2-Carbaborane-3-phenyl-1H-indoles-Synthesis via McMurry Reaction and Cyclooxygenase (COX) Inhibition Activity

Radiosynthesis of a 18F-labeled 2,3-diarylsubstituted indole via McMurry coupling for functional characterization of cyclooxygenase-2 (COX-2) in vitro and in vivo

(2012) Torsten Kniess et al.   BIOORGANIC & MEDICINAL CHEMISTRY

ortho-Carbaborane derivatives of indomethacin as cyclooxygenase (COX)-2 selective inhibitors

(2012) Matthias Scholz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carboranes Increase the Potency of Small Molecule Inhibitors of Nicotinamide Phosphoribosyltranferase

(2012) Mark W. Lee et al.   JOURNAL OF MEDICINAL CHEMISTRY

Imitation and modification of bioactive lead structures via integration of boron clusters

(2012) Sven Stadlbauer et al.   PURE AND APPLIED CHEMISTRY

Synthesis and evaluation of carbaborane derivatives of indomethacin as cyclooxygenase inhibitors

(2011) Matthias Scholz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Fluorinated COX-2 Inhibitors as Agents in PET Imaging of Inflammation and Cancer

(2011) M. J. Uddin et al.   Cancer Prevention Research

Carbaboranes as Pharmacophores: Properties, Synthesis, and Application Strategies

(2011) Matthias Scholz et al.   CHEMICAL REVIEWS

Boron in Drug Discovery: Carboranes as Unique Pharmacophores in Biologically Active Compounds

(2011) Fatiah Issa et al.   CHEMICAL REVIEWS

Carbaboranes as pharmacophores: Similarities and differences between aspirin and asborin

(2011) Matthias Scholz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cyclooxygenase-2 inhibitors: a literature and patent review (2009 – 2010)

(2011) Baker Jawabrah Al-Hourani et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Incorporation ofortho-Carbaboranyl-Nε-Modifiedl-Lysine into Neuropeptide Y Receptor Y1- and Y2-Selective Analogues

(2011) Verena M. Ahrens et al.   JOURNAL OF MEDICINAL CHEMISTRY

Celecoxib Enhances Radiation Response of Secondary Bone Tumors of a Human Non-Small Cell Lung Cancer via Antiangiogenesis In Vivo

(2011) Frank Michael Klenke et al.   STRAHLENTHERAPIE UND ONKOLOGIE

Selective Visualization of Cyclooxygenase-2 in Inflammation and Cancer by Targeted Fluorescent Imaging Agents

(2010) Md. Jashim Uddin et al.   CANCER RESEARCH

[123I]-Celecoxib Analogues as SPECT Tracers of Cyclooxygenase-2 in Inflammation

(2010) Md. Jashim Uddin et al.   ACS Medicinal Chemistry Letters

Asborin: The Carbaborane Analogue of Aspirin

(2009) Matthias Scholz et al.   ChemMedChem

Polyhedral Boranes for Medical Applications: Current Status and Perspectives

(2009) Igor B. Sivaev et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

The search for new COX-2 inhibitors: a review of 2002 – 2008 patents

(2009) Teodorico C Ramalho et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

The COXIB Experience: A Look in the Rearview Mirror

(2008) Lawrence J. Marnett   Annual Review of Pharmacology and Toxicology

Exploration of physicochemical properties and molecular modelling studies of 2-sulfonyl-phenyl-3-phenyl-indole analogs as cyclooxygenase-2 inhibitors

(2007) Arun Kumar Gupta et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY