Bromide-catalyzed electrochemical trifluoromethylation/cyclization of N-arylacrylamides with low catalyst loading

Copper-Mediated Di- and Monofluoromethanesulfonylation of Arenediazonium Tetrafluoroborates: Probing the Fluorine Effect

(2018) Bo Xing et al.   CHINESE JOURNAL OF CHEMISTRY

Design, synthesis and biological evaluation of 1, 4-dihydro indeno[1,2- c ] pyrazole linked oxindole analogues as potential anticancer agents targeting tubulin and inducing p53 dependent apoptosis

(2018) Irfan Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Nucleophilic difluoromethylation of aromatic aldehydes using trimethyl(trifluoromethyl)silane (TMSCF 3 )

(2018) Sankarganesh Krishnamoorthy et al.   JOURNAL OF FLUORINE CHEMISTRY

Electrochemical Formation of N-Acyloxy Amidyl Radicals and Their Application: Regioselective Intramolecular Amination of sp2 and sp3 C–H Bonds

(2018) Sheng Zhang et al.   ORGANIC LETTERS

Nickel-catalyzed C H trifluoromethylation of pyridine N -oxides with Togni’s reagent

(2018) Xianying Gao et al.   TETRAHEDRON LETTERS

Selective remote C–H trifluoromethylation of aminoquinolines with CF3SO2Na under visible light irradiation in the absence of an external photocatalyst

(2018) Lulu Zhao et al.   Organic Chemistry Frontiers

Synthesis of Spiro[pyrazolin-3,3′-oxindoles] and 3-Arylcarbonylmethyl Substituted Ylideneoxindoles by 1,3-Dipolar Cycloadditions of 3-Ylideneoxindoles and In-Situ-Generated α-Diazoketones

(2017) Shan Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(I)-Catalyzed Interrupted Click Reaction with TMSCF3: Synthesis of 5-Trifluoromethyl 1,2,3-Triazoles

(2017) Kelvin Pak Shing Cheung et al.   ORGANIC LETTERS

1-Trifluoromethylisoquinolines from α-Benzylated Tosylmethyl Isocyanide Derivatives in a Modular Approach

(2017) Lin Wang et al.   ORGANIC LETTERS

Asymmetric Synthesis of α-Fluoro-β-Amino-oxindoles with Tetrasubstituted C–F Stereogenic Centers via Cooperative Cation-Binding Catalysis

(2017) Sushovan Paladhi et al.   ORGANIC LETTERS

Electrocatalytic Minisci Acylation Reaction of N-Heteroarenes Mediated by NH4I

(2017) Qing-Qing Wang et al.   ORGANIC LETTERS

Benzylic C–H Trifluoromethylation via Photoenol

(2017) Takafumi Ide et al.   ORGANIC LETTERS

Transition-metal-free direct trifluoromethylthiolation of electron-rich aromatics using CF 3 SO 2 Na in the presence of PhPCl 2

(2017) Xia Zhao et al.   TETRAHEDRON

Visible-light-induced oxidant and metal-free dehydrogenative cascade trifluoromethylation and oxidation of 1,6-enynes with water

(2017) Sadhan Jana et al.   Chemical Science

Silver-mediated fluorination of alkyl iodides with TMSCF3 as the fluorinating agent

(2017) Liyan Wang et al.   Organic Chemistry Frontiers

Free Radical Chemistry Enabled by Visible Light-Induced Electron Transfer

(2016) Daryl Staveness et al.   ACCOUNTS OF CHEMICAL RESEARCH

Practical Photocatalytic Trifluoromethylation and Hydrotrifluoromethylation of Styrenes in Batch and Flow

(2016) Natan J. W. Straathof et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Direct Difluoromethylenation of Carbonyl Compounds by Using TMSCF3: The Right Conditions

(2016) Sankarganesh Krishnamoorthy et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Electrochemically catalyzed amino-oxygenation of styrenes: n-Bu4NI induced C–N followed by a C–O bond formation cascade for the synthesis of indolines

