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Multidrug resistance proteins (MRPs): Structure, function and the overcoming of cancer multidrug resistance

(2021) Jing-Quan Wang et al.   DRUG RESISTANCE UPDATES

Global cancer statistics 2020: GLOBOCAN estimates of incidence and mortality worldwide for 36 cancers in 185 countries

(2021) Hyuna Sung et al.   CA-A CANCER JOURNAL FOR CLINICIANS

ABCG2 transports anticancer drugs via a closed-to-open switch

(2020) Benjamin J. Orlando et al.   Nature Communications

Pyrimidine: A promising scaffold for optimization to develop the inhibitors of ABC transporters

(2020) Zhang-Xu He et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Superior Pyrimidine Derivatives as Selective ABCG2 Inhibitors and Broad-spectrum ABCB1, ABCC1, and ABCG2 Antagonists

(2020) Katja Silbermann et al.   JOURNAL OF MEDICINAL CHEMISTRY

Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2

(2020) Emile Roussel et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cellular expression and function of naturally occurring variants of the human ABCG2 multidrug transporter

(2019) Boglárka Zámbó et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Role of ATP-binding cassette transporters in cancer initiation and progression

(2019) Stefania Nobili et al.   SEMINARS IN CANCER BIOLOGY

New desulfured troglitazone derivatives: Improved synthesis and biological evaluation

(2019) Dorian Dupommier et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Polymorphisms of ABCG2 and its impact on clinical relevance

(2018) Wenji Zhang et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Understanding of human ATP binding cassette superfamily and novel multidrug resistance modulators to overcome MDR

(2018) Imran Shair Mohammad et al.   BIOMEDICINE & PHARMACOTHERAPY

New Inhibitors of Breast Cancer Resistance Protein (ABCG2) Containing a 2,4-Disubstituted Pyridopyrimidine Scaffold

(2018) Michael K. Krapf et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer’s disease therapy

(2018) Youssef Dgachi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Mammalian drug efflux transporters of the ATP binding cassette (ABC) family in multidrug resistance: A review of the past decade

(2016) Zhaolin Chen et al.   CANCER LETTERS

Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Aβ1−42Aggregation Inhibitors for Alzheimer's Disease Therapy

(2016) Youssef Dgachi et al.   ChemMedChem

Molecular mechanisms for tumour resistance to chemotherapy

(2016) Shu-Ting Pan et al.   CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY

Overcoming ABC transporter-mediated multidrug resistance: Molecular mechanisms and novel therapeutic drug strategies

(2016) Wen Li et al.   DRUG RESISTANCE UPDATES

Synthesis and Biological Evaluation of 4-Anilino-quinazolines and -quinolines as Inhibitors of Breast Cancer Resistance Protein (ABCG2)

(2016) Michael K. Krapf et al.   JOURNAL OF MEDICINAL CHEMISTRY

Scaffold Identification of a New Class of Potent and Selective BCRP Inhibitors

(2015) Federico Marighetti et al.   ChemMedChem

The controversial role of ABC transporters in clinical oncology

(2011) Akina Tamaki et al.   Essays in Biochemistry

Synthesis and biological evaluation of a small molecule library of 3rd generation multidrug resistance modulators

(2009) Werner Klinkhammer et al.   BIOORGANIC & MEDICINAL CHEMISTRY

ABC Efflux Pump-Based Resistance to Chemotherapy Drugs

(2009) Paul D. W. Eckford et al.   CHEMICAL REVIEWS

Aromatic 2-(Thio)ureidocarboxylic Acids As a New Family of Modulators of Multidrug Resistance-Associated Protein 1: Synthesis, Biological Evaluation, and Structure−Activity Relationships

(2009) Hans-Georg Häcker et al.   JOURNAL OF MEDICINAL CHEMISTRY

Three-Component Synthesis of Pyrimidine and Pyrimidinone Derivatives in the Presence of High-Surface-Area MgO, a Highly Effective Heterogeneous Base Catalyst

(2009) Hassan Sheibani et al.   SYNTHETIC COMMUNICATIONS

A 4-aminobenzoic acid derivative as novel lead for selective inhibitors of multidrug resistance-associated proteins

(2008) Stefan Leyers et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Dimethoxyaurones: Potent inhibitors of ABCG2 (breast cancer resistance protein)

(2008) Hong-May Sim et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES