18F-Labeled Peptides: The Future Is Bright

An Organotrifluoroborate for Broadly Applicable One-Step18F-Labeling

(2014) Zhibo Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and in Vitro and in Vivo Evaluation of SiFA-Tagged Bombesin and RGD Peptides as Tumor Imaging Probes for Positron Emission Tomography

(2014) Simon Lindner et al.   BIOCONJUGATE CHEMISTRY

Fully automated synthesis and coupling of [18F]FBEM to glutathione using the iPHASE FlexLab module

(2014) Uwe Ackermann et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Al18F labeling of peptides and proteins

(2014) Peter Laverman et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Preclinical Evaluation of a High-Affinity 18F-Trifluoroborate Octreotate Derivative for Somatostatin Receptor Imaging

(2014) Z. Liu et al.   JOURNAL OF NUCLEAR MEDICINE

18F-Labeled Silicon-Based Fluoride Acceptors: Potential Opportunities for Novel Positron Emitting Radiopharmaceuticals

(2014) Vadim Bernard-Gauthier et al.   Biomed Research International

The Druggable Genome: Evaluation of Drug Targets in Clinical Trials Suggests Major Shifts in Molecular Class and Indication

(2013) Mathias Rask-Andersen et al.   Annual Review of Pharmacology and Toxicology

Imaging integrin alpha-v-beta-3 expression in tumors with an18F-labeled dimeric RGD peptide

(2013) Ingrid Dijkgraaf et al.   Contrast Media & Molecular Imaging

A Comparative Study of Radiolabeled Bombesin Analogs for the PET Imaging of Prostate Cancer

(2013) Y. Liu et al.   JOURNAL OF NUCLEAR MEDICINE

First Experience of 18F-Alfatide in Lung Cancer Patients Using a New Lyophilized Kit for Rapid Radiofluorination

(2013) W. Wan et al.   JOURNAL OF NUCLEAR MEDICINE

"To Serve and Protect": Enzyme Inhibitors as Radiopeptide Escorts Promote Tumor Targeting

(2013) B. A. Nock et al.   JOURNAL OF NUCLEAR MEDICINE

Application of [18F]FDG in radiolabeling reactions using microfluidic technology

(2013) Vincent R. Bouvet et al.   LAB ON A CHIP

Recent Trends in Bioorthogonal Click-Radiolabeling Reactions Using Fluorine-18

(2013) Marc Pretze et al.   MOLECULES

Using 5-deoxy-5-[18F]fluororibose to glycosylate peptides for positron emission tomography

(2013) Xiang-Guo Li et al.   Nature Protocols

Synthesis and radiopharmacological evaluation of a high-affinity and metabolically stabilized 18F-labeled bombesin analogue for molecular imaging of gastrin-releasing peptide receptor-expressing prostate cancer

(2013) Susan Richter et al.   NUCLEAR MEDICINE AND BIOLOGY

Synthesis and evaluation of an 18F-labelled norbornene derivative for copper-free click chemistry reactions

(2013) James C. Knight et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Microfluidics for Synthesis of Peptide-Based PET Tracers

(2013) Yang Liu et al.   Biomed Research International

Radiofluorination using aluminum-fluoride (Al18F)

(2013) William J McBride et al.   EJNMMI Research

Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase: a comparative study

(2012) Manuela Kuchar et al.   AMINO ACIDS

Optimization of the solid-phase synthesis of [18F] radiolabeled peptides for positron emission tomography

(2012) Jason B. White et al.   APPLIED RADIATION AND ISOTOPES

New Lyophilized Kit for Rapid Radiofluorination of Peptides

(2012) William J. McBride et al.   BIOCONJUGATE CHEMISTRY

Labeling Strategies of Peptides with 18F for Positron Emission Tomography

(2012) D. E. Olberg et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Rationale for the use of radiolabelled peptides in diagnosis and therapy

(2012) K. P. Koopmans et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

PET of Tumors Expressing Gastrin-Releasing Peptide Receptor with an 18F-Labeled Bombesin Analog

(2012) I. Dijkgraaf et al.   JOURNAL OF NUCLEAR MEDICINE

One-step 18F-labeling of peptides for positron emission tomography imaging using the SiFA methodology

(2012) Carmen Wängler et al.   Nature Protocols

18F-Labeled phosphopeptide-cell-penetrating peptide dimers with enhanced cell uptake properties in human cancer cells

(2012) Susan Richter et al.   NUCLEAR MEDICINE AND BIOLOGY

Evaluation of an integrin αvβ6-specific peptide labeled with [18F]fluorine by copper-free, strain-promoted click chemistry

