Transition‐Metal‐Free Three‐Component Synthesis of Tertiary Aryl Amines from Nitro Compounds, Boronic Acids, and Trialkyl Phosphites

PEt3-mediated deoxygenative C –N coupling of nitroarenes and boronic acids

(2019) Trevor V. Nykaza et al.   TETRAHEDRON

Pinacol-Derived Chlorohydrosilane in Metal-Free Reductive Amination for the Preparation of Tertiary Alkylphenolmethyl Amines

(2019) Benedicta Assoah et al.   ORGANIC LETTERS

Iridium-Catalyzed Alkylation of Amine and Nitrobenzene with Alcohol to Tertiary Amine under Base- and Solvent-Free Conditions

(2019) Chao Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalyst Free Reductive Coupling of Aromatic and Aliphatic Nitro Compounds with Organohalides

(2019) Marian Rauser et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tandem N,N-Dialkylation Reaction of N-Trimethylsilyl α-Iminoesters Utilizing an Umpolung Reaction and Characteristics of the Silyl Substituent: Synthesis of Pyrrolidine, Piperidine, and Iminodiacetate

(2019) Isao Mizota et al.   ORGANIC LETTERS

Sustainable Amine Synthesis: Iron Catalyzed Reactions of Hydrosilanes with Imines, Amides, Nitroarenes and Nitriles

(2019) Nadim S. Shaikh   ChemistrySelect

Palladium-catalyzed oxidative allylation of bis[(pinacolato)boryl]methane: synthesis of homoallylic boronic esters

(2018) Chunsheng Li et al.   CHEMICAL COMMUNICATIONS

Direct Reductive N -Functionalization of Aliphatic Nitro Compounds

(2018) Marian Rauser et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organic synthesis provides opportunities to transform drug discovery

(2018) David C. Blakemore et al.   Nature Chemistry

Synthesis of Di(hetero)arylamines from Nitrosoarenes and Boronic Acids: A General, Mild, and Transition-Metal-Free Coupling

(2018) Silvia Roscales et al.   ORGANIC LETTERS

Remote sp 3 C–H Amination of Alkenes with Nitroarenes

(2018) Jichao Xiao et al.   Chem

Molybdenum-Catalyzed Sustainable Friedländer Synthesis of Quinolines

(2018) Rubén Rubio-Presa et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Carbonylative Synthesis of α,β-Unsaturated Amides from Styrenes and Nitroarenes

(2018) Jin-Bao Peng et al.   ORGANIC LETTERS

Reductive Molybdenum-Catalyzed Direct Amination of Boronic Acids with Nitro Compounds

(2018) Samuel Suárez-Pantiga et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Intermolecular Reductive C–N Cross Coupling of Nitroarenes and Boronic Acids by PIII/PV═O Catalysis

(2018) Trevor V. Nykaza et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Development of (4-Cyanophenyl)glycine Derivatives as Reversible Inhibitors of Lysine Specific Demethylase 1

(2017) Daniel P. Mould et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Biphilic Phosphetane Catalyzes N–N Bond-Forming Cadogan Heterocyclization via PIII/PV═O Redox Cycling

(2017) Trevor V. Nykaza et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Molybdenum-Catalyzed Synthesis of Nitrogenated Polyheterocycles from Nitroarenes and Glycols with Reuse of Waste Reduction Byproduct

(2017) Rubén Rubio-Presa et al.   ORGANIC LETTERS

PLK1-Targeted Fluorescent Tumor Imaging with High Signal-to-Background Ratio

(2017) Ji-Ting Hou et al.   ACS Sensors

Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions

(2016) Paula Ruiz-Castillo et al.   CHEMICAL REVIEWS

Amine-bis(phenolate) Iron(III)-Catalyzed Formal Hydroamination of Olefins

(2016) Kailong Zhu et al.   Chemistry-An Asian Journal

Chan–Evans–Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem

(2016) Julien C. Vantourout et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemoselective nitro reduction and hydroamination using a single iron catalyst

(2016) Kailong Zhu et al.   Chemical Science

Amine synthesis via iron-catalysed reductive coupling of nitroarenes with alkyl halides

