Copper-Catalyzed Regioselective Direct C-H Thiolation and Thiocyanation of Uracils

Efficient Buchwald-Hartwig-Migita Cross-Coupling for DNA Thioglycoconjugation

(2018) Nicolas Probst et al.   CHEMISTRY-A EUROPEAN JOURNAL

Direct Photocatalytic S–H Bond Cyanation with Green “CN” Source

(2018) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Sulfenylation, Sulfonylation, and Selenylation of 2,3-Allenoic Acids with Disulfides or Diselenides

(2018) Ya-Xun Xin et al.   JOURNAL OF ORGANIC CHEMISTRY

DABCO-catalyzed silver-promoted direct thiolation of pyrazolones with diaryl disulfides

(2018) Akkharaphong Thupyai et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Persulfate-promoted oxidative C–N bond coupling of quinoxalinones and NH-sulfoximines

(2018) Ladawan Sumunnee et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Iodine-Catalyzed Oxidative Cross-Dehydrogenative Coupling of Quinoxalinones and Indoles: Synthesis of 3-(Indol-2-yl)quinoxalin-2-one under Mild and Ambient Conditions

(2018) Sirilata Yotphan et al.   SYNTHESIS-STUTTGART

Uses of K2S2O8 in Metal-Catalyzed and Metal-Free Oxidative Transformations

(2018) Sudip Mandal et al.   ACS Catalysis

Metal-free direct oxidative C–C bond coupling of pyrazolones and quinoxalinones

(2018) Saowanee Toonchue et al.   Organic Chemistry Frontiers

Copper/Persulfate-Promoted Oxidative Decarboxylative C−H Acylation of Pyrazolones with α-Oxocarboxylic Acids: Direct Access to 4-Acylpyrazolones under Mild Conditions

(2018) Tanakorn Kittikool et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct thiolation of aza-heteroaromatic N-oxides with disulfides via copper-catalyzed regioselective C–H bond activation

(2018) Miao Lai et al.   Organic Chemistry Frontiers

Enantioselective and Regiodivergent Allylation of Pyrimidines with Terminal Allenes: An Approach to Pyrimidine Acyclic Nucleosides

(2018) Lei Liang et al.   Organic Chemistry Frontiers

Cobalt-Catalyzed Direct C–H Thiolation of Aromatic Amides with Disulfides: Application to the Synthesis of Quetiapine

(2018) Mingliang Li et al.   ORGANIC LETTERS

Copper-Catalyzed Aerobic Oxidative Regioselective Thiocyanation of Aromatics and Heteroaromatics

(2017) Huanfeng Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Regio- and Stereoselective C-Nucleoside Synthesis from Unactivated Uracils and Pyranoid Glycals

(2017) Faheem Rasool et al.   ORGANIC LETTERS

Copper-Catalyzed Intermolecular Cyclization between Oximes and Alkenes: A Facile Access to Spiropyrrolines

(2017) Bo Zhao et al.   ACS Catalysis

Expedient C–H Chalcogenation of Indolines and Indoles by Positional-Selective Copper Catalysis

(2017) Parthasarathy Gandeepan et al.   ACS Catalysis

DMSO-promoted regioselective synthesis of sulfenylated pyrazoles via a radical pathway

(2017) Pengfei Sun et al.   Organic Chemistry Frontiers

Synthesis of Thio and Selenoethers of Cyclic β-Hydroxy Carbonyls and Amino Uracils: A Metal-Free Regioselective I2 /DMSO Mediated Reaction

(2017) Asim Jana et al.   ChemistrySelect

Recent advances in the chemistry of organic thiocyanates

(2016) Thomas Castanheiro et al.   CHEMICAL SOCIETY REVIEWS

Sulfur Containing Scaffolds in Drugs: Synthesis and Application in Medicinal Chemistry

(2016) Minghao Feng et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Synthesis of 2-Sulfenylindenones via One-Pot Tandem Meyer–Schuster Rearrangement and Radical Cyclization of Arylpropynols with Disulfides

