Scavenging strategy for specific activity improvement: application to a new CXCR4-specific cyclopentapeptide positron emission tomography tracer

Fully automated radiosynthesis of [1-(2-[18F]fluoroethyl),1H[1,2,3]triazole 4-ethylene] triphenylphosphonium bromide as a potential positron emission tomography tracer for imaging apoptosis

(2013) Anna Haslop et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Imaging agents for the chemokine receptor 4 (CXCR4)

(2012) Joeri Kuil et al.   CHEMICAL SOCIETY REVIEWS

The emerging role of CXC chemokines and their receptors in cancer

(2012) Victoria Vinader et al.   Future Medicinal Chemistry

Nuclear (PET/SPECT) and optical imaging probes targeting the CXCR4 chemokine receptor

(2012) James C. Knight et al.   MedChemComm

Radiolabeled Peptides: Valuable Tools for the Detection and Treatment of Cancer

(2012) M. Fani et al.   Theranostics

Synthesis and in vitro evaluation of [18F]fluoroethyl triazole labelled [Tyr3]octreotate analogues using click chemistry

(2011) Lisa Iddon et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

18F-labelling of a cyclic pentapeptide inhibitor of the chemokine receptor CXCR4

(2011) Ola Åberg et al.   JOURNAL OF FLUORINE CHEMISTRY

CXCR4-Based Imaging Agents

(2011) L. E. Woodard et al.   JOURNAL OF NUCLEAR MEDICINE

Radiolabelled proteins for positron emission tomography: Pros and cons of labelling methods

(2010) Vladimir Tolmachev et al.   BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS

Effects of a Flexible Alkyl Chain on a Ligand for CuAAC Reaction

(2010) Keisuke Asano et al.   ORGANIC LETTERS

Structures of the CXCR4 Chemokine GPCR with Small-Molecule and Cyclic Peptide Antagonists

(2010) B. Wu et al.   SCIENCE

‘Click labelling’ in PET radiochemistry

(2009) Matthias Glaser et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Physicochemical Determinants of Human Renal Clearance

(2009) Manthena V. S. Varma et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids

(2009) Tomohiro Tanaka et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

CXCR4, Inhibitors and Mechanisms of Action

(2008) Xiangyang Liang   Chemical Biology & Drug Design

Molecular Imaging with PET

(2008) Simon M. Ametamey et al.   CHEMICAL REVIEWS

Tumor Receptor Imaging

(2008) D. A. Mankoff et al.   JOURNAL OF NUCLEAR MEDICINE

Structure-activity relationship study of CXCR4 antagonists bearing the cyclic pentapeptide scaffold: identification of the new pharmacophore

(2008) Tomohiro Tanaka et al.   ORGANIC & BIOMOLECULAR CHEMISTRY