Stapling monomeric GCN4 peptides allows for DNA binding and enhanced cellular uptake

Peptidosteroid Tweezers Revisited: DNA Binding Through an Optimised Design

(2014) Lieselot L. G. Carrette et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Hydrocarbon-Stapled Peptides: Principles, Practice, and Progress

(2014) Loren D. Walensky et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cell-Permeable Stapled Peptides Based on HIV-1 Integrase Inhibitors Derived from HIV-1 Gene Products

(2013) Wataru Nomura et al.   ACS Chemical Biology

Stimuli-responsive selection of target DNA sequences by synthetic bZIP peptides

(2013) Jesús Mosquera et al.   Nature Communications

Stapled Peptides with Improved Potency and Specificity That Activate p53

(2012) Christopher J. Brown et al.   ACS Chemical Biology

Temporary Electrostatic Impairment of DNA Recognition: Light-Driven DNA Binding of Peptide Dimers

(2012) Adrián Jiménez-Balsa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Development of α-Helical Calpain Probes by Mimicking a Natural Protein–Protein Interaction

(2012) Hyunil Jo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of cell-permeable stapled peptide dual inhibitors of the p53-Mdm2/Mdmx interactions via photoinduced cycloaddition

(2011) Michael M. Madden et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

DNA Recognition by Synthetic Constructs

(2011) Elena Pazos et al.   CHEMBIOCHEM

Achieving cell penetration with distance-matching cysteine cross-linkers: a facile route to cell-permeable peptide dual inhibitors of Mdm2/Mdmx

(2011) Avinash Muppidi et al.   CHEMICAL COMMUNICATIONS

Stapling of a 310-Helix with Click Chemistry

(2011) Øyvind Jacobsen et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of all-hydrocarbon stapled α-helical peptides by ring-closing olefin metathesis

(2011) Young-Woo Kim et al.   Nature Protocols

Enantioselective epoxidation of α,β-unsaturated ketones catalyzed by stapled helical l-Leu-based peptides

(2011) Yosuke Demizu et al.   TETRAHEDRON

Front cover

(2010)   CHEMICAL COMMUNICATIONS

Contemporary strategies for the stabilization of peptides in the α-helical conformation

(2008) Laura K Henchey et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

A Cell-penetrating Helical Peptide as a Potential HIV-1 Inhibitor

(2008) Hongtao Zhang et al.   JOURNAL OF MOLECULAR BIOLOGY