One-step 18F-labeling of peptides for positron emission tomography imaging using the SiFA methodology

New Lyophilized Kit for Rapid Radiofluorination of Peptides

(2012) William J. McBride et al.   BIOCONJUGATE CHEMISTRY

Synthesis of [18F]SiFB: a prosthetic group for direct protein radiolabeling for application in positron emission tomography

(2012) Alexey P Kostikov et al.   Nature Protocols

Protein labeling with the labeling precursor [18F]SiFA-SH for positron emission tomography

(2012) Björn Wängler et al.   Nature Protocols

Silicon-[18F]Fluorine Radiochemistry: Basics, Applications and Challenges

(2012) Carmen Wängler et al.   Applied Sciences-Basel

Rapid and Simple One-Step F-18 Labeling of Peptides

(2011) Orit Jacobson et al.   BIOCONJUGATE CHEMISTRY

High-Yielding Aqueous18F-Labeling of Peptides via Al18F Chelation

(2011) Christopher A. D’Souza et al.   BIOCONJUGATE CHEMISTRY

[18F]Azadibenzocyclooctyne ([18F]ADIBO): A biocompatible radioactive labeling synthon for peptides using catalyst free [3+2] cycloaddition

(2011) Selvanathan Arumugam et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Inorganic approaches for radiolabelling biomolecules with fluorine-18 for imaging with Positron Emission Tomography

(2011) Gareth E. Smith et al.   DALTON TRANSACTIONS

Synthesis and hydrolytic stability of novel 3-[18F]fluoroethoxybis(1-methylethyl)silyl]propanamine-based prosthetic groups

(2011) Eva Balentova et al.   JOURNAL OF FLUORINE CHEMISTRY

t-Bu2SiF-Derivatized D2-Receptor Ligands: The First SiFA-Containing Small Molecule Radiotracers for Target-Specific PET-Imaging

(2011) Ljuba Iovkova-Berends et al.   MOLECULES

Preparation of 18F-labeled peptides using the copper(I)-catalyzed azide-alkyne 1,3-dipolar cycloaddition

(2011) Herman S Gill et al.   Nature Protocols

SiFA Azide: A New Building Block for PET Imaging Using Click Chemistry

(2011) Lutz Tietze et al.   SYNLETT

Towards kit-like 18F-labeling of marimastat, a noncovalent inhibitor drug for in vivo PET imaging cancer associated matrix metalloproteases

(2011) Ying Li et al.   MedChemComm

One-Step18F-Labeling of Carbohydrate-Conjugated Octreotate-Derivatives Containing a Silicon-Fluoride-Acceptor (SiFA): In Vitro and in Vivo Evaluation as Tumor Imaging Agents for Positron Emission Tomography (PET)

(2010) Carmen Wängler et al.   BIOCONJUGATE CHEMISTRY

Improved18F Labeling of Peptides with a Fluoride-Aluminum-Chelate Complex

(2010) William J. McBride et al.   BIOCONJUGATE CHEMISTRY

Click-Chemistry Reactions in Radiopharmaceutical Chemistry: Fast & Easy Introduction of Radiolabels into Biomolecules for In Vivo Imaging

(2010) C. Wangler et al.   CURRENT MEDICINAL CHEMISTRY

N-(4-(di-tert-butyl[18F]fluorosilyl)benzyl)-2-hydroxy-N,N-dimethylethylammonium bromide ([18F]SiFAN+Br−): A novel lead compound for the development of hydrophilic SiFA-based prosthetic groups for 18F-labeling

(2010) Alexey P. Kostikov et al.   JOURNAL OF FLUORINE CHEMISTRY

One Step Radiosynthesis of 6-[18F]Fluoronicotinic Acid 2,3,5,6-Tetrafluorophenyl Ester ([18F]F-Py-TFP): A New Prosthetic Group for Efficient Labeling of Biomolecules with Fluorine-18

(2010) Dag E. Olberg et al.   JOURNAL OF MEDICINAL CHEMISTRY

Solid-phase synthesis of short α-helices stabilized by the hydrogen bond surrogate approach

(2010) Anupam Patgiri et al.   Nature Protocols

Labeling and Glycosylation of Peptides Using Click Chemistry: A General Approach to 18F-Glycopeptides as Effective Imaging Probes for Positron Emission Tomography

(2009) Simone Maschauer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Novel Method for Direct Site-Specific Radiolabeling of Peptides Using [18F]FDG

(2009) Mohammad Namavari et al.   BIOCONJUGATE CHEMISTRY

Direct One-Step18F-Labeling of Peptides via Nucleophilic Aromatic Substitution

(2009) Jessica Becaud et al.   BIOCONJUGATE CHEMISTRY

Radiolabelling of proteins with fluorine-18 via click chemistry

(2009) Theres Ramenda et al.   CHEMICAL COMMUNICATIONS

para-Functionalized Aryl-di-tert-butylfluorosilanes as Potential Labeling Synthons for18F Radiopharmaceuticals

(2009) Ljuba Iovkova et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organofluorosilanes as Model Compounds for18F-Labeled Silicon-Based PET Tracers and their Hydrolytic Stability: Experimental Data and Theoretical Calculations (PET=Positron Emission Tomography)

(2009) Aileen Höhne et al.   CHEMISTRY-A EUROPEAN JOURNAL

Nucleophilic ring-opening of activated aziridines: A one-step method for labeling biomolecules with fluorine-18

(2009) Ulrike Roehn et al.   JOURNAL OF FLUORINE CHEMISTRY

‘Click labelling’ in PET radiochemistry

(2009) Matthias Glaser et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

A Modular Platform for the Rapid Site-Specific Radiolabeling of Proteins with18F Exemplified by Quantitative Positron Emission Tomography of Human Epidermal Growth Factor Receptor 2

(2009) Herman S. Gill et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Novel Method of 18F Radiolabeling for PET

(2009) W. J. McBride et al.   JOURNAL OF NUCLEAR MEDICINE

Recent Applications of Click Chemistry for the Synthesis of Radiotracers for Molecular Imaging

(2009) Constantin Mamat et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Methods for 18F-labeling of RGD peptides: comparison of aminooxy [18F]fluorobenzaldehyde condensation with ‘click labeling’ using 2-[18F]fluoroethylazide, and S-alkylation with [18F]fluoropropanethiol

(2008) Matthias Glaser et al.   AMINO ACIDS

Systematic comparison of two novel, thiol-reactive prosthetic groups for 18F labeling of peptides and proteins with the acylation agent succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)

(2008) Frank Wuest et al.   AMINO ACIDS

Silicon-Based Building Blocks for One-Step18F-Radiolabeling of Peptides for PET Imaging

(2008) Linjing Mu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis,18F-Labeling, andin Vitroandin VivoStudies of Bombesin Peptides Modified with Silicon-Based Building Blocks

(2008) Aileen Höhne et al.   BIOCONJUGATE CHEMISTRY

Chemistry with [18F]Fluoride Ion

(2008) Lisheng Cai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Radiosynthesis and bioconjugation of [18F]FPy5yne, a prosthetic group for the18F labeling of bioactive peptides

(2008) James A. H. Inkster et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Toward [18F]-Labeled Aryltrifluoroborate Radiotracers: In Vivo Positron Emission Tomography Imaging of Stable Aryltrifluoroborate Clearance in Mice

(2008) Richard Ting et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY