Tandem reactions initiated by copper-catalyzed cross-coupling: A new strategy towards heterocycle synthesis

One-Pot Synthesis of Triazolothiadiazepine 1,1-Dioxide Derivatives via Copper-Catalyzed Tandem [3+2] Cycloaddition/N-Arylation

(2011) Deepak Kumar Barange et al.   ADVANCED SYNTHESIS & CATALYSIS

Cu(I)-Catalyzed Domino Reactions: Efficient and Selective Synthesis of 4H-Chromenes and Naphthalenes

(2011) Chandi C. Malakar et al.   ORGANIC LETTERS

Copper-Catalyzed Domino Synthesis of Quinazolinones via Ullmann-Type Coupling and Aerobic Oxidative C−H Amidation

(2011) Wei Xu et al.   ORGANIC LETTERS

Aqueous C–S cross-coupling: synthesis of 2-iminobenzo-1,3-oxathioles via CuCl2·H2O-catalyzed tandem reaction of 2-iodophenols with isothiocyanates

(2011) Qiuping Ding et al.   TETRAHEDRON LETTERS

Highly Efficient Ligands for the Palladium-Assisted DoubleN-Arylation of Primary Amines for One-Sep Construction of Carbazoles

(2010) Yibo Zhou et al.   ADVANCED SYNTHESIS & CATALYSIS

Efficient Synthesis of 2-Fluoromethylated Quinolines via Copper-Catalyzed Alkynylation and Cyclization of Fluorinated Imidoyl Iodides

(2010) Shan Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed One-Pot Synthesis of Substituted Benzimidazoles

(2010) Hongwei Jin et al.   ADVANCED SYNTHESIS & CATALYSIS

Well-Defined Allylnickel Chloride/N-Heterocyclic Carbene [(NHC)Ni(allyl)Cl] Complexes as Highly Active Precatalysts for CN and CS Cross-Coupling Reactions

(2010) María José Iglesias et al.   ADVANCED SYNTHESIS & CATALYSIS

An Efficient Domino Synthesis of Quinoxalin-2(1H)-ones via an SNAr/Coupling/Demesylation Reaction Catalyzed by Copper(I) as Key Step

(2010) Dingben Chen et al.   ADVANCED SYNTHESIS & CATALYSIS

A Simple Copper-Catalyzed Cascade Synthesis of 2-Amino-1H-indole-3-carboxylate Derivatives

(2010) Xiaobo Yang et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Benzoxazole and Benzimidazole Derivatives via Ligand-Free Copper(I)-Catalyzed Cross-Coupling Reaction of o-Halophenols or o-Haloanilines with Carbodiimides

(2010) Guodong Shen et al.   ADVANCED SYNTHESIS & CATALYSIS

A General and Practical Access to Chiral Quinoxalinones with Low Copper-Catalyst Loading

(2010) Shinji Tanimori et al.   ADVANCED SYNTHESIS & CATALYSIS

Assembly of Substituted Phenothiazines by a Sequentially Controlled CuI/ L-Proline-Catalyzed Cascade CS and CN Bond Formation

(2010) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Domino Condensation/S-Arylation/Heterocyclization Reactions: Copper-Catalyzed Three-Component Synthesis of 2-N-Substituted Benzothiazoles

(2010) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Catalyzed Trifluoromethylation of Aryl Halides

(2010) Rylan J. Lundgren et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Concise copper-catalyzed one-pot tandem synthesis of benzimidazo[1,2-b]isoquinolin-11-one derivatives

(2010) Juyou Lu et al.   CHEMICAL COMMUNICATIONS

C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3CH Activation

(2010) Hana Prokopcová et al.   CHEMISTRY-A EUROPEAN JOURNAL

CuI/L-Proline-Catalyzed Coupling of Substituted 3-Iodoprop-2-en-1-ols with 1-Alkynes and Subsequent Cyclization: A Convenient Approach for Synthesizing Polysubstituted Furans

