Infection Medications: Assessment In‐Vitro Glutathione S‐Transferase Inhibition and Molecular Docking Study

Synthesis of N ‐alkylated pyrazolo[3,4‐ d ]pyrimidine analogs and evaluation of acetylcholinesterase and carbonic anhydrase inhibition properties

(2021) Busra O. Aydin et al.   ARCHIV DER PHARMAZIE

Synthesis, Characterization, and Inhibition Study of Novel Substituted Phenylureido Sulfaguanidine Derivatives as α‐Glycosidase and Cholinesterase Inhibitors

(2021) Suleyman Akocak et al.   CHEMISTRY & BIODIVERSITY

Design, synthesis, characterization, in vitro and in silico evaluation of novel imidazo[2,1-b][1,3,4]thiadiazoles as highly potent acetylcholinesterase and non-classical carbonic anhydrase inhibitors

(2021) Sercan Askin et al.   BIOORGANIC CHEMISTRY

Identification of a new class of potent aldose reductase inhibitors: Design, microwave-assisted synthesis, in vitro and in silico evaluation of 2-pyrazolines

(2021) Belgin Sever et al.   CHEMICO-BIOLOGICAL INTERACTIONS

Transition‐Metal Complexes of Bidentate Schiff‐Base Ligands: In Vitro and In Silico Evaluation as Non‐Classical Carbonic Anhydrase and Potential Acetylcholinesterase Inhibitors

(2021) Ümit Yaşar et al.   ChemistrySelect

Calcium Channel Blockers: The Effect of Glutathione S‐Transferase Enzyme Activity and Molecular Docking Studies

(2021) Cüneyt Türkeş et al.   ChemistrySelect

Molecular Docking Studies and Inhibition Properties of Some Antineoplastic Agents against Paraoxonase-I

(2020) Yeliz Demir et al.   Anti-Cancer Agents in Medicinal Chemistry

Calcium Channel Blockers: Molecular Docking and Inhibition Studies on Carbonic Anhydrase I and II Isoenzymes

(2020) Cüneyt Türkeş et al.   JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS

Sulfonamides incorporating ketene N,S -acetal bioisosteres as potent carbonic anhydrase and acetylcholinesterase inhibitors

(2020) Qëndresa Istrefi et al.   ARCHIV DER PHARMAZIE

Determination of anticancer properties and inhibitory effects of some metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, alpha glycosidase of some compounds with molecular docking study

(2020) Fikret Türkan et al.   JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS

Synthesis, characterization, biological evaluation, and in silico studies of novel 1,3‐diaryltriazene‐substituted sulfathiazole derivatives

(2020) Mesut Işık et al.   ARCHIV DER PHARMAZIE

Synthesis, characterization, inhibition effects, and molecular docking studies as acetylcholinesterase, α-glycosidase, and carbonic anhydrase inhibitors of novel benzenesulfonamides incorporating 1,3,5-triazine structural motifs

(2020) Nebih Lolak et al.   BIOORGANIC CHEMISTRY

Benzenesulfonamide derivatives as potent acetylcholinesterase, α-glycosidase, and glutathione S-transferase inhibitors: biological evaluation and molecular docking studies

(2020) Parham Taslimi et al.   JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS

In vivo efficacy of ganciclovir by using single-walled carbon nanotubes as a drug carrier against infectious spleen and kidney necrosis virus in mandarin fish

(2020) Zhao Zhao et al.   AQUACULTURE

The distribution of mutations and hotspots in transcription regulators of resistance-nodulation-cell division efflux pumps in tigecycline non-susceptible Acinetobacter baumannii in China

(2020) Qingye Xu et al.   INTERNATIONAL JOURNAL OF MEDICAL MICROBIOLOGY

Glutathione-S-transferase Fusion Protein Nanosensor

(2020) Ryan M. Williams et al.   NANO LETTERS

Inhibitory effects of usnic and carnosic acid on some metabolic enzymes: an in vitro study

(2019) Hamid Ceylan et al.   PROTEIN AND PEPTIDE LETTERS

Investigation of Potential Paraoxonase-I Inhibitors by Kinetic and Molecular Docking Studies: Chemotherapeutic Drugs

(2019) Cüneyt Türkeş   PROTEIN AND PEPTIDE LETTERS

Anti-diabetic Properties of Calcium Channel Blockers: Inhibition Effects on Aldose Reductase Enzyme Activity

(2019) Cüneyt Türkeş et al.   APPLIED BIOCHEMISTRY AND BIOTECHNOLOGY

Inhibition of Human Serum Paraoxonase-I with Antimycotic Drugs: In Vitro and In Silico Studies

(2019) Cüneyt Türkeş et al.   APPLIED BIOCHEMISTRY AND BIOTECHNOLOGY

Gadolinium-based contrast agents: in vitro paraoxonase 1 inhibition, in silico studies

(2019) Şükrü Beydemir et al.   DRUG AND CHEMICAL TOXICOLOGY

A potential risk factor for paraoxonase 1: in silico and in‐vitro analysis of the biological activity of proton‐pump inhibitors

(2019) Cüneyt Türkeş   JOURNAL OF PHARMACY AND PHARMACOLOGY

Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors

(2019) Cüneyt Türkeş et al.   BIOORGANIC CHEMISTRY

In Vitro and In Silico Studies on the Toxic Effects of Antibacterial Drugs as Human Serum Paraoxonase 1 Inhibitor

(2019) Cüneyt Türkeş et al.   ChemistrySelect

Benzenesulfonamide derivatives containing imine and amine groups: Inhibition on human paraoxonase and molecular docking studies

(2019) Mesut Işık et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

New Isoindole‐1,3‐dione Substituted Sulfonamides as Potent Inhibitors of Carbonic Anhydrase and Acetylcholinesterase: Design, Synthesis, and Biological Evaluation

(2019) Saliha Gündoğdu et al.   ChemistrySelect

Evaluation of chalcones as inhibitors of glutathione S-transferase

(2018) Muhammet Serhat Özaslan et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Evaluation of synergistic anticandidal and apoptotic effects of ferulic acid and caspofungin against Candida albicans

(2018) Zerrin Canturk   JOURNAL OF FOOD AND DRUG ANALYSIS

The effects of some cephalosporins on acetylcholinesterase and glutathione S-transferase: an in vivo and in vitro study

(2018) Fikret Türkan et al.   ARCHIVES OF PHYSIOLOGY AND BIOCHEMISTRY

Glutathione transferases: substrates, inihibitors and pro-drugs in cancer and neurodegenerative diseases

(2018) Nerino Allocati et al.   Oncogenesis

Investigation of the effects of cephalosporin antibiotics on glutathione S-transferase activity in different tissues of rats in vivo conditions in order to drug development research

(2018) Fikret Türkan et al.   DRUG AND CHEMICAL TOXICOLOGY

The toxicological impact of some avermectins on human erythrocytes glutathione S-transferase enzyme

(2018) Fikret Türkan et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Organometallic Glutathione S-Transferase Inhibitors

(2017) Emilia Păunescu et al.   ORGANOMETALLICS

Drug resistance and treatment failure in leishmaniasis: A 21st century challenge

(2017) Alicia Ponte-Sucre et al.   PLoS Neglected Tropical Diseases

Epidemiology and microbiology of skin and soft tissue infections

(2016) Silvano Esposito et al.   CURRENT OPINION IN INFECTIOUS DISEASES

In vitro inhibitory effects of palonosetron hydrochloride, bevacizumab and cyclophosphamide on purified paraoxonase-I (hPON1) from human serum

(2016) Cüneyt Türkeş et al.   ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY

In vitro activity of anidulafungin in combination with amphotericin B or voriconazole against biofilms of five Candida species

(2016) A. Valentín et al.   JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY

Rosmarinic acid inhibits some metabolic enzymes including glutathione S-transferase, lactoperoxidase, acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase isoenzymes

(2016) İlhami Gülçin et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Influence of glutathione-S-transferase (GST) inhibition on lung epithelial cell injury: role of oxidative stress and metabolism

(2015) Marianne E. Fletcher et al.   AMERICAN JOURNAL OF PHYSIOLOGY-LUNG CELLULAR AND MOLECULAR PHYSIOLOGY

Antioxidant role of glutathione S-transferases: 4-Hydroxynonenal, a key molecule in stress-mediated signaling

(2015) Sharad S. Singhal et al.   TOXICOLOGY AND APPLIED PHARMACOLOGY

Changes in the anti-oxidant system in adult epilepsy patients receiving anti-epileptic drugs

(2015) Mesut Işık et al.   ARCHIVES OF PHYSIOLOGY AND BIOCHEMISTRY

Human serum paraoxonase-1 (hPON1):in vitroinhibition effects of moxifloxacin hydrochloride, levofloxacin hemihidrate, cefepime hydrochloride, cefotaxime sodium and ceftizoxime sodium

(2014) Cüneyt Türkeş et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Effect of calcium channel blockers on paraoxonase-1 (PON1) activity and oxidative stress

(2014) Cüneyt Türkeş et al.   Pharmacological Reports

Computational modelling of novel inhibitors targeting the human GSTP1*D homology domain

(2013) Yu Xu et al.   MOLECULAR SIMULATION

Purification and characterization of glutathione S-transferase from turkey liver and inhibition effects of some metal ions on enzyme activity

(2012) Ebru Akkemik et al.   ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY

Synthesis and paroxonase activities of novel bromophenols

(2012) Yusuf Akbaba et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

A novel method for screening the glutathione transferase inhibitors

(2009) Zhijun Wang et al.   BMC BIOCHEMISTRY

Limonin Methoxylation Influences the Induction of GlutathioneS-Transferase and Quinone Reductase

(2009) Jose Luis Perez et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

The Anti-cancer Drug Chlorambucil as a Substrate for the Human Polymorphic Enzyme Glutathione Transferase P1-1: Kinetic Properties and Crystallographic Characterisation of Allelic Variants

(2008) Lorien J. Parker et al.   JOURNAL OF MOLECULAR BIOLOGY