Synthesis of Heterocycles via Nucleophilic Substitution of Hydrogen in Nitroarenes

Simple synthesis of pyrrolo[3,2-e]indole-1-carbonitriles

(2013) Adam Trawczyński et al.   Beilstein Journal of Organic Chemistry

Synthesis of SF5-containing benzisoxazoles, quinolines, and quinazolines by the Davis reaction of nitro-(pentafluorosulfanyl)benzenes

(2013) Petr Beier et al.   Beilstein Journal of Organic Chemistry

Efficient Synthesis of 1-Arylquinoxalin-2(1H)-onesviaCyclocondensation ofN-Aryl-Substituted 2-Nitrosoanilines with Functionalized Alkyl Acetates

(2013) Zbigniew Wróbel et al.   HELVETICA CHIMICA ACTA

Synthesis and biological evaluation of novel isoxazolo[4,3-e]indoles as antibacterial agents

(2013) Mehdi Pordel et al.   RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY

A Short Preparation of Pyrroloquinoxalinones via a Cascade Reaction of N-Aryl-5-alkylamino-2-nitrosoanilines with Methyl 2-Cyanoalkanoates: Unexpected Direction of Nucleophilic Substitution of Hydrogen

(2013) Zbigniew Wróbel et al.   SYNLETT

Synthesis of Pentafluorosulfanyl-Containing Indoles and Oxindoles

(2013) Petr Beier et al.   SYNLETT

Progress in palladium-based catalytic systems for the sustainable synthesis of annulated heterocycles: a focus on indole backbones

(2012) Mélanie Platon et al.   CHEMICAL SOCIETY REVIEWS

Phenazines and cancer

(2012) A. Cimmino et al.   NATURAL PRODUCT REPORTS

Development of Scalable Manufacturing Routes to AZD1981. Application of the Semmler–Wolff Aromatisation for Synthesis of the Indole-4-amide Core

(2012) Manjunatha Sulur et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Expedient Synthesis of 1-Hydroxy-4- and 1-Hydroxy-6-nitroindoles

(2012) Krzysztof Wojciechowski et al.   SYNLETT

New Simple Synthesis of Quinoline-4-carbonitriles

(2012) Krzysztof Wojciechowski et al.   SYNLETT

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

(2011) Matthieu Jeanty et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

An efficient one-pot synthesis of a new heterocyclic system with high-fluorescent properties

(2011) Mohammad Rahimizadeh et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Preparation of SF5Aromatics by Vicarious Nucleophilic Substitution Reactions of Nitro(pentafluorosulfanyl)benzenes with Carbanions

(2011) Petr Beier et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent advances in indole syntheses: New routes for a classic target

(2011) Rubén Vicente   ORGANIC & BIOMOLECULAR CHEMISTRY

N-Aryl-2-nitrosoanilines as Intermediates in the Two-Step Synthesis of Substituted 1,2-Diarylbenzimidazoles from Simple Nitroarenes

(2011) Zbigniew Wróbel et al.   SYNLETT

Nucleophilic Substitution of Hydrogen in Nitroarenes: A New Chapter of Aromatic Chemistry

(2011) Mieczysław Mąkosza   SYNTHESIS-STUTTGART

A base-modulated chemoselective synthesis of 3-cyanoindoles or 4-cyanoquinolines using a palladium-catalyzed N-heterocyclization

(2011) Serge R. Banini et al.   TETRAHEDRON

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

N-Aryl-2-nitrosoanilines as intermediates in the synthesis of substituted phenazines from nitroarenes

(2011) Andrzej Kwast et al.   TETRAHEDRON LETTERS

3-(Arylsulfonyl)-1-(azacyclyl)-1H-indoles are 5-HT6 receptor modulators

(2010) Ronald C. Bernotas et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Nucleophilic substitution of hydrogen in electron-deficient arenes, a general process of great practical value

(2010) Mieczysław Mąkosza   CHEMICAL SOCIETY REVIEWS

Vicarious nucleophilic substitution in nitro derivatives of imidazo[1,2-a]pyridine

(2010) Mohammad Rahimizadeh et al.   MENDELEEV COMMUNICATIONS

Short and Simple Method of Synthesis of Some Pyrrolo[3,2-b]quinoline Derivatives from Easily Available Nitrobenzene Derivatives

(2010) Zbigniew Wróbel et al.   SYNLETT

Simple Synthesis of N-Aryl-2-nitrosoanilines in the Reaction of Nitroarenes with Aniline Anion Derivatives

(2010) Zbigniew Wróbel et al.   SYNTHESIS-STUTTGART

Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: Exploration of 5–6 fused rings as alternative S1 moieties

(2009) Kenji Yoshikawa et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Dual acting norepinephrine reuptake inhibitors and 5-HT2A receptor antagonists: Identification, synthesis and activity of novel 4-aminoethyl-3-(phenylsulfonyl)-1H-indoles

(2009) Gavin D. Heffernan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT6 receptor ligands

(2009) Ronald C. Bernotas et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of α-(Nitroaryl)benzylphosphonates via Oxidative Nucleophilic Substitution of Hydrogen in Nitroarenes†

(2009) Mieczysław Ma̧kosza et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of imidazo[4,5-a]acridones and imidazo[4,5-a]acridines as potential antibacterial agents

(2009) Mohammad Rahimizadeh et al.   MONATSHEFTE FUR CHEMIE

Novel approach to synthesis of substituted 3-aminoquinolines from nitroarenes and protected ethyl aminocrotonate

(2009) Robert Bujok et al.   TETRAHEDRON

Substituent Effects on the Electrophilic Activity of Nitroarenes in Reactions with Carbanions

(2008) Sylwia Błażej et al.   CHEMISTRY-A EUROPEAN JOURNAL

Reactions of Nitroheteroarenes with Carbanions: Bridging Aromatic, Heteroaromatic, and Vinylic Electrophilicity

(2008) Florian Seeliger et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and adrenolytic activity of 1-(1H-indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)ethyl]amino}propan-2-ol and its enantiomers. Part 1

(2008) Grażyna Groszek et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Selective Ortho Methylation of Nitroheteroaryls by Vicarious Nucleophilic Substitution

(2008) Michał Achmatowicz et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of C3-Substituted 4-Azaindoles: An Easy Access to 4-Azamelatonin and Protected 4-Azatryptophan

(2008) Matthieu Jeanty et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Eudistomin C and E: Improved Preparation of the Indole Unit

(2008) Hiroaki Yamagishi et al.   ORGANIC LETTERS

Palladium-Catalyzed Synthesis of 3-Indolecarboxylic Acid Derivatives

(2008) Björn Söderberg et al.   SYNTHESIS-STUTTGART

Synthesis of 2-aryl-6-methyl-5-nitroquinoline derivatives as potential prodrug systems for reductive activation

(2008) Gavin D. Couch et al.   TETRAHEDRON