- Home
- Publications
- Publication Search
- Publication Details
Title
Pharmacochemistry of the platelet purinergic receptors
Authors
Keywords
-
Journal
Purinergic Signalling
Volume 7, Issue 3, Pages 305-324
Publisher
Springer Nature
Online
2011-02-17
DOI
10.1007/s11302-011-9216-0
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Novel Alexa Fluor-488 labeled antagonist of the A2A adenosine receptor: Application to a fluorescence polarization-based receptor binding assay
- (2010) Miklós Kecskés et al. BIOCHEMICAL PHARMACOLOGY
- Functionalized Congeners of P2Y1Receptor Antagonists: 2-Alkynyl (N)-Methanocarba 2′-Deoxyadenosine 3′,5′-Bisphosphate Analogues and Conjugation to a Polyamidoamine (PAMAM) Dendrimer Carrier
- (2010) Sonia de Castro et al. BIOCONJUGATE CHEMISTRY
- Part II: Piperazinyl-glutamate-pyridines as potent orally bioavailable P2Y12 antagonists for inhibition of platelet aggregation
- (2010) John J. Parlow et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Benzofuran-substituted urea derivatives as novel P2Y1 receptor antagonists
- (2010) Reema K. Thalji et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- New P2Y 12 Inhibitors
- (2010) Marco Cattaneo CIRCULATION
- P2Y nucleotide receptors: promise of therapeutic applications
- (2010) Kenneth A. Jacobson et al. DRUG DISCOVERY TODAY
- Mutational analysis of residues important for ligand interaction with the human P2Y12 receptor
- (2010) Yingying Mao et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- P2X purinergic receptor ligands: recently patented compounds
- (2010) Hendra Gunosewoyo et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- NF449 Is a Novel Inhibitor of Fibroblast Growth Factor Receptor 3 (FGFR3) Signaling Active in Chondrocytes and Multiple Myeloma Cells
- (2010) Pavel Krejci et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Charged residues in the C-terminus of the P2Y1 receptor constitute a basolateral-sorting signal
- (2010) S. C. Wolff et al. JOURNAL OF CELL SCIENCE
- Physiological implications of adenosine receptor-mediated platelet aggregation
- (2010) Hillary A. Johnston-Cox et al. JOURNAL OF CELLULAR PHYSIOLOGY
- 2-MeS-β,γ-CCl2-ATP is a Potent Agent for Reducing Intraocular Pressure†
- (2010) Shay Eliahu et al. JOURNAL OF MEDICINAL CHEMISTRY
- A Novel Insulin Secretagogue Based on a Dinucleoside Polyphosphate Scaffold(1)
- (2010) Shay Eliahu et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structure-Based Discovery of Novel Chemotypes for Adenosine A2AReceptor Antagonists
- (2010) Vsevolod Katritch et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structure-Based Discovery of A2AAdenosine Receptor Ligands
- (2010) Jens Carlsson et al. JOURNAL OF MEDICINAL CHEMISTRY
- Development of Potent and Selective Inhibitors ofecto-5′-Nucleotidase Based on an Anthraquinone Scaffold
- (2010) Younis Baqi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Piperazinyl Glutamate Pyridines as Potent Orally Bioavailable P2Y12Antagonists for Inhibition of Platelet Aggregation
- (2010) John J. Parlow et al. JOURNAL OF MEDICINAL CHEMISTRY
- A new role for the A2b adenosine receptor in regulating platelet function
- (2010) D. YANG et al. JOURNAL OF THROMBOSIS AND HAEMOSTASIS
- Quantification of recombinant and platelet P2Y1 receptors utilizing a [125I]-labeled high-affinity antagonist 2-iodo-N6-methyl-(N)-methanocarba-2′-deoxyadenosine-3′,5′-bisphosphate ([125I]MRS2500)
- (2010) Philippe Ohlmann et al. PHARMACOLOGICAL RESEARCH
- BF0801, a novel adenine derivative, inhibits platelet activation via phosphodiesterase inhibition and P2Y12 antagonism
- (2010) Si Zhang et al. THROMBOSIS AND HAEMOSTASIS
- PEGylated Dendritic Unimolecular Micelles as Versatile Carriers for Ligands of G Protein-Coupled Receptors
- (2009) Yoonkyung Kim et al. BIOCONJUGATE CHEMISTRY
- 6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors
- (2009) Pamela Crepaldi et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Piperazinyl-glutamate-pyridines as potent orally bioavailable P2Y12 antagonists for inhibition of platelet aggregation
- (2009) John J. Parlow et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Ticagrelor: The First Reversibly Binding Oral P2Y12Receptor Antagonist
- (2009) Steen Husted et al. Cardiovascular Therapeutics
- Extracellular NAD+ induces a rise in [Ca2+]i in activated human monocytes via engagement of P2Y1 and P2Y11 receptors
- (2009) Carina Klein et al. CELL CALCIUM
- New P2Y12 antagonists
- (2009) Alan D Michelson CURRENT OPINION IN HEMATOLOGY
- High-Affinity, Non-Nucleotide-Derived Competitive Antagonists of Platelet P2Y12Receptors
- (2009) Younis Baqi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Human P2Y14Receptor Agonists: Truncation of the Hexose Moiety of Uridine-5′-Diphosphoglucose and Its Replacement with Alkyl and Aryl Groups
- (2009) Arijit Das et al. JOURNAL OF MEDICINAL CHEMISTRY
- Contribution of the region Glu181 to Val200 of the extracellular loop of the human P2X1 receptor to agonist binding and gating revealed using cysteine scanning mutagenesis1
- (2009) Jonathan A. Roberts et al. JOURNAL OF NEUROCHEMISTRY
- Interaction of New, Very Potent Non-Nucleotide Antagonists with Arg256 of the Human Platelet P2Y12 Receptor
- (2009) K. Hoffmann et al. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
- Ticagrelor binds to human P2Y12independently from ADP but antagonizes ADP-induced receptor signaling and platelet aggregation
- (2009) J. J. J. VAN GIEZEN et al. JOURNAL OF THROMBOSIS AND HAEMOSTASIS
- Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
- (2009) R. L. Carter et al. MOLECULAR PHARMACOLOGY
- Crystal structure of the ATP-gated P2X4 ion channel in the closed state
- (2009) Toshimitsu Kawate et al. NATURE
- Comparison of ticagrelor and thienopyridine P2Y12 binding characteristics and antithrombotic and bleeding effects in rat and dog models of thrombosis/hemostasis
- (2009) J.J.J. van Giezen et al. THROMBOSIS RESEARCH
- Agonist and antagonist effects of diadenosine tetraphosphate, a platelet dense granule constituent, on platelet P2Y1, P2Y12 and P2X1 receptors
- (2009) Hung Chang et al. THROMBOSIS RESEARCH
- Involvement of basic amino acid residues in transmembrane regions 6 and 7 in agonist and antagonist recognition of the human platelet P2Y12-receptor
- (2008) Kristina Hoffmann et al. BIOCHEMICAL PHARMACOLOGY
- Tetrahydro-4-quinolinamines identified as novel P2Y1 receptor antagonists
- (2008) Ángel I. Morales-Ramos et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- P2Y1 receptor antagonists as novel antithrombotic agents
- (2008) Jeffrey A. Pfefferkorn et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Adenosine Receptor Antagonists: Translating Medicinal Chemistry and Pharmacology into Clinical Utility
- (2008) Pier Giovanni Baraldi et al. CHEMICAL REVIEWS
- Carba-nucleosides as Potent Antagonists of the Adenosine 5′-Diphosphate (ADP) Purinergic Receptor (P2Y12) on Human Platelets
- (2008) Hong Ye et al. ChemMedChem
- Inter-subunit disulfide cross-linking in homomeric and heteromeric P2X receptors
- (2008) Benjamin Marquez-Klaka et al. EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS
- Identification of hydrolytically stable and selective P2Y1 receptor agonists
- (2008) Shay E. Eliahu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Constitutive and Agonist-induced Dimerizations of the P2Y1Receptor
- (2008) Roy C. Y. Choi et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Lipophilic Modifications to Dinucleoside Polyphosphates and Nucleotides that Confer Antagonist Properties at the Platelet P2Y12Receptor
- (2008) James G. Douglass et al. JOURNAL OF MEDICINAL CHEMISTRY
- Rapid resensitization of purinergic receptor function in human platelets
- (2008) S. J. MUNDELL et al. JOURNAL OF THROMBOSIS AND HAEMOSTASIS
- Interaction of the active metabolite of prasugrel, R-138727, with cysteine 97 and cysteine 175 of the human P2Y12receptor
- (2008) I. ALGAIER et al. JOURNAL OF THROMBOSIS AND HAEMOSTASIS
- Acyl derivatives of coenzyme A inhibit platelet function via antagonism at P2Y1and P2Y12receptors: A new finding that may influence the design of anti-thrombotic agents
- (2008) P. Manolopoulos et al. PLATELETS
- The 2.6 Angstrom Crystal Structure of a Human A2A Adenosine Receptor Bound to an Antagonist
- (2008) V.-P. Jaakola et al. SCIENCE
- Novel P2Y12 adenosine diphosphate receptor antagonists for inhibition of platelet aggregation (I): In vitro effects on platelets
- (2008) Judi Bryant et al. THROMBOSIS RESEARCH
- The Adenosine A2b Receptor: Its Role in Inflammation
- (2008) J. Ham et al. Endocrine Metabolic & Immune Disorders-Drug Targets
- Hetero-oligomerization of the P2Y11receptor with the P2Y1receptor controls the internalization and ligand selectivity of the P2Y11receptor
- (2007) Denise Ecke et al. BIOCHEMICAL JOURNAL
- Caged agonist of P2Y1 and P2Y12 receptors for light-directed facilitation of platelet aggregation
- (2007) Zhan-Guo Gao et al. BIOCHEMICAL PHARMACOLOGY
Find the ideal target journal for your manuscript
Explore over 38,000 international journals covering a vast array of academic fields.
SearchBecome a Peeref-certified reviewer
The Peeref Institute provides free reviewer training that teaches the core competencies of the academic peer review process.
Get Started