Scaffold Identification of a New Class of Potent and Selective BCRP Inhibitors

Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2)

(2013) Kapil Juvale et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2

(2013) Kapil Juvale et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

4-Substituted-2-phenylquinazolines as inhibitors of BCRP

(2012) Kapil Juvale et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and Quantitative Structure-Activity Relationships of Selective BCRP Inhibitors

(2012) Federico Marighetti et al.   ChemMedChem

Tyrosine Kinase Inhibitors Influence ABCG2 Expression in EGFR-Positive MDCK BCRP Cells via the PI3K/Akt Signaling Pathway

(2012) Anne Pick et al.   ChemMedChem

Structure–Activity Relationships, Ligand Efficiency, and Lipophilic Efficiency Profiles of Benzophenone-Type Inhibitors of the Multidrug Transporter P-Glycoprotein

(2012) Ishrat Jabeen et al.   JOURNAL OF MEDICINAL CHEMISTRY

Investigation of chalcones and benzochalcones as inhibitors of breast cancer resistance protein

(2011) Kapil Juvale et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Structure–activity relationships of flavonoids as inhibitors of breast cancer resistance protein (BCRP)

(2010) Anne Pick et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Specific Inhibitors of the Breast Cancer Resistance Protein (BCRP)

(2010) Anne Pick et al.   ChemMedChem

Novel lead for potent inhibitors of breast cancer resistance protein (BCRP)

(2009) Anne Pick et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Physiological and pharmacological roles of ABCG2 (BCRP): Recent findings in Abcg2 knockout mice

(2008) Maria L.H. Vlaming et al.   ADVANCED DRUG DELIVERY REVIEWS

Membrane Topology of the Human Breast Cancer Resistance Protein (BCRP/ABCG2) Determined by Epitope Insertion and Immunofluorescence†

(2008) Honggang Wang et al.   BIOCHEMISTRY

Structure–activity relationships of new inhibitors of breast cancer resistance protein (ABCG2)

(2008) Anne Pick et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Drug transporters: recent advances concerning BCRP and tyrosine kinase inhibitors

(2008) C Lemos et al.   BRITISH JOURNAL OF CANCER

Functional assay and structure–activity relationships of new third-generation P-glycoprotein inhibitors

(2007) Henrik Müller et al.   BIOORGANIC & MEDICINAL CHEMISTRY