(2010) You Wang et al.   Chemistry-An Asian Journal

Alumina-Supported Cu(II), A Versatile and Recyclable Catalyst for Regioselective Ring Opening of Aziridines and Epoxides and Subsequent Cyclization to Functionalized 1,4-Benzoxazines and 1,4-Benzodioxanes

(2010) Sukalyan Bhadra et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Annulation of 2-Formylazoles witho-Aminoiodoarenes

(2010) Jonathan T. Reeves et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Cascade Syntheses of 2H-benzo[b][1,4]thiazin-3(4H)-ones and Quinoxalin-2(1H)-ones through Capturing S and N Atom Respectively from AcSH and TsNH2

(2010) Dingben Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Synthesis of Quinazoline Derivatives via Ullmann-Type Coupling and Aerobic Oxidation

(2010) Chen Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Conjugated Diene-Assisted Allylic C−H Bond Activation: Cationic Rh(I)-Catalyzed Syntheses of Polysubstituted Tetrahydropyrroles, Tetrahydrofurans, and Cyclopentanes from Ene-2-Dienes

(2010) Qian Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-catalyzed tandem process: an efficient approach to 2-substituted-1,4-benzodioxanes

(2010) Yunyun Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

One-Pot Synthesis of Pyrimido[1,6-a]indol-1(2H)-one Derivatives by a Nucleophilic Addition/Cu-Catalyzed N-Arylation/Pd-Catalyzed C−H Activation Sequential Process

(2010) Zhi-Jing Wang et al.   ORGANIC LETTERS

Simple and Efficient Copper-Catalyzed Approach to 2,4-Disubstituted Imidazolones

(2010) Xiaoyu Gong et al.   ORGANIC LETTERS

Synthesis of Aza-Fused Polycyclic Quinolines through Copper-Catalyzed Cascade Reactions

(2010) Qian Cai et al.   ORGANIC LETTERS

Domino N−H/C−H Bond Activation: Copper-Catalyzed Synthesis of Nitrogen-Bridgehead Heterocycles Using Azoles and 1,4-Dihalo-1,3-dienes

(2010) Qian Liao et al.   ORGANIC LETTERS

Copper-Catalyzed Tandem Reactions of 1-(2-Iodoary)-2-yn-1-ones with Isocyanides for the Synthesis of 4-Oxo-indeno[1,2-b]pyrroles

(2010) Qian Cai et al.   ORGANIC LETTERS

An efficient synthesis of 6,9-disubstituted purin-8-ones via copper-catalyzed coupling/cyclization

(2010) Qi-Fei Zhong et al.   TETRAHEDRON

Domino synthesis of 2-arylbenzo[b]furans by copper(II)-catalyzed coupling of o-iodophenols and aryl acetylenes

(2010) E.A. Jaseer et al.   TETRAHEDRON

Assembly of N-substituted pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones via copper catalyzed aryl amination

(2010) Xu Lu et al.   TETRAHEDRON

One-pot synthesis of substituted indolines via a copper-catalyzed sequential multicomponent/C–N coupling reaction

(2010) Hongwei Jin et al.   TETRAHEDRON

A ligand-free, copper-catalyzed cascade sequence to indole-2-carboxylic esters

(2010) Stefan G. Koenig et al.   TETRAHEDRON LETTERS

Copper-Catalyzed Synthesis of 1,2,4-Benzothiadiazine 1,1-Dioxide Derivatives by Coupling of 2-Halobenzenesulfonamides with Amidines

(2009) Daoshan Yang et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-CatalyzedN-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore

(2009) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

Efficient and Economical Access to Substituted Benzothiazoles: Copper-Catalyzed Coupling of 2-Haloanilides with Metal Sulfides and Subsequent Condensation

(2009) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Meta-Selective Transition-Metal Catalyzed Arene CH Bond Functionalization