(2016) Sen Liang et al.   GREEN CHEMISTRY

Electrochemical C–H functionalization and subsequent C–S and C–N bond formation: paired electrosynthesis of 3-amino-2-thiocyanato-α,β-unsaturated carbonyl derivatives mediated by bromide ions

(2016) Li-Shuo Kang et al.   GREEN CHEMISTRY

Electrochemically initiated formation of sulfonyl radicals: synthesis of oxindoles via difunctionalization of acrylamides mediated by bromide ion

(2016) Yang-Ye Jiang et al.   GREEN CHEMISTRY

Unexpected, Latent Radical Reaction of Methane Propagated by Trifluoromethyl Radicals

(2016) Nima Zargari et al.   JOURNAL OF ORGANIC CHEMISTRY

Electrochemically Oxidative α-C–H Functionalization of Ketones: A Cascade Synthesis of α-Amino Ketones Mediated by NH4I

(2016) Sen Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Principles and Applications of Photoredox Catalysis:Trifluoromethylation and Beyond

(2016) Munetaka Akita et al.   JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN

Iodine-mediated regioselective synthesis of vinyl triflones from styrenes with CF3SO2Na

(2016) Li-Na Hua et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Recent advances in photoinduced trifluoromethylation and difluoroalkylation

(2016) Xiaolin Pan et al.   Organic Chemistry Frontiers

Introduction: Fluorine Chemistry

(2015) Veronique Gouverneur et al.   CHEMICAL REVIEWS

Carbon Trifluoromethylation Reactions of Hydrocarbon Derivatives and Heteroarenes

(2015) Concepción Alonso et al.   CHEMICAL REVIEWS

Recent Developments in the Trifluoromethylation of Alkynes

(2015) Pin Gao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Sunlight-driven trifluoromethylation of olefinic substrates by photoredox catalysis: A green organic process

(2015) Munetaka Akita et al.   COMPTES RENDUS CHIMIE

Molecular diversity of spirooxindoles. Synthesis and biological activity

(2015) Tetyana L. Pavlovska et al.   MOLECULAR DIVERSITY

NMP and O2 as Radical Initiator: Trifluoromethylation of Alkenes to Tertiary β-Trifluoromethyl Alcohols at Room Temperature

(2015) Chao Liu et al.   ORGANIC LETTERS

Radical CH Functionalization of Heteroarenes under Electrochemical Control

(2014) Alexander G. O'Brien et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Electrophilic Trifluoromethylation by Use of Hypervalent Iodine Reagents

(2014) Julie Charpentier et al.   CHEMICAL REVIEWS

Redox catalysis in organic electrosynthesis: basic principles and recent developments

(2014) Robert Francke et al.   CHEMICAL SOCIETY REVIEWS

Catalyst-free direct arylsulfonylation of N-arylacrylamides with sulfinic acids: a convenient and efficient route to sulfonated oxindoles

(2014) Wei Wei et al.   GREEN CHEMISTRY

Copper-Catalyzed Intermolecular Trifluoromethylarylation of Alkenes: Mutual Activation of Arylboronic Acid and CF3+ Reagent

(2014) Fei Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Trifluoromethylation by Visible-Light-Driven Photoredox Catalysis

(2014) Takashi Koike et al.   TOPICS IN CATALYSIS

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

Synthesis of Sulfonated Oxindoles by Potassium Iodide Catalyzed Arylsulfonylation of Activated Alkenes with Sulfonylhydrazides in Water

(2013) Xiaoqing Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of α-CF3-Substituted Carbonyl Compounds with Relative and Absolute Stereocontrol Using Electrophilic CF3-Transfer Reagents

(2011) Václav Matoušek et al.   ORGANIC LETTERS

A High-Speed Passive-Matrix Electrochromic Display Using a Mesoporous TiO2 Electrode with Vertical Porosity

(2010) Wu Weng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selectively Nonselective Kinase Inhibition: Striking the Right Balance

(2009) Richard Morphy   JOURNAL OF MEDICINAL CHEMISTRY

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS