Design, Synthesis, In Vitro Evaluation and Docking Studies of Pyrazole-Thiazole Hybrids as Antimicrobial and Antibiofilm Agents

Synthesis, Anticholinesterase, Antioxidant, and Anti-Aflatoxigenic Activity of Novel Coumarin Carbamate Derivatives

(2018) Belma Zengin Kurt et al.   ChemistrySelect

Synthesis and Characterization of Chalcone-Pyridinium Hybrids as Potential Anti-Cancer and Anti-Microbial Agents

(2018) Ramesh Gondru et al.   ChemistrySelect

Pyrazole derived ultra-short antimicrobial peptidomimetics with potent anti-biofilm activity

(2017) Mija Ahn et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and docking study of novel coumarin ligands as potential selective acetylcholinesterase inhibitors

(2017) Fatih Sonmez et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors

(2017) Belma Zengin Kurt et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Thiazole: A Review on Chemistry, Synthesis and Therapeutic Importance of its Derivatives

(2016) Mahesh T. Chhabria et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Synthesis, antimicrobial activity and advances in structure-activity relationships (SARs) of novel tri-substituted thiazole derivatives

(2016) Guda Mallikarjuna Reddy et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of ( Z )-1-(1,3-diphenyl-1 H -pyrazol-4-yl)-3-(phenylamino)prop-2-en-1-one derivatives as potential anticancer and apoptosis inducing agents

(2016) T. Srinivasa Reddy et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The therapeutic voyage of pyrazole and its analogs: A review

(2016) Mohemmed Faraz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors

(2016) Marina Gjorgjieva et al.   JOURNAL OF MEDICINAL CHEMISTRY

Hybrid Bioactive Heterocycles as Potential Antimicrobial Agents: A Review

(2016) Nisheeth Desai et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

A Green Ultrasound Synthesis, Characterization and Antibacterial Evaluation of 1,4-Disubstituted 1,2,3-Triazoles Tethering Bioactive Benzothiazole Nucleus

(2016) Nadjet Rezki   MOLECULES

Biofilms: an emergent form of bacterial life

(2016) Hans-Curt Flemming et al.   NATURE REVIEWS MICROBIOLOGY

In vitro inhibition effects on erythrocyte carbonic anhydrase I and II and structure-activity relationships of cumarylthiazole derivatives

(2016) Belma Z. Kurt et al.   RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY

Synthesis of novel ( E )- N ′-(2-chloropyrimidin-4-yl)- N -(5-cyano-2-hydroxy-6-phenylpyrimidin-4-yl) formamidine derivatives and their antimicrobial activity

(2016) C. Mallikarjunaswamy et al.   Journal of Saudi Chemical Society

Candida albicansBiofilms and Human Disease

(2015) Clarissa J. Nobile et al.   Annual Review of Microbiology

One-pot multicomponent synthesis of indole incorporated thiazolylcoumarins and their antibacterial, anticancer and DNA cleavage studies

(2015) Rajitha Gali et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, biological activity evaluation and molecular docking studies of novel coumarin substituted thiazolyl-3-aryl-pyrazole-4-carbaldehydes

(2015) Krishnaiah Vaarla et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, antioxidant and anticholinesterase activities of novel coumarylthiazole derivatives

(2015) Belma Zengin Kurt et al.   BIOORGANIC CHEMISTRY

Synthesis, antimicrobial, antiquorum-sensing and cytotoxic activities of new series of benzothiazole derivatives

(2015) Moustafa T. Gabr et al.   CHINESE CHEMICAL LETTERS

A comprehensive review in current developments of benzothiazole-based molecules in medicinal chemistry

(2015) Rangappa S. Keri et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimicrobial activity of novel structural hybrids of benzofuroxan and benzothiazole derivatives

(2015) Elena Chugunova et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Potential of aryl–urea–benzofuranylthiazoles hybrids as multitasking agents in Alzheimer's disease

(2015) Belma Zengin Kurt et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

(2015) Adile Ayati et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Designing, synthesis of selective and high-affinity chalcone-benzothiazole hybrids as Brugia malayi thymidylate kinase inhibitors: In vitro validation and docking studies

(2015) Koneni V. Sashidhara et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Therapeutic potential of benzothiazoles: a patent review (2010 – 2014)

(2015) Ahmed Kamal et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

New Synthesis and Biological Evaluation of Benzothiazole Derivates as Antifungal Agents

(2015) Natividad Herrera Cano et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Synthesis, antioxidant and carbonic anhydrase I and II inhibitory activities of novel sulphonamide-substituted coumarylthiazole derivatives

(2015) Belma Zengin Kurt et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Efficient ultrasound-assisted synthesis, spectroscopic, crystallographic and biological investigations of pyrazole-appended quinolinyl chalcones

(2015) R. Prasath et al.   JOURNAL OF MOLECULAR STRUCTURE

Coumarin heterocyclic derivatives: chemical synthesis and biological activity

(2015) Fernanda G. Medina et al.   NATURAL PRODUCT REPORTS

Regioselective synthesis, antimicrobial evaluation and theoretical studies of 2-styryl quinolines

(2015) Ahmed Kamal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rational approaches, design strategies, structure activity relationship and mechanistic insights for anticancer hybrids

(2014) Kunal Nepali et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent Advances in the Synthesis of Coumarin Derivatives via Knoevenagel Condensation: A Review

(2014) Rajesh H. Vekariya et al.   SYNTHETIC COMMUNICATIONS

Synthesis, characterization and biological evaluation of fused thiazolo[3,2-a]pyrimidine derivatives

(2014) Janardhan Banothu et al.   RSC Advances

Synthesis and biological evaluation of novel formyl-pyrazoles bearing coumarin moiety as potent antimicrobial and antioxidant agents

(2013) Nagamallu Renuka et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Accelerating resistance, inadequate antibacterial drug pipelines and international responses

(2012) Ursula Theuretzbacher   INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS

Indole-Based Fibrates as Potential Hypolipidemic and Antiobesity Agents

(2012) Koneni V. Sashidhara et al.   JOURNAL OF MEDICINAL CHEMISTRY

Candida biofilms associated with CVC and medical devices

(2012) Jyotsna Chandra et al.   MYCOSES

From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles

(2011) Santos Fustero et al.   CHEMICAL REVIEWS

Synthesis, characterization and anti-microbial studies of some novel 2,4-disubstituted thiazoles

(2010) A.M. Vijesh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Promise and challenges in drug discovery and development of hybrid anticancer drugs

(2009) Lalji K Gediya et al.   Expert Opinion on Drug Discovery