(2009) Yang Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Copper-Catalyzed Tandem Synthesis of Indolo- and Pyrrolo[2,1-a]isoquinolines

(2009) Akhilesh Kumar Verma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions

(2009) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Domino Direct Arylation/N-Arylation: Convenient Synthesis of Phenanthridines

(2009) David A. Candito et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-catalyzed cyclization reactions for the synthesis of alkaloids

(2009) Gwilherm Evano et al.   CHEMICAL COMMUNICATIONS

Synthesis of 2-fluoroalkylbenzimidazoles via copper(i)-catalyzed tandem reactions

(2009) Jiangtao Zhu et al.   CHEMICAL COMMUNICATIONS

Assembly of indole-2-carboxylic acid esters through a ligand-free copper-catalysed cascade process

(2009) Qian Cai et al.   CHEMICAL COMMUNICATIONS

Synthesis ofN-Substituted-2-Aminobenzothiazoles by Ligand-Free Copper(I)-Catalyzed Cross-Coupling Reaction of 2-Haloanilines with Isothiocyanates

(2009) Guodong Shen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper(I)-Catalyzed Cascade Synthesis of 2-Substituted 1,3-Benzothiazoles: Direct Access to Benzothiazolones

(2009) Siva Murru et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Reactivity-Controlled Regioselectivity: A Regiospecific Synthesis of 1,2-Disubstituted Benzimidazoles

(2009) Xiaohu Deng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2-Aminobenzothiazole via Copper(I)-Catalyzed Tandem Reaction of 2-Iodobenzenamine with Isothiocyanate

(2009) Qiuping Ding et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Copper(I)-Catalyzed One-Pot Synthesis of 2H-1,4-Benzoxazin-3-(4H)-ones fromo-Halophenols and 2-Chloroacetamides

(2009) Enguang Feng et al.   JOURNAL OF ORGANIC CHEMISTRY

CuI-Catalyzed Amination of Arylhalides with Guanidines or Amidines: A Facile Synthesis of 1-H-2-Substituted Benzimidazoles

(2009) Xiaohu Deng et al.   JOURNAL OF ORGANIC CHEMISTRY

Assembly of Substituted 1H-Benzimidazoles and 1,3-Dihydrobenzimidazol-2-ones via CuI/l-Proline Catalyzed Coupling of Aqueous Ammonia with 2-Iodoacetanilides and 2-Iodophenylcarbamates

(2009) Xiaoqiong Diao et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Cascade Addition/Cyclization: An Efficient and Versatile Synthesis ofN-Substituted 2-Heterobenzimidazoles

(2009) Xin Lv et al.   JOURNAL OF ORGANIC CHEMISTRY

An efficient cascade synthesis of various 2H-1,4-benzoxazin-3-(4H)-ones from o-halophenols and 2-halo-amides catalyzed by CuI

(2009) Dingben Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

An efficient copper-catalyzed synthesis of hexahydro-1H- phenothiazines

(2009) D. J. C. Prasad et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

An Efficient One-Pot Copper-Catalyzed Approach to Isoquinolin-1(2H)-one Derivatives

(2009) Feng Wang et al.   ORGANIC LETTERS

Highly Efficient Copper-Catalyzed Domino Ring Opening and Goldberg Coupling Cyclization for the Synthesis of 3,4-Dihydro-2H-1,4-benzoxazines†

(2009) R. Koteshwar Rao et al.   ORGANIC LETTERS

Assembly of Substituted 3-Methyleneisoindolin-1-ones via a CuI/l-Proline-Catalyzed Domino Reaction Process of 2-Bromobenzamides and Terminal Alkynes

(2009) Li Li et al.   ORGANIC LETTERS

Facile synthesis of 1,4-benzodiazepin-3-ones from o-bromobenzylamines and amino acids via a cascade coupling/condensation process

