Synthesis of novel 5-(2,5-bis(2,2,2-trifluoroethoxy)phenyl)-1,3,4-oxadiazole-2-thiol derivatives as potential glucosidase inhibitors
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Title
Synthesis of novel 5-(2,5-bis(2,2,2-trifluoroethoxy)phenyl)-1,3,4-oxadiazole-2-thiol derivatives as potential glucosidase inhibitors
Authors
Keywords
Antidiabetic agent, 1,3,4-Oxadiazole, Antioxidant, α-Amylase, α-Glucosidase, Molecular docking
Journal
BIOORGANIC CHEMISTRY
Volume 114, Issue -, Pages 105046
Publisher
Elsevier BV
Online
2021-05-31
DOI
10.1016/j.bioorg.2021.105046
References
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- Synthesis and molecular modelling studies of phenyl linked oxadiazole-phenylhydrazone hybrids as potent antileishmanial agents
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- Synthesis, characterization and biological evaluation of novel 2,5 substituted-1,3,4 oxadiazole derivatives
- (2017) Selvaraj Kavitha et al. SAUDI PHARMACEUTICAL JOURNAL
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- Clinical Review of Antidiabetic Drugs: Implications for Type 2 Diabetes Mellitus Management
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- UsingDrosophilato discover mechanisms underlying type 2 diabetes
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- Synthesis of novel inhibitors of α-glucosidase based on the benzothiazole skeleton containing benzohydrazide moiety and their molecular docking studies
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- Design, synthesis, in silico molecular docking and biological evaluation of novel oxadiazole based thiazolidine-2,4-diones bis-heterocycles as PPAR-γ agonists
- (2014) Syed Nazreen et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and molecular docking studies of potent α-glucosidase inhibitors based on biscoumarin skeleton
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- Development of Thiadiazole as an Antidiabetic Agent- A Review
- (2014) Prasanna Datar et al. MINI-REVIEWS IN MEDICINAL CHEMISTRY
- The majority of patients with long-duration type 1 diabetes are insulin microsecretors and have functioning beta cells
- (2013) Richard A. Oram et al. DIABETOLOGIA
- Mexican Antidiabetic Herbs: Valuable Sources of Inhibitors of α-Glucosidases
- (2013) Rachel Mata et al. JOURNAL OF NATURAL PRODUCTS
- Identification, optimisation and in vivo evaluation of oxadiazole DGAT-1 inhibitors for the treatment of obesity and diabetes
- (2012) William McCoull et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis, hypoglycemic and hypolipidemic activities of novel thiazolidinedione derivatives containing thiazole/triazole/oxadiazole ring
- (2012) A.K. Mohammed Iqbal et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of variously coupled conjugates of d-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase
- (2011) Sándor Kun et al. CARBOHYDRATE RESEARCH
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- (2011) Mayurkumar B. Patel et al. Journal of Functional Foods
- Derivatives of benzimidazole pharmacophore: Synthesis, anticonvulsant, antidiabetic and DNA cleavage studies
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