The synthesis of perfluoroalkylated indolizines via tandem cyclization/aromatization

Facile preparation and conversion of 4,4,4-trifluorobut-2-yn-1-ones to aromatic and heteroaromatic compounds

(2021) Takashi Yamazaki et al.   Beilstein Journal of Organic Chemistry

Cu(I)-Catalyzed [2 + 2 + 1] Cycloaddition of Amines, Alkynes, and Ketenes: An Umpolung and Regioselective Approach to Full-Substituted β-Pyrrolinones

(2021) Hao Wu et al.   ORGANIC LETTERS

New Visible Light‐triggered Photocatalytic Trifluoromethylation Reactions of Carbon‐carbon Multiple Bonds and (Hetero)aromatic Compounds

(2020) SEBASTIAN BARATA-VALLEJO et al.   CHEMISTRY-A EUROPEAN JOURNAL

Contribution of Organofluorine Compounds to Pharmaceuticals

(2020) Munenori Inoue et al.   ACS Omega

Progress in Electrochemical Trifluoromethylation Reactions

(2020) Rasmi P. Bhaskaran et al.   ADVANCED SYNTHESIS & CATALYSIS

Base-promoted [3+2] cycloaddition/aromatization cascade reaction under air: An approach to access perfluoroalkylated pyrrolo[2,1-a]isoquinolines

(2019) Wei Zhou et al.   JOURNAL OF FLUORINE CHEMISTRY

Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design

(2018) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Potassium iodide promoted one-pot synthesis of fluoroalkylated quinoxalines via a tandem Michael addition / azidation / cycloamination approach

(2018) Jun Wu et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium(III)-Catalyzed Directed C–H Coupling with Methyl Trifluoroacrylate: Diverse Synthesis of Fluoroalkenes and Heterocycles

(2018) Tian-Jun Gong et al.   ORGANIC LETTERS

Novel synthesis of perfluoroalkylated indolizinylphosphonates via a DIPEA-promoted one-pot process

(2018) Hao Liu et al.   TETRAHEDRON

Iron-Catalyzed Indolizine Synthesis from Pyridines, Diazo Compounds, and Alkynes

(2017) Tim Douglas et al.   ORGANIC LETTERS

Trifluoromethyl nitrogen heterocycles: synthetic aspects and potential biological targets

(2016) F. Meyer   CHEMICAL COMMUNICATIONS

Copper-Catalyzed C-H Alkynylation/Intramolecular Cyclization Cascade for the First Synthesis of Trifluoromethylated Pyrrolo[1,2-a]quinolines

(2016) Zhiliang Xu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Recent advances in the synthesis of indolizines and their π-expanded analogues

(2016) Bartłomiej Sadowski et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A [4 + 1] Cyclative Capture Access to Indolizines via Cobalt(III)-Catalyzed Csp2–H Bond Functionalization

(2016) Xun Chen et al.   ORGANIC LETTERS

Rh(III)-Catalyzed Oxidative Annulation Leading to Substituted Indolizines by Cleavage of C(sp2)–H/C(sp3)–H Bonds

(2016) Bingxue Shen et al.   ORGANIC LETTERS

1,3-Dipolar Cycloaddition with Diazo Groups: Noncovalent Interactions Overwhelm Strain

(2016) Brian Gold et al.   ORGANIC LETTERS

Trifluoromethyl aldimines: an overview in the last ten years

(2016) Stefania Fioravanti   TETRAHEDRON

External-Photocatalyst-Free Visible-Light-Mediated Synthesis of Indolizines

(2015) Basudev Sahoo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Carbon Trifluoromethylation Reactions of Hydrocarbon Derivatives and Heteroarenes

(2015) Concepción Alonso et al.   CHEMICAL REVIEWS

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Mild and Efficient One-Pot Synthesis of 2-(Perfluoroalkyl)indoles by Means of Sequential Michael-Type Addition and Pd(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) Reaction

(2015) Dandan Shen et al.   ORGANIC LETTERS

Application of Langlois’ Reagent in Trifluoromethylation Reactions

(2014) Cai Zhang   ADVANCED SYNTHESIS & CATALYSIS

Trifluoromethyltrimethylsilane: Nucleophilic Trifluoromethylation and Beyond

(2014) Xiao Liu et al.   CHEMICAL REVIEWS

Electrophilic Trifluoromethylation by Use of Hypervalent Iodine Reagents

(2014) Julie Charpentier et al.   CHEMICAL REVIEWS

Indolizine: a biologically active moiety

(2014) Vikas Sharma et al.   MEDICINAL CHEMISTRY RESEARCH

Recent advances in trifluoromethylation of organic compounds using Umemoto's reagents

(2014) Cai Zhang   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(I)-Catalyzed Coupling Cyclization of Methyl Perfluoroalk-2-ynoates with 2-Aminobenzonitriles: Synthesis of 2-Perfluoroalkylated Quinolines

(2013) Jing Han et al.   ADVANCED SYNTHESIS & CATALYSIS

Domino Knoevenagel Condensation/Intramolecular Aldol Cyclization Route to Diverse Indolizines with Densely Functionalized Pyridine Units

(2013) Myungock Kim et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium and Copper Cocatalyzed Tandem N–H/C–H Bond Functionalization: Synthesis of CF3-Containing Indolo- and Pyrrolo[2,1-a]isoquinolines

(2012) Lei-Lei Sun et al.   JOURNAL OF ORGANIC CHEMISTRY

First one-pot stereoselective synthesis of cis-2,3-dihydro-4-perfluoroalkyl-1H-1,5-benzodiazepines via a catalyst-free three-component reaction

(2011) Jiechao Xu et al.   CHEMICAL COMMUNICATIONS

Recent progress in synthesis and bioactivity studies of indolizines

(2011) Girija S. Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY