Recent developments with boron as a platform for novel drug design

Carborane-based design of a potent vitamin D receptor agonist

(2016) Rocio Otero et al.   Chemical Science

Boron-Based Drug Design

(2015) Hyun Seung Ban et al.   CHEMICAL RECORD

Synthesis and Applications of Boronic Acid-Containing Polymers: From Materials to Medicine

(2015) William L. A. Brooks et al.   CHEMICAL REVIEWS

nido-Dicarbaborate Induces Potent and Selective Inhibition of Cyclooxygenase-2

(2015) Wilma Neumann et al.   ChemMedChem

Synthesis and in vitro antiviral activity of lipophilic pyrimidine nucleoside/carborane conjugates

(2015) Magdalena Białek-Pietras et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Boron clusters in medicinal chemistry: perspectives and problems

(2015) Detlef Gabel   PURE AND APPLIED CHEMISTRY

The First CNS-Active Carborane: A Novel P2X7 Receptor Antagonist with Antidepressant Activity

(2014) Shane M. Wilkinson et al.   ACS Chemical Neuroscience

Carborane-Derived Local Anesthetics are Isomer Dependent

(2014) George R. Kracke et al.   ChemMedChem

Carborane-Based Carbonic Anhydrase Inhibitors

(2013) Jiří Brynda et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Potency and Spectrum of Activity of AN3365, a Novel Boron-Containing Protein Synthesis Inhibitor, Tested against Clinical Isolates of Enterobacteriaceae and Nonfermentative Gram-Negative Bacilli

(2013) Rodrigo E. Mendes et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

2-Carbaborane-3-phenyl-1H-indoles-Synthesis via McMurry Reaction and Cyclooxygenase (COX) Inhibition Activity

(2013) Markus Laube et al.   ChemMedChem

Boron chemicals in diagnosis and therapeutics

(2013) Bhaskar C Das et al.   Future Medicinal Chemistry

QM/MM Calculations Reveal the Different Nature of the Interaction of Two Carborane-Based Sulfamide Inhibitors of Human Carbonic Anhydrase II

(2013) Adam Pecina et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Effect of adenosine modified with a boron cluster pharmacophore on reactive oxygen species production by human neutrophils

(2012) Katarzyna Bednarska et al.   BIOORGANIC & MEDICINAL CHEMISTRY

ortho-Carbaborane derivatives of indomethacin as cyclooxygenase (COX)-2 selective inhibitors

(2012) Matthias Scholz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and evaluation of carbaborane derivatives of indomethacin as cyclooxygenase inhibitors

(2011) Matthias Scholz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbaboranes as Pharmacophores: Properties, Synthesis, and Application Strategies

(2011) Matthias Scholz et al.   CHEMICAL REVIEWS

Boron in Drug Discovery: Carboranes as Unique Pharmacophores in Biologically Active Compounds

(2011) Fatiah Issa et al.   CHEMICAL REVIEWS

Carbaboranes as pharmacophores: Similarities and differences between aspirin and asborin

(2011) Matthias Scholz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Boron Cluster-based Development of Potent Nonsecosteroidal Vitamin D Receptor Ligands: Direct Observation of Hydrophobic Interaction between Protein Surface and Carborane

(2011) Shinya Fujii et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Proteomic Analysis of Excretory-Secretory Products of Heligmosomoides polygyrus Assessed with Next-Generation Sequencing Transcriptomic Information

(2011) Yovany Moreno et al.   PLoS Neglected Tropical Diseases

Asborin Inhibits Aldo/Keto Reductase 1A1

(2010) Matthias Scholz et al.   ChemMedChem

Adenosine and 2′-Deoxyadenosine Modified with Boron Cluster Pharmacophores as New Classes of Human Blood Platelet Function Modulators

(2010) Katarzyna Bednarska et al.   ChemMedChem

ADVANCES AT THE INTERFACE OF POLYHEDRAL BORANE CHEMISTRY AND MEDICINE

(2010) M. Frederick Hawthorne   COMMENTS ON INORGANIC CHEMISTRY

Asborin: The Carbaborane Analogue of Aspirin

(2009) Matthias Scholz et al.   ChemMedChem

Therapeutic potential of boron-containing compounds

(2009) Stephen J Baker et al.   Future Medicinal Chemistry

Discovery of 3-acetyl-4-hydroxy-2-pyranone derivatives and their difluoridoborate complexes as a novel class of HIV-1 integrase Inhibitors

(2008) Kavya Ramkumar et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure

(2008) Shinya Fujii et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Self-assembled 2D supramolecular networks of copper(i) carborane complexes through C–H⋯H–B dihydrogen bonding interactions

(2008) Jianmin Dou et al.   DALTON TRANSACTIONS

The dipeptidyl peptidase-4 inhibitor PHX1149 improves blood glucose control in patients with type 2 diabetes mellitus

(2008) G. Garcia-Soria et al.   DIABETES OBESITY & METABOLISM

The kinetics and mechanism of the acid-catalysed detritylation of nucleotides in non-aqueous solution

(2008) Mark A. Russell et al.   ORGANIC & BIOMOLECULAR CHEMISTRY