(2016) Chi Wai Cheung et al.   Nature Communications

Hydroaminations of Alkenes: A Radical, Revised, and Expanded Version

(2015) Matteo Villa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Boron-Catalyzed N-Alkylation of Amines using Carboxylic Acids

(2015) Ming-Chen Fu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Electrophilic Amination: The Case of Nitrenoids

(2015) Pavel Starkov et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Advances in Reductive Amination Catalysis and Its Applications

(2015) Heshmatollah Alinezhad et al.   CURRENT ORGANIC CHEMISTRY

Chemoselective Reductive Amination of Carbonyl Compounds for the Synthesis of Tertiary Amines Using SnCl2·2H2O/PMHS/MeOH

(2015) Onkar S. Nayal et al.   JOURNAL OF ORGANIC CHEMISTRY

Buchwald–Hartwig Amination of (Hetero)Aryl Tosylates Using a Well-Defined N-Heterocyclic Carbene/Palladium(II) Precatalyst

(2015) Yin Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-Catalyzed Regio- and Enantioselective Aminolysis of 3,4-Epoxy Alcohols

(2015) Chuan Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Streamlining amine synthesis

(2015) L. Kurti   SCIENCE

Practical olefin hydroamination with nitroarenes

(2015) J. Gui et al.   SCIENCE

Tungsten-Catalyzed Regio- and Enantioselective Aminolysis oftrans-2,3-Epoxy Alcohols: An Entry to Virtually Enantiopure Amino Alcohols

(2014) Chuan Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rapid Synthesis of Fused N-Heterocycles by Transition-Metal-Free Electrophilic Amination of Arene CH Bonds

(2014) Hongyin Gao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

Ruthenium-Catalyzed N-Alkylation of Amines with Alcohols under Mild Conditions Using the Borrowing Hydrogen Methodology

(2014) Arrey B. Enyong et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoredox α-Vinylation of α-Amino Acids and N-Aryl Amines

(2014) Adam Noble et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Olefin Hydroamination with Aminium Radical Cations: A Photoredox Method for Direct C–N Bond Formation

(2014) Andrew J. Musacchio et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent Advances in Electrophilic Amination Reactions

(2014) Corinne Gosmini et al.   SYNTHESIS-STUTTGART

Asymmetric ring-opening of oxabenzonorbornadiene with amines promoted by a chiral iridium-monophosphine catalyst

(2013) Renshi Luo et al.   CHEMICAL COMMUNICATIONS

C–N bond forming cross-coupling reactions: an overview

(2013) Jitender Bariwal et al.   CHEMICAL SOCIETY REVIEWS

Arylamine organic dyes for dye-sensitized solar cells

(2013) Mao Liang et al.   CHEMICAL SOCIETY REVIEWS

Copper-Catalyzed N- and O-Alkylation of Amines and Phenols using Alkylborane Reagents

(2013) Shunsuke Sueki et al.   ORGANIC LETTERS

A New Strategy for the Construction of α-Amino Acid Esters via Decarboxylation

(2013) Jie Zhang et al.   ORGANIC LETTERS

N-Methylation of Peptides and Proteins: An Important Element for Modulating Biological Functions

(2012) Jayanta Chatterjee et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Mediated N-Arylation with Arylboronic Acids: An Avenue to Chan–Lam Coupling

(2012) Dushyant Singh Raghuvanshi et al.   ORGANIC LETTERS

Intermolecular Rhodium-Catalysed Hydroamination of Non-Activated Olefins: Effect of Olefin, Amine, Phosphine and Phosphonium Salt

(2012) Mireia Rodriguez-Zubiri et al.   ChemPlusChem

Semiconducting π-Conjugated Systems in Field-Effect Transistors: A Material Odyssey of Organic Electronics

(2011) Chengliang Wang et al.   CHEMICAL REVIEWS

The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates

(2011) Stephen D. Roughley et al.   JOURNAL OF MEDICINAL CHEMISTRY

Dialkylbiaryl phosphines in Pd-catalyzed amination: a user's guide

(2010) David S. Surry et al.   Chemical Science

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions

(2009) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Progress in Three-Component Reactions. An Update

(2009) M. Syamala   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL