Metal-Free Direct C-H Thiolation and Thiocyanation of Pyrazolones

Ligand-Promoted RhIII -Catalyzed Thiolation of Benzamides with a Broad Disulfide Scope

(2019) Yan-Shang Kang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Regioselective Direct C-H Thiolation and Thiocyanation of Uracils

(2019) Medena Noikham et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Ruthenium(II)-Catalyzed Oxidative Double C–H Activation and Annulation Reaction: Synthesis of Indolo[2,1-a]isoquinolines

(2019) Somadrita Borthakur et al.   ORGANIC LETTERS

The application of sulfur-containing peptides in drug discovery

(2018) Jiaoyan Zhao et al.   CHINESE CHEMICAL LETTERS

Direct Photocatalytic S–H Bond Cyanation with Green “CN” Source

(2018) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

DABCO-catalyzed silver-promoted direct thiolation of pyrazolones with diaryl disulfides

(2018) Akkharaphong Thupyai et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Persulfate-promoted oxidative C–N bond coupling of quinoxalinones and NH-sulfoximines

(2018) Ladawan Sumunnee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Gold(i)- and rhodium(iii)-catalyzed formal regiodivergent C–H alkynylation of 1-arylpyrazolones

(2018) Xueli Wang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Iodine-Catalyzed Oxidative Cross-Dehydrogenative Coupling of Quinoxalinones and Indoles: Synthesis of 3-(Indol-2-yl)quinoxalin-2-one under Mild and Ambient Conditions

(2018) Sirilata Yotphan et al.   SYNTHESIS-STUTTGART

Cu-catalyzed direct C-H thiolation of electron-rich arenes with arylsulfonyl hydrazides

(2018) Lingjuan Chen et al.   TETRAHEDRON

Metal-free direct oxidative C–C bond coupling of pyrazolones and quinoxalinones

(2018) Saowanee Toonchue et al.   Organic Chemistry Frontiers

Copper/Persulfate-Promoted Oxidative Decarboxylative C−H Acylation of Pyrazolones with α-Oxocarboxylic Acids: Direct Access to 4-Acylpyrazolones under Mild Conditions

(2018) Tanakorn Kittikool et al.   ADVANCED SYNTHESIS & CATALYSIS

Pyrazolone: a powerful synthon for asymmetric diverse derivatizations

(2018) Siyuan Liu et al.   CHEMICAL COMMUNICATIONS

Direct Assembly of Polysubstituted Furans via C(sp3)-H Bonds Functionalization Reaction Using Dimethyl Sulfoxide as a Dual Synthon

(2018) Yufeng Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct Oxidative Disulfenylation/Cyclization of 2′-Hydroxyacetophenones with Thiophenols for the Synthesis of 2,2-Dithio-Benzofuran-3(2H )-Ones

(2018) Biao Hu et al.   ADVANCED SYNTHESIS & CATALYSIS

Sodium Salts (NaI/NaBr/NaCl) for the Halogenation of Imidazo-Fused Heterocycles

(2018) Rashmi Semwal et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Oxidative Thioesterification of Methyl Ketones with Thiols/Disulfides for the Synthesis of α-Ketothioesters

(2018) Biao Hu et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine/TBHP-Promoted One-Pot Deoxygenation and Direct 2-Sulfonylation of QuinolineN-Oxides with Sodium Sulfinates: Facile and Regioselective Synthesis of 2-Sulfonylquinolines

(2017) Ladawan Sumunnee et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iodine-Catalyzed Cross Dehydrogenative Coupling Reaction: Sulfenylation of Enaminones Using Dimethyl Sulfoxide as an Oxidant

(2017) Yogesh Siddaraju et al.   JOURNAL OF ORGANIC CHEMISTRY

DMSO-promoted regioselective synthesis of sulfenylated pyrazoles via a radical pathway

(2017) Pengfei Sun et al.   Organic Chemistry Frontiers

Cobalt-Catalyzed C−H Thiolation through Dehydrogenative Cross-Coupling

(2016) Tobias Gensch et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iodine-catalyzed thiolation of electron-rich aromatics using sulfonyl hydrazides as sulfenylation reagents

