Stapling peptides using cysteine crosslinking

Chemical Protein Modification through Cysteine

(2016) Smita B. Gunnoo et al.   CHEMBIOCHEM

Hydrocarbon Stapled Peptides as Modulators of Biological Function

(2015) Philipp M. Cromm et al.   ACS Chemical Biology

A Thiol-Ene Coupling Approach to Native Peptide Stapling and Macrocyclization

(2015) Yuanxiang Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Acetone-Linked Peptides: A Convergent Approach for Peptide Macrocyclization and Labeling

(2015) Naila Assem et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Peptide stapling techniques based on different macrocyclisation chemistries

(2015) Yu Heng Lau et al.   CHEMICAL SOCIETY REVIEWS

Peptide/Protein Stapling and Unstapling: Introduction of s-Tetrazine, Photochemical Release, and Regeneration of the Peptide/Protein

(2015) Stephen P. Brown et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organometallic palladium reagents for cysteine bioconjugation

(2015) Ekaterina V. Vinogradova et al.   NATURE

An enhanced functional interrogation/manipulation of intracellular signaling pathways with the peptide ‘stapling’ technology

(2015) Y He et al.   ONCOGENE

Stapling monomeric GCN4 peptides allows for DNA binding and enhanced cellular uptake

(2015) Abhishek Iyer et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Peptide Ligands Stabilized by Small Molecules

(2014) Shiyu Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Constraining Cyclic Peptides To Mimic Protein Structure Motifs

(2014) Timothy A. Hill et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design of antiviral stapled peptides containing a biphenyl cross-linker

(2014) Avinash Muppidi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Peptides-Staple Method Development and Its Application in Cancer Therapy

(2014) Q.Z. Zhang et al.   CURRENT MEDICINAL CHEMISTRY

Hydrocarbon-Stapled Peptides: Principles, Practice, and Progress

(2014) Loren D. Walensky et al.   JOURNAL OF MEDICINAL CHEMISTRY

Phage Selection of Photoswitchable Peptide Ligands

(2014) Silvia Bellotto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of cell-permeable stapled BH3 peptide-based Mcl-1 inhibitors containing simple aryl and vinylaryl cross-linkers

(2014) Avinash Muppidi et al.   TETRAHEDRON

Light-Regulated Stapled Peptides to Inhibit Protein-Protein Interactions Involved in Clathrin-Mediated Endocytosis

(2013) Laura Nevola et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cover Picture: Recoding the Genetic Code with Selenocysteine (Angew. Chem. Int. Ed. 1/2014)

(2013) Markus J. Bröcker et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Perfluoroaryl-Cysteine SNAr Chemistry Approach to Unprotected Peptide Stapling

(2013) Alexander M. Spokoyny et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Convergent diversity-oriented side-chain macrocyclization scan for unprotected polypeptides

(2013) Yekui Zou et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Nonequilibrium dynamics of helix reorganization observed by transient 2D IR spectroscopy

(2013) M. J. Tucker et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Bicyclic Peptide Inhibitor Reveals Large Contact Interface with a Protease Target

(2012) Alessandro Angelini et al.   ACS Chemical Biology

In Vitro Selection of Highly Modified Cyclic Peptides That Act as Tight Binding Inhibitors

(2012) Yollete V. Guillen Schlippe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rational Design of Proteolytically Stable, Cell-Permeable Peptide-Based Selective Mcl-1 Inhibitors

(2012) Avinash Muppidi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Development of α-Helical Calpain Probes by Mimicking a Natural Protein–Protein Interaction

(2012) Hyunil Jo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Water-Soluble Scaffolds for Peptide Cyclization, Labeling, and Ligation

(2012) Linde E. J. Smeenk et al.   ORGANIC LETTERS

Synthesis and Activity of Thioether-Containing Analogues of the Complement Inhibitor Compstatin

(2011) Patrick J. Knerr et al.   ACS Chemical Biology

Achieving cell penetration with distance-matching cysteine cross-linkers: a facile route to cell-permeable peptide dual inhibitors of Mdm2/Mdmx

(2011) Avinash Muppidi et al.   CHEMICAL COMMUNICATIONS

α-Conotoxin ImI Incorporating Stable Cystathionine Bridges Maintains Full Potency and Identical Three-Dimensional Structure

(2011) Zoltan Dekan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Photocontrollable Peptide-Based Switches Target the Anti-Apoptotic Protein Bcl-xL

(2008) Sabine Kneissl et al.   CHEMBIOCHEM