Strain-Promoted Copper-Free “Click” Chemistry for 18F Radiolabeling of Bombesin

In Vitro and In Vivo Evaluation of 64Cu-Labeled SarAr-Bombesin Analogs in Gastrin-Releasing Peptide Receptor-Expressing Prostate Cancer

(2011) K. A. Lears et al.   JOURNAL OF NUCLEAR MEDICINE

Readily Accessible Bicyclononynes for Bioorthogonal Labeling and Three-Dimensional Imaging of Living Cells

(2010) Jan Dommerholt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A DOTA–peptide conjugate by copper-free click chemistry

(2010) Molly E. Martin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Bombesin derivative radiolabeled with technetium-99m as agent for tumor identification

(2010) André Luís Branco de Barros et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

A standardised study to compare prostate cancer targeting efficacy of five radiolabelled bombesin analogues

(2010) Rogier P. J. Schroeder et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Metal-Free Sequential [3 + 2]-Dipolar Cycloadditions using Cyclooctynes and 1,3-Dipoles of Different Reactivity

(2010) Brian C. Sanders et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-free click chemistry in living animals

(2010) P. V. Chang et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Bioorthogonal Chemistry: Fishing for Selectivity in a Sea of Functionality

(2009) Ellen M. Sletten et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct One-Step18F-Labeling of Peptides via Nucleophilic Aromatic Substitution

(2009) Jessica Becaud et al.   BIOCONJUGATE CHEMISTRY

18F,64Cu, and68Ga Labeled RGD-Bombesin Heterodimeric Peptides for PET Imaging of Breast Cancer

(2009) Zhaofei Liu et al.   BIOCONJUGATE CHEMISTRY

Phosphoramidite accelerated copper(i)-catalyzed [3 + 2] cycloadditions of azides and alkynes

(2009) Lachlan S. Campbell-Verduyn et al.   CHEMICAL COMMUNICATIONS

Radiolabelling of proteins with fluorine-18 via click chemistry

(2009) Theres Ramenda et al.   CHEMICAL COMMUNICATIONS

Aza-dibenzocyclooctynes for fast and efficient enzyme PEGylation via copper-free (3+2) cycloaddition

(2009) Marjoke F. Debets et al.   CHEMICAL COMMUNICATIONS

True radiotracers: Cu-64 targeting vectors based upon bombesin peptide

(2009) Timothy J. Hoffman et al.   NUCLEAR MEDICINE AND BIOLOGY

Visualizing Metabolically Labeled Glycoconjugates of Living Cells by Copper-Free and Fast Huisgen Cycloadditions

(2008) Xinghai Ning et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis,18F-Labeling, andin Vitroandin VivoStudies of Bombesin Peptides Modified with Silicon-Based Building Blocks

(2008) Aileen Höhne et al.   BIOCONJUGATE CHEMISTRY

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

“Click‐to‐Chelate”: Design and Incorporation of Triazole‐Containing Metal‐Chelating Systems into Biomolecules of Diagnostic and Therapeutic Interest

(2008) Harriet Struthers et al.   CHEMISTRY-A EUROPEAN JOURNAL

Nuclear Imaging of Prostate Cancer with Gastrin-Releasing-Peptide- Receptor Targeted Radiopharmaceuticals

(2008) H. Ananias et al.   CURRENT PHARMACEUTICAL DESIGN

In Vivo Positron Emission Tomography (PET) Imaging with an αvβ6Specific Peptide Radiolabeled using18F-“Click” Chemistry: Evaluation and Comparison with the Corresponding 4-[18F]Fluorobenzoyl- and 2-[18F]Fluoropropionyl-Peptides

(2008) Sven H. Hausner et al.   JOURNAL OF MEDICINAL CHEMISTRY

Dual Integrin and Gastrin-Releasing Peptide Receptor Targeted Tumor Imaging Using18F-labeled PEGylated RGD-Bombesin Heterodimer18F-FB-PEG3-Glu-RGD-BBN

(2008) Zhaofei Liu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Radiolabeled bombesin analogs for prostate cancer diagnosis: preclinical studies

(2008) Bluma Linkowski Faintuch et al.   NUCLEAR MEDICINE AND BIOLOGY

Rapid in situ synthesis of [11C]methyl azide and its application in 11C click-chemistry

(2008) Ralf Schirrmacher et al.   TETRAHEDRON LETTERS