(2016) Xing-Song Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-mediated arylsulfanylations and arylselanylations of pyrimidine or 7-deazapurine nucleosides and nucleotides

(2016) Filip Botha et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The involvement of the trisulfur radical anion in electron-catalyzed sulfur insertion reactions: facile synthesis of benzothiazine derivatives under transition metal-free conditions

(2016) Zheng-Yang Gu et al.   Chemical Science

Thiazole: A promising heterocycle for the development of potent CNS active agents

(2015) Chandra Bhushan Mishra et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

In search of uracil derivatives as bioactive agents. Uracils and fused uracils: Synthesis, biological activity and applications

(2015) Aleksandra Pałasz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

(2015) Adile Ayati et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Silver-Catalyzed Direct Thiolation of Quinones by Activation of Aryl Disulfides to Synthesize Quinonyl Aryl Thioethers

(2015) Cheng Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Direct Arylation of 5-Halouracils and 5-Halouracil Nucleosides with Arenes and Heteroarenes Promoted by TBAF

(2014) Yong Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Three-Component Coupling Reaction Triggered by Insertion of Arynes into the S═O Bond of DMSO

(2014) Feng-Lei Liu et al.   ORGANIC LETTERS

Switching between Reaction Pathways by an Alcohol Cosolvent Effect: SmI2–Ethylene Glycol vs SmI2–H2O Mediated Synthesis of Uracils

(2014) Michal Szostak et al.   ORGANIC LETTERS

Palladium-catalyzed direct thiolation of ethers with sodium sulfinates

(2014) Shengrong Guo et al.   TETRAHEDRON LETTERS

Dehydrogenative alkenylation of uracils via palladium-catalyzed regioselective C–H activation

(2013) Yi-Yun Yu et al.   CHEMICAL COMMUNICATIONS

Direct C–H sulfenylation of purines and deazapurines

(2013) Martin Klečka et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Postsynthetic on Column RNA Labeling via Stille Coupling

(2012) Lena Wicke et al.   BIOCONJUGATE CHEMISTRY

Regioselective Direct C–H Arylations of Protected Uracils. Synthesis of 5- and 6-Aryluracil Bases

(2011) Miroslava Čerňová et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine mediated an efficient and greener thiocyanation of aminopyrimidines by a modification of the Kaufmann’s reaction

(2011) Ricaurte Rodríguez et al.   TETRAHEDRON LETTERS

Palladium-catalyzed direct 5-arylation of 1,3-dimethyluracil with aryl bromides: an electrophilic metalation–deprotonation with electrophilic arylpalladium intermediate

(2011) Ko Hoon Kim et al.   TETRAHEDRON LETTERS

Pd(II)-Catalyzed Acetoxylation of Uracil via Electrophilic Palladation

(2010) Hyun-Seung Lee et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

An Efficient Copper-Catalyzed Carbon−Sulfur Bond Formation Protocol in Water

(2010) Fang Ke et al.   ORGANIC LETTERS

Enzymology of Purine and Pyrimidine Antimetabolites Used in the Treatment of Cancer

(2009) William B. Parker   CHEMICAL REVIEWS

Novel Cambinol Analogs as Sirtuin Inhibitors: Synthesis, Biological Evaluation, and Rationalization of Activity

(2009) Federico Medda et al.   JOURNAL OF MEDICINAL CHEMISTRY

Aminophenyl- and Nitrophenyl-Labeled Nucleoside Triphosphates: Synthesis, Enzymatic Incorporation, and Electrochemical Detection

(2008) Hana Cahová et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of SodiumR-(+)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl]-1-phenylethylamino}butyrate (Elagolix), a Potent and Orally Available Nonpeptide Antagonist of the Human Gonadotropin-Releasing Hormone Receptor

(2008) Chen Chen et al.   JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed Carbon−Sulfur Cross-Coupling Reactions with Indium Tri(organothiolate) and Its Application to Sequential One-Pot Processes

(2008) Jae-Young Lee et al.   JOURNAL OF ORGANIC CHEMISTRY