Hydrophobic Pocket Occupation Design of Difluoro-Biphenyl-Diarylpyrimidines as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: from N-Alkylation to Methyl Hopping on the Pyrimidine Ring
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Title
Hydrophobic Pocket Occupation Design of Difluoro-Biphenyl-Diarylpyrimidines as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: from N-Alkylation to Methyl Hopping on the Pyrimidine Ring
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 64, Issue 8, Pages 5067-5081
Publisher
American Chemical Society (ACS)
Online
2021-04-16
DOI
10.1021/acs.jmedchem.1c00128
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