Highly stereoselective one-pot construction of trisubstituted tetrahydro-β-carboline-fused diketopiperazines: a synthetic route towards cialis analogues

Isocyanide-based multicomponent reactions towards cyclic constrained peptidomimetics

(2014) Gijs Koopmanschap et al.   Beilstein Journal of Organic Chemistry

The diketopiperazine-fused tetrahydro-β-carboline scaffold as a model peptidomimetic with an unusual α-turn secondary structure

(2013) Francesco Airaghi et al.   Beilstein Journal of Organic Chemistry

Enantioselective Synthesis and Antimicrobial Activities of Tetrahydro-Β-Carboline Diketopiperazines

(2013) Yangmin Ma et al.   CHIRALITY

Highly Diastereoselective Synthesis of 1-Carbamoyl-4-aminoindoloazepinone Derivatives via the Ugi Reaction

(2013) Mouhamad Jida et al.   ORGANIC LETTERS

Ugi Four-Component Reaction with Tandem Deprotection, Cyclization and Pictet-Spengler Reaction: A Concise Route to N-Fused Polycyclic Indoledi­ketopiperazine Alkaloid Analogues

(2013) Prem Chauhan et al.   SYNLETT

Ugi/Aldol Sequence: Expeditious Entry to Several Families of Densely Substituted Nitrogen Heterocycles

(2012) Zhigang Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles in Multicomponent Processes (MCPs)

(2012) Morteza Shiri   CHEMICAL REVIEWS

2,5-Diketopiperazines: Synthesis, Reactions, Medicinal Chemistry, and Bioactive Natural Products

(2012) Alan D. Borthwick   CHEMICAL REVIEWS

Chemistry and Biology Of Multicomponent Reactions

(2012) Alexander Dömling et al.   CHEMICAL REVIEWS

Racemic and diastereoselective construction of indole alkaloids under solvent- and catalyst-free microwave-assisted Pictet–Spengler condensation

(2012) Mouhamad Jida et al.   GREEN CHEMISTRY

The Pictet-Spengler Reaction in Nature and in Organic Chemistry

(2011) Joachim Stöckigt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Expedient entry to the piperazinohydroisoquinoline ring system using a sequential Ugi/Pictet–Spengler/reductive methylation reaction protocol

(2011) Ma.-Angeles Cano-Herrera et al.   CHEMICAL COMMUNICATIONS

Drug to Genome to Drug: Discovery of New Antiplasmodial Compounds

(2011) Terence B. Beghyn et al.   JOURNAL OF MEDICINAL CHEMISTRY

A facile and rapid synthesis of N-benzyl-2-substituted piperazines

(2011) Mouhamad Jida et al.   TETRAHEDRON LETTERS

An Efficient and General Method for the Stereodivergent Syntheses of Tadalafil-Like Tetracyclic Compounds

(2010) Sen Xiao et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Marriage of Convenience: Combining the Power of Isocyanide-Based Multicomponent Reactions with the Versatility of (Hetero)norbornene Chemistry

(2010) Andrea Basso et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Solvent-free microwave-assisted Meyers’ lactamization

(2010) Mouhamad Jida et al.   GREEN CHEMISTRY

Synthesis and Molecular Modeling of Novel Tetrahydro-β-carboline Derivatives with Phosphodiesterase 5 Inhibitory and Anticancer Properties

(2010) Heba A. Mohamed et al.   JOURNAL OF MEDICINAL CHEMISTRY

Mechanistic Studies on theCistoTransEpimerization of Trisubstituted 1,2,3,4-Tetrahydro-β-carbolines

(2010) Michael L. Van Linn et al.   JOURNAL OF ORGANIC CHEMISTRY

Polycyclic Compounds by Ugi−Pictet−Spengler Sequence

(2010) Wei Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Piperazine Scaffolds via Isocyanide-Based Multicomponent Reactions

(2010) Alexander Dömling et al.   SYNTHESIS-STUTTGART

Polycyclic indole alkaloid-type compounds by MCR

(2009) Wei Wang et al.   CHEMICAL COMMUNICATIONS

Multiple Multicomponent Macrocyclizations (MiBs): A Strategic Development Toward Macrocycle Diversity

(2009) Ludger A. Wessjohann et al.   CHEMICAL REVIEWS

Coupling Isocyanide-Based Multicomponent Reactions with Aliphatic or Acyl Nucleophilic Substitution Processes

(2009) Luca Banfi et al.   SYNLETT

Syntheses of chiral 1,3-disubstituted tetrahydro-β-carbolines via CIAT process: highly stereoselective Pictet–Spengler reaction of d-tryptophan ester hydrochlorides with various aldehydes

(2009) Sen Xiao et al.   TETRAHEDRON-ASYMMETRY

Palladium-Catalyzed Domino Intramolecular N-Arylation/Intermolecular C−C Bond Formation for the Synthesis of Functionalized Benzodiazepinediones

(2008) Angela Salcedo et al.   ORGANIC LETTERS