A stable meta -carborane enables the generation of boron-rich peptide agonists targeting the ghrelin receptor

Direct carborane-peptide conjugates: Synthesis and evaluation as non-natural lipopeptide mimetics

(2018) Tamara Lützenburg et al.   CHEMISTRY AND PHYSICS OF LIPIDS

Towards carborane-functionalised structures for the treatment of brain cancer

(2018) Gianpiero Calabrese et al.   DRUG DISCOVERY TODAY

Development of Albumin-closo -Dodecaborate Conjugates as Boron Carriers for Neutron-Capture Therapy by Ru(bpy)3 -Photocatalyzed Modification of Tyrosine

(2017) Shinichi Sato et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

C-terminus of a hexapeptidic ghrelin receptor inverse agonist can switch peptide behavior from inverse agonism to agonism

(2016) Sylvia Els-Heindl et al.   BIOPOLYMERS

Tumor-specific delivery of BSH-3R for boron neutron capture therapy and positron emission tomography imaging in a mouse brain tumor model

(2015) Yoshiya Iguchi et al.   BIOMATERIALS

High metabolic in vivo stability and bioavailability of a palmitoylated ghrelin receptor ligand assessed by mass spectrometry

(2015) Katja B. Kostelnik et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Advancements in Tumor Targeting Strategies for Boron Neutron Capture Therapy

(2015) Micah John Luderer et al.   PHARMACEUTICAL RESEARCH

The acceleration of boron neutron capture therapy using multi-linked mercaptoundecahydrododecaborate (BSH) fused cell-penetrating peptide

(2014) Hiroyuki Michiue et al.   BIOMATERIALS

Receptor-Mediated Uptake of Boron-Rich Neuropeptide Y Analogues for Boron Neutron Capture Therapy

(2014) Verena M. Ahrens et al.   ChemMedChem

MECHANISMS IN ENDOCRINOLOGY: Regulation of glucose metabolism by the ghrelin system: multiple players and multiple actions

(2014) Kristy M Heppner et al.   EUROPEAN JOURNAL OF ENDOCRINOLOGY

N3-substituted thymidine bioconjugates for cancer therapy and imaging

(2013) Ahmed Khalil et al.   Future Medicinal Chemistry

An Aromatic Region To Induce a Switch between Agonism and Inverse Agonism at the Ghrelin Receptor

(2012) Sylvia Els et al.   JOURNAL OF MEDICINAL CHEMISTRY

Current status of boron neutron capture therapy of high grade gliomas and recurrent head and neck cancer

(2012) Rolf F Barth et al.   Radiation Oncology

Synthesis and evaluation of cyclic RGD-boron cluster conjugates to develop tumor-selective boron carriers for boron neutron capture therapy

(2011) Sadaaki Kimura et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbaboranes as Pharmacophores: Properties, Synthesis, and Application Strategies

(2011) Matthias Scholz et al.   CHEMICAL REVIEWS

Unique Interaction Pattern for a Functionally Biased Ghrelin Receptor Agonist

(2011) Bjørn Sivertsen et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Incorporation ofortho-Carbaboranyl-Nε-Modifiedl-Lysine into Neuropeptide Y Receptor Y1- and Y2-Selective Analogues

(2011) Verena M. Ahrens et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structure–Activity Relationships of GHRP-6 Azapeptide Ligands of the CD36 Scavenger Receptor by Solid-Phase Submonomer Azapeptide Synthesis

(2011) David Sabatino et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ghrelin: A potential therapeutic target for cancer

(2010) Dimitrios Nikolopoulos et al.   REGULATORY PEPTIDES

A novel boronated-porphyrin as a radio-sensitizing agent for boron neutron capture therapy of tumours: In vitro and in vivo studies

(2009) G Jori et al.   APPLIED RADIATION AND ISOTOPES

Biological evaluation of boronated unnatural amino acids as new boron carriers

(2009) G.W. Kabalka et al.   APPLIED RADIATION AND ISOTOPES

Convection enhanced delivery of boronated EGF as a molecular targeting agent for neutron capture therapy of brain tumors

(2009) Weilian Yang et al.   JOURNAL OF NEURO-ONCOLOGY

Biodistribution of10B for Boron Neutron Capture Therapy (BNCT) in a Mouse Model after Injection of Sodium Mercaptoundecahydro-closo-dodecaborate and l-para-Boronophenylalanine

(2009) Andrea Wittig et al.   RADIATION RESEARCH

closo-Borane Conjugated Regulatory Peptides Retain High Biological Affinity: Synthesis ofcloso-Borane Conjugated Tyr3-Octreotate Derivatives for BNCT

(2008) Thomas Betzel et al.   BIOCONJUGATE CHEMISTRY