(2009) Hexiang Wang et al.   TETRAHEDRON

Copper-catalyzed synthesis of five-membered heterocycles via double C–N bond formation: an efficient synthesis of pyrroles, dihydropyrroles, and carbazoles

(2009) Ende Li et al.   TETRAHEDRON

Copper-catalyzed tandem synthesis of [1,2,3]triazolo[5,1-a]isoquinolines and their transformation to 1,3-disubstituted isoquinolines

(2009) Yuan-Yuan Hu et al.   TETRAHEDRON

Synthesis of polysubstituted 1,2-dihydroisoquinolines via a CuI-catalyzed arylation/condensation cascade process

(2009) Yangyang Wu et al.   TETRAHEDRON LETTERS

Copper-catalyzed tandem reactions of 2-halobenzenamines with isothiocyanates under ligand- and base-free conditions

(2009) Yan-Jin Guo et al.   TETRAHEDRON LETTERS

Copper(I)-Catalyzed One-Pot Synthesis of 2-Iminobenzo- 1,3-oxathioles fromortho-Iodophenols and Isothiocyanates

(2008) Xin Lv et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions: Copper Makes a Difference

(2008) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Simple and Efficient Approach to Quinazolinones under Mild Copper-Catalyzed Conditions

(2008) Xiaowei Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly efficient copper-catalyzed cascade synthesis of quinazoline and quinazolinone derivatives

(2008) Cheng Huang et al.   CHEMICAL COMMUNICATIONS

Coinage Metal-Assisted Synthesis of Heterocycles

(2008) Nitin T. Patil et al.   CHEMICAL REVIEWS

Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis

(2008) Gwilherm Evano et al.   CHEMICAL REVIEWS

Palladium and copper-catalysed arylation reactions in the presence of water, with a focus on carbon–heteroatom bond formation

(2008) Mónica Carril et al.   CHEMICAL SOCIETY REVIEWS

Synthesis of 1-Amino-1H-indole-3-carboxylates by Copper(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand Melkonyan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of N-Substituted Indole-3-carboxylic Acid Derivatives via Cu(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand S. Melkonyan et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Synthesis of Benzimidazoles via Cascade Reactions ofo-Haloacetanilide Derivatives with Amidine Hydrochlorides

(2008) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

A One-Pot Coupling/Hydrolysis/Condensation Process to Pyrrolo[1,2-a]quinoxaline

(2008) Qiliang Yuan et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Domino Annulation Approaches to the Synthesis of Benzoxazoles under Microwave-Accelerated and Conventional Thermal Conditions

(2008) Russell D. Viirre et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 6,7,8-Trisubstituted Purines via a Copper-Catalyzed Amidation Reaction

(2008) Nada Ibrahim et al.   JOURNAL OF ORGANIC CHEMISTRY

Elaboration of 2-(Trifluoromethyl)indoles via a Cascade Coupling/Condensation/Deacylation Process

(2008) Yu Chen et al.   ORGANIC LETTERS

Synthesis of Indolines via a Domino Cu-Catalyzed Amidation/Cyclization Reaction

(2008) Ana Minatti et al.   ORGANIC LETTERS

Concise Synthesis of Indole-Fused 1,4-Diazepines through Copper(I)-Catalyzed Domino Three-Component Coupling−Cyclization−N-Arylation under Microwave Irradiation

(2008) Yusuke Ohta et al.   ORGANIC LETTERS

Cu2O-Catalyzed Tandem Ring-Opening/Coupling Cyclization Process for the Synthesis of 2,3-Dihydro-1,4-benzodioxins

(2008) Weiliang Bao et al.   ORGANIC LETTERS

Assembly of Isoquinolines via CuI-Catalyzed Coupling of β-Keto Esters and 2-Halobenzylamines

(2008) Bao Wang et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed Carbon-Carbon Bond Formation via Carbon-Hydrogen Bond Cleavage

(2008) Fumitoshi Kakiuchi et al.   SYNTHESIS-STUTTGART