAl-NOTA-PRGD2, [18F]FPPRGD2, and [68Ga]Ga-NOTA-PRGD2 for PET Imaging of U87MG Tumors in Mice

(2011) Lixin Lang et al.   BIOCONJUGATE CHEMISTRY

Selective Formation of Covalent Protein Heterodimers with an Unnatural Amino Acid

(2011) Benjamin M. Hutchins et al.   CHEMISTRY & BIOLOGY

A fast, simple, and reproducible automated synthesis of [18F]FPyKYNE-c(RGDyK) for αvβ3 receptor positron emission tomography imaging

(2011) Ana C. Valdivia et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Monitoring Tumor Response to Antiangiogenic Sunitinib Therapy with 18F-Fluciclatide, an 18F-Labeled  V 3-Integrin and  V 5-Integrin Imaging Agent

(2011) M. R. Battle et al.   JOURNAL OF NUCLEAR MEDICINE

A new 18F-labeled BBN-RGD peptide heterodimer with a symmetric linker for prostate cancer imaging

(2010) Yongjun Yan et al.   AMINO ACIDS

A Novel Facile Method of Labeling Octreotide with 18F-Fluorine

(2010) P. Laverman et al.   JOURNAL OF NUCLEAR MEDICINE

Ligands for Mapping αvβ3-Integrin Expression in Vivo

(2009) Margret Schottelius et al.   ACCOUNTS OF CHEMICAL RESEARCH

A Novel Method for Direct Site-Specific Radiolabeling of Peptides Using [18F]FDG

(2009) Mohammad Namavari et al.   BIOCONJUGATE CHEMISTRY

18F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK)

(2009) Christina Hultsch et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Targeting the  v 3 Integrin for Small-Animal PET/CT of Osteolytic Bone Metastases

(2009) T. J. Wadas et al.   JOURNAL OF NUCLEAR MEDICINE

Molecular imaging targeting peptide receptors

(2009) Margret Schottelius et al.   METHODS

Methods for 18F-labeling of RGD peptides: comparison of aminooxy [18F]fluorobenzaldehyde condensation with ‘click labeling’ using 2-[18F]fluoroethylazide, and S-alkylation with [18F]fluoropropanethiol

(2008) Matthias Glaser et al.   AMINO ACIDS

Assessment of  v 3 integrin expression after myocardial infarction by positron emission tomography

(2008) T. Higuchi et al.   CARDIOVASCULAR RESEARCH

Molecular Imaging with PET

(2008) Simon M. Ametamey et al.   CHEMICAL REVIEWS

Integrin αvβ3-targeted cancer therapy

(2008) Zhaofei Liu et al.   DRUG DEVELOPMENT RESEARCH

Chemistry with [18F]Fluoride Ion

(2008) Lisheng Cai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Phase I Trial of the Positron-Emitting Arg-Gly-Asp (RGD) Peptide Radioligand 18F-AH111585 in Breast Cancer Patients

(2008) L. M. Kenny et al.   JOURNAL OF NUCLEAR MEDICINE

Recommendations on the Use of 18F-FDG PET in Oncology

(2008) J. W. Fletcher et al.   JOURNAL OF NUCLEAR MEDICINE

Preparation of a Promising Angiogenesis PET Imaging Agent: 68Ga-Labeled c(RGDyK)-Isothiocyanatobenzyl-1,4,7-Triazacyclononane-1,4,7-Triacetic Acid and Feasibility Studies in Mice

(2008) J. M. Jeong et al.   JOURNAL OF NUCLEAR MEDICINE