(2012) Sven H. Hausner et al.   NUCLEAR MEDICINE AND BIOLOGY

Strain-Promoted Copper-Free “Click” Chemistry for 18F Radiolabeling of Bombesin

(2011) Lachlan S. Campbell-Verduyn et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)

(2011) Torsten Kniess et al.   APPLIED RADIATION AND ISOTOPES

[18F]Azadibenzocyclooctyne ([18F]ADIBO): A biocompatible radioactive labeling synthon for peptides using catalyst free [3+2] cycloaddition

(2011) Selvanathan Arumugam et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Tetrazine-trans-cyclooctene ligation for the rapid construction of integrin αvβ3 targeted PET tracer based on a cyclic RGD peptide

(2011) Ramajeyam Selvaraj et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Stable aluminium fluoride chelates with triazacyclononane derivatives proved by X-ray crystallography and 18F-labeling study

(2011) Dinesh Shetty et al.   CHEMICAL COMMUNICATIONS

Recent Progress in Radiofluorination of Peptides for PET Molecular Imaging

(2011) Shuanglong Liu et al.   CURRENT ORGANIC SYNTHESIS

One-step radiosynthesis of 18F-AlF-NOTA-RGD2 for tumor angiogenesis PET imaging

(2011) Shuanglong Liu et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Evaluation of 177Lu-DOTA-sst2 Antagonist Versus 177Lu-DOTA-sst2 Agonist Binding in Human Cancers In Vitro

(2011) R. Cescato et al.   JOURNAL OF NUCLEAR MEDICINE

Fully Automated Preparation and Conjugation of N-Succinimidyl 4-[18F]Fluorobenzoate ([18F]SFB) with RGD Peptide Using a GE FASTlab™ Synthesizer

(2011) David Thonon et al.   MOLECULAR IMAGING AND BIOLOGY

Towards kit-like 18F-labeling of marimastat, a noncovalent inhibitor drug for in vivo PET imaging cancer associated matrix metalloproteases

(2011) Ying Li et al.   MedChemComm

Automated radiochemical synthesis of [18F]FBEM: A thiol reactive synthon for radiofluorination of peptides and proteins

(2010) Dale O. Kiesewetter et al.   APPLIED RADIATION AND ISOTOPES

Click-Chemistry Reactions in Radiopharmaceutical Chemistry: Fast & Easy Introduction of Radiolabels into Biomolecules for In Vivo Imaging

(2010) C. Wangler et al.   CURRENT MEDICINAL CHEMISTRY

A Novel Facile Method of Labeling Octreotide with 18F-Fluorine

(2010) P. Laverman et al.   JOURNAL OF NUCLEAR MEDICINE

Labeling and Glycosylation of Peptides Using Click Chemistry: A General Approach to 18F-Glycopeptides as Effective Imaging Probes for Positron Emission Tomography

(2009) Simone Maschauer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

New Strategy for the Preparation of Clickable Peptides and Labeling with 1-(Azidomethyl)-4-[18F]-fluorobenzene for PET

(2009) David Thonon et al.   BIOCONJUGATE CHEMISTRY

Direct labelling of peptides with 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG)

(2009) Frank Wuest et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Organofluorosilanes as Model Compounds for18F-Labeled Silicon-Based PET Tracers and their Hydrolytic Stability: Experimental Data and Theoretical Calculations (PET=Positron Emission Tomography)

(2009) Aileen Höhne et al.   CHEMISTRY-A EUROPEAN JOURNAL

18F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK)

(2009) Christina Hultsch et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

A Novel Method of 18F Radiolabeling for PET

(2009) W. J. McBride et al.   JOURNAL OF NUCLEAR MEDICINE

Molecular imaging targeting peptide receptors

(2009) Margret Schottelius et al.   METHODS

Recent Applications of Click Chemistry for the Synthesis of Radiotracers for Molecular Imaging

(2009) Constantin Mamat et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†

(2008) Frank Wuest et al.   BIOCONJUGATE CHEMISTRY

Synthesis,18F-Labeling, andin Vitroandin VivoStudies of Bombesin Peptides Modified with Silicon-Based Building Blocks

(2008) Aileen Höhne et al.   BIOCONJUGATE CHEMISTRY

Facile synthesis ofN-succinimidyl 4-[18F]fluorobenzoate ([18F]SFB) for protein labeling

(2008) G. Tang et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

In Vivo Positron Emission Tomography (PET) Imaging with an αvβ6Specific Peptide Radiolabeled using18F-“Click” Chemistry: Evaluation and Comparison with the Corresponding 4-[18F]Fluorobenzoyl- and 2-[18F]Fluoropropionyl-Peptides

(2008) Sven H. Hausner et al.   JOURNAL OF MEDICINAL CHEMISTRY