Bridging C−H Activation: Mild and Versatile Cleavage of the 8-Aminoquinoline Directing Group

Copper-Mediatedortho-Arylation of Benzamides with Arylboronic Acid

(2016) Qingwen Gui et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly mono-selective ortho-trifluoromethylation of benzamides via 8-aminoquinoline assisted Cu-promoted C–H activations

(2016) Liang Hu et al.   CHEMICAL COMMUNICATIONS

Photocatalytic/Cu-Promoted C−H Activations: Visible-light-Inducedortho-Selective Perfluoroalkylation of Benzamides

(2016) Xiang Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Pd-Catalyzed Directed Chlorination of Unactivated C(sp3 )-H Bonds at Room Temperature

(2016) Heng-Ying Xiong et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Making the Least Reactive Electrophile the First in Class: Domino Electrophilic Activation of Amides

(2016) Daniel Kaiser et al.   JOURNAL OF ORGANIC CHEMISTRY

Stereoselective Synthesis of Diazabicyclic β-Lactams through Intramolecular Amination of Unactivated C(sp3)–H Bonds of Carboxamides by Palladium Catalysis

(2016) Shi-Jin Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Access to Different Isomeric Dibenzoxazepinones through Copper-Catalyzed C–H Etherification and C–N Bond Construction with Controllable Smiles Rearrangement

(2016) Yunfei Zhou et al.   ORGANIC LETTERS

Strong Bonds Made Weak: Towards the General Utility of Amides as Synthetic Modules

(2015) Stefan A. Ruider et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ligand-Promoted Borylation of C(sp3 )H Bonds with Palladium(II) Catalysts

(2015) Jian He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(0)/PAr3-Catalyzed Intermolecular Amination of C(sp3)H Bonds: Synthesis of β-Amino Acids

(2015) Jian He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Directed C(sp3)-H Arylation of Saturated Heterocycles at C-3 Using a Concise Optimization Approach

(2015) Dominic P. Affron et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Direct Observation of Intermediates Involved in the Interruption of the Bischler–Napieralski Reaction

(2015) Kolby L. White et al.   JOURNAL OF ORGANIC CHEMISTRY

Regio- and Stereoselective Pd-Catalyzed Direct Arylation of Unactivated sp3 C(3)–H Bonds of Tetrahydrofuran and 1,4-Benzodioxane Systems

(2015) Ramarao Parella et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Intramolecular Dehydrogenative Amidation of Unactivated C(sp3)–H Bonds Using O2 as the Sole Oxidant

(2015) Chunxia Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Aromatic abietane diterpenoids: their biological activity and synthesis

(2015) Miguel A. González   NATURAL PRODUCT REPORTS

Conversion of amides to esters by the nickel-catalysed activation of amide C–N bonds

(2015) Liana Hie et al.   NATURE

Copper-Mediated Oxidative Coupling of Benzamides with Maleimides via Directed C–H Cleavage

(2015) Wataru Miura et al.   ORGANIC LETTERS

Bidentate ligand 8-aminoquinoline-aided Pd-catalyzed diastereoselective β-arylation of the prochiral secondary sp3 C–H bonds of 2-phenylbutanamides and related aliphatic carboxamides

(2015) Bojan Gopalakrishnan et al.   TETRAHEDRON

Cobalt-catalysed site-selective intra- and intermolecular dehydrogenative amination of unactivated sp3 carbons

(2015) Xuesong Wu et al.   Nature Communications

Sulfonamide-Promoted Palladium(II)-Catalyzed Alkylation of Unactivated Methylene C(sp3)H Bonds with Alkyl Iodides

(2014) Kai Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-Catalyzed C(sp2)H Alkylation of Carboxamides with Primary Electrophiles

(2014) Brendan M. Monks et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Intramolecular C(sp3)H and C(sp2)H Amidation by Oxidative Cyclization

(2014) Zhen Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Site-Selective Intramolecular Amidation of Unactivated C(sp3)H Bonds

(2014) Xuesong Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed CH Alkylations: Direct Secondary Alkylations and Trifluoroethylations of Arenes

(2014) Weifeng Song et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Unlocking nature’s CH bonds

(2014) Marcus E. Farmer et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Nickel-Catalyzed Site-Selective Amidation of Unactivated C(sp3)H Bonds

(2014) Xuesong Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Applications of C–H Functionalization Logic to Cyclobutane Synthesis

(2014) Will R. Gutekunst et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Aryl C–H Olefination with Unactivated, Aliphatic Alkenes

(2014) Arghya Deb et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Anthranilic Acid Derivatives through Iron-Catalyzed Ortho Amination of Aromatic Carboxamides with N-Chloroamines

(2014) Tatsuaki Matsubara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regio- and Stereospecific Synthesis of C-3 Functionalized Proline Derivatives by Palladium Catalyzed Directed C(sp3)–H Arylation

(2014) Dominic P. Affron et al.   ORGANIC LETTERS

Cobalt-Catalyzed, Aminoquinoline-Directed Coupling of sp2 C–H Bonds with Alkenes

(2014) Liene Grigorjeva et al.   ORGANIC LETTERS

Copper-Mediated Direct C(sp3)–H and C(sp2)–H Acetoxylation

(2014) Zhen Wang et al.   ORGANIC LETTERS

Copper-Mediated Tandem Oxidative C(sp2)–H/C(sp)–H Alkynylation and Annulation of Arenes with Terminal Alkynes

(2014) Jiaxing Dong et al.   ORGANIC LETTERS

Palladium-catalyzed trifluoroacetate-promoted mono-arylation of the β-methyl group of alanine at room temperature: synthesis of β-arylated α-amino acids through sequential C–H functionalization

(2014) Bo Wang et al.   Chemical Science

An Efficient Palladium-Catalyzed CH Alkoxylation of Unactivated Methylene and Methyl Groups with Cyclic Hypervalent Iodine (I3+) Oxidants

(2013) Gang Shan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

8-Aminoquinoline: A Powerful Directing Group in Metal-Catalyzed Direct Functionalization of CH Bonds

(2013) Matthieu Corbet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Use of a Readily Removable Auxiliary Group for the Synthesis of Pyrrolidones by the Palladium-Catalyzed Intramolecular Amination of Unactivated γ C(sp3)H Bonds

(2013) Gang He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

β-Arylation of Carboxamides via Iron-Catalyzed C(sp3)–H Bond Activation

(2013) Rui Shang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nickel-Catalyzed Direct Alkylation of C–H Bonds in Benzamides and Acrylamides with Functionalized Alkyl Halides via Bidentate-Chelation Assistance

(2013) Yoshinori Aihara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nickel-Catalyzed Direct Arylation of C(sp3)–H Bonds in Aliphatic Amides via Bidentate-Chelation Assistance

(2013) Yoshinori Aihara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Unactivated C(sp3)–H Bond Activation and Intramolecular Amination of Carboxamides: A New Approach to β-Lactams

(2013) Wen-Wu Sun et al.   ORGANIC LETTERS

Copper-Promoted Sulfenylation of sp2 C–H Bonds

(2012) Ly Dieu Tran et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Unexpected Electrophilic Rearrangements of Amides: A Stereoselective Entry to Challenging Substituted Lactones

(2010) Claire Madelaine et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of the Leu–Trp Component of the Celogentin Family of Cyclic Peptides Through a C–H Activation–Cross-Coupling Strategy

(2010) Barbara T. Y. Li et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Auxiliary-Assisted Palladium-Catalyzed Arylation and Alkylation of sp2and sp3Carbon−Hydrogen Bonds

(2010) Dmitry Shabashov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Facile Benzo-Ring Construction via Palladium-Catalyzed Functionalization of Unactivated sp3C−H Bonds under Mild Reaction Conditions

(2010) Yiqing Feng et al.   ORGANIC LETTERS

Total Synthesis of Celogentin C by Stereoselective CH Activation

(2009) Yiqing Feng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pd(II)-Catalyzed Cross-Coupling of sp3C−H Bonds with sp2and sp3Boronic Acids Using Air as the Oxidant

(2008) Dong-Hui Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY