Improving the metabolic stability of antifungal compounds based on a scaffold hopping strategy: Design, synthesis, and structure-activity relationship studies of dihydrooxazole derivatives
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Title
Improving the metabolic stability of antifungal compounds based on a scaffold hopping strategy: Design, synthesis, and structure-activity relationship studies of dihydrooxazole derivatives
Authors
Keywords
CYP51, Azole antifungals, Metabolic stability, Dihydrooxazole derivatives
Journal
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 224, Issue -, Pages 113715
Publisher
Elsevier BV
Online
2021-07-22
DOI
10.1016/j.ejmech.2021.113715
References
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