(2016) Xia Zhao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Recent advances in C–S bond formation via C–H bond functionalization and decarboxylation

(2015) Chao Shen et al.   CHEMICAL SOCIETY REVIEWS

Thiazole: A promising heterocycle for the development of potent CNS active agents

(2015) Chandra Bhushan Mishra et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

(2015) Adile Ayati et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Iodine-Catalyzed Oxidative Amination of Sodium Sulfinates: A Convenient Approach to the Synthesis of Sulfonamides under Mild Conditions

(2015) Chonchanok Buathongjan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Tertiary Amine Pyrazolones and Their Salts as Inhibitors of Mutant Superoxide Dismutase 1-Dependent Protein Aggregation for the Treatment of Amyotrophic Lateral Sclerosis

(2015) Yinan Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Catalyst-Free Regioselective C-3 Thiocyanation of Imidazopyridines

(2015) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine-Catalyzed Oxidative Cross-Coupling of Indoles and Azoles: Regioselective Synthesis of N-Linked 2-(Azol-1-yl)indole Derivatives

(2015) Danupat Beukeaw et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Aryl Sulfides: Metal-Free C–H Sulfenylation of Electron-Rich Arenes

(2015) Thomas Hostier et al.   ORGANIC LETTERS

NaI-Mediated Acetamidosulphenylation of Alkenes with Nitriles as the Nucleophiles: A Direct Access to Acetamidosulfides

(2015) Yang Zheng et al.   ORGANIC LETTERS

Nickel-Catalyzed Direct Thiolation of C(sp3)–H Bonds in Aliphatic Amides

(2015) Xie Wang et al.   ORGANIC LETTERS

Synthesis and cytostatic activity of 7-arylsulfanyl-7-deazapurine bases and ribonucleosides

(2015) Martin Klečka et al.   MedChemComm

Organocatalytic Carbon–Sulfur Bond-Forming Reactions

(2014) Pankaj Chauhan et al.   CHEMICAL REVIEWS

Development of Pyrazolone and Isoxazol-5-one Cambinol Analogues as Sirtuin Inhibitors

(2014) Sumit S. Mahajan et al.   JOURNAL OF MEDICINAL CHEMISTRY

Transition-Metal-Free Acid-Mediated Synthesis of Aryl Sulfides from Thiols and Thioethers

(2014) Anna M. Wagner et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sulfonyl Hydrazides

(2013) Fu-Lai Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An easy direct arylation of 5-pyrazolones

(2013) Hao Gong et al.   Beilstein Journal of Organic Chemistry

Room-Temperature Direct Alkenylation of 5-Pyrazolones

(2013) Yiwen Yang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Direct C–H sulfenylation of purines and deazapurines

(2013) Martin Klečka et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Design of a Potent CB1 Receptor Antagonist Series: Potential Scaffold for Peripherally-Targeted Agents

(2012) Robert L. Dow et al.   ACS Medicinal Chemistry Letters

Antiproliferative activity and QSAR studies of a series of new 4-aminomethylidene derivatives of some pyrazol-5-ones

(2011) Violeta Marković et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Copper-Mediated C–H Activation/C–S Cross-Coupling of Heterocycles with Thiols

(2011) Sadananda Ranjit et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and reactions of some 6-aryl and 2,6-diaryl-4-(4′-antipyrinyl)-2,3,4,5-tetrahydropyridazin-3-ones and screening for their antibacterial activities

(2010) G. H. Sayed et al.   CHINESE JOURNAL OF CHEMISTRY

Design, Synthesis, and Pharmacological Activity of Nonallergenic Pyrazolone-Type Antipyretic Analgesics

(2010) Naoto Uramaru et al.   JOURNAL OF MEDICINAL CHEMISTRY

An Efficient Copper-Catalyzed Carbon−Sulfur Bond Formation Protocol in Water

(2010) Fang Ke et al.   ORGANIC LETTERS

The Novel Antioxidant Edaravone: From Bench to Bedside

(2008) Toshiaki Watanabe et al.   Cardiovascular Therapeutics