Tetrazole regioisomers in the development of nitro group-containing antitubercular agents

Towards a new combination therapy for tuberculosis with next generation benzothiazinones

(2014) V. Makarov et al.   EMBO Molecular Medicine

1-Substituted-5-[(3,5-dinitrobenzyl)sulfanyl]-1H-tetrazoles and their isosteric analogs: A new class of selective antitubercular agents active against drug-susceptible and multidrug-resistant mycobacteria

(2014) Galina Karabanovich et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Structure-Activity Relationships of 2-Benzylsulfanylbenzothiazoles: Synthesis and Selective Antimycobacterial Properties

(2014) Vera Klimesova et al.   Medicinal Chemistry

Advances in the development of new tuberculosis drugs and treatment regimens

(2013) Alimuddin Zumla et al.   NATURE REVIEWS DRUG DISCOVERY

One-pot synthesis of 1-substituted-5-alkylselanyl-1 H -tetrazoles from isoselenocyanates: unexpected formation of N -alkyl- N -arylcyanamides and ( Z )- Se -alkyl- N -cyano- N , N′ -diarylisoselenoureas

(2013) Galina Karabanovich et al.   TETRAHEDRON

Synthesis and biological evaluation of new N-acyl-homoserine-lactone analogues, based on triazole and tetrazole scaffolds, acting as LuxR-dependent quorum sensing modulators

(2012) Mohamad Sabbah et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Recent Advances in the Research of Heterocyclic Compounds as Antitubercular Agents

(2012) Mi Yan et al.   ChemMedChem

Synthesis and Functionalization of 5-Substituted Tetrazoles

(2012) Jaroslav Roh et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

New Drugs for the Treatment of Tuberculosis: Needs, Challenges, Promise, and Prospects for the Future

(2012) Christian Lienhardt et al.   JOURNAL OF INFECTIOUS DISEASES

Antituberculosis Drug Research: A Critical Overview

(2012) Beena et al.   MEDICINAL RESEARCH REVIEWS

Delamanid for Multidrug-Resistant Pulmonary Tuberculosis

(2012) Maria Tarcela Gler et al.   NEW ENGLAND JOURNAL OF MEDICINE

Benzothiazinones Are Suicide Inhibitors of Mycobacterial Decaprenylphosphoryl-β-d-ribofuranose 2′-Oxidase DprE1

(2011) Claudia Trefzer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Heme Oxygenase Inhibition by 2-Oxy-substituted 1-Azolyl-4-phenylbutanes: Effect of Variation of the Azole Moiety. X-Ray Crystal Structure of Human Heme Oxygenase-1 in Complex with 4-Phenyl-1-(1H-1,2,4-triazol-1-yl)-2-butanone

(2009) Gheorghe Roman et al.   Chemical Biology & Drug Design

Synthesis of some new 5-substituted 1H-tetrazoles

(2009) A. Dişli et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis

(2009) V. Makarov et al.   SCIENCE

High Content Screening Identifies Decaprenyl-Phosphoribose 2′ Epimerase as a Target for Intracellular Antimycobacterial Inhibitors

(2009) Thierry Christophe et al.   PLoS Pathogens

Optimization of the Central Heterocycle of α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase

(2008) Joie Garfunkle et al.   JOURNAL OF MEDICINAL CHEMISTRY

Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation

(2007) Giorgio Ortar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY