Direct Assembly of Benzo[e]indoles by Diels-Alder Reaction of Arynes and 2-Vinylpyrroles

Expedient Iodocyclization Approach Toward Polysubstituted 3H-Benzo[e]indoles

(2015) Guilherme M. Martins et al.   ADVANCED SYNTHESIS & CATALYSIS

Recent Advances in Aryne Double Bond Insertion

(2015) Chunrui Wu et al.   CHINESE JOURNAL OF ORGANIC CHEMISTRY

Total Syntheses of Aporphine Alkaloids via Benzyne Chemistry: An Approach to the Formation of Aporphine Cores

(2015) Allan F. C. Rossini et al.   JOURNAL OF ORGANIC CHEMISTRY

Triple Benzannulation of Naphthalene via a 1,3,6-Naphthotriyne Synthetic Equivalent. Synthesis of Dibenz[a,c]anthracene

(2015) Philip Z. Mannes et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Benzo[c]carbazoles and Their Antitumor Derivatives through the Diels–Alder Reaction of 2-Alkenylindoles and Arynes

(2015) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

Facile synthesis of benzoindoles and naphthofurans through carbonaceous material-catalyzed cyclization of naphthylamines/naphthols with nitroolefins in water

(2015) Furen Zhang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The Aryne aza-Diels–Alder Reaction: Flexible Syntheses of Isoquinolines

(2015) Juan-Carlos Castillo et al.   ORGANIC LETTERS

A practical, multi-gram synthesis of (±)-herbindole A, (±)-herbindole B, and (±)-herbindole C from a common intermediate via 6,7-indole aryne cycloaddition and Pd(0)-catalyzed cross-coupling reactions

(2015) Nalin Chandrasoma et al.   TETRAHEDRON LETTERS

Facile Synthesis of Chiral Spirooxindole-Based Isotetronic Acids and 5-1H-Pyrrol-2-ones through Cascade Reactions with Bifunctional Organocatalysts

(2014) Wengang Guo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Diels–Alder Reaction of Tropones with Arynes: Synthesis of Functionalized Benzobicyclo[3.2.2]nonatrienones

(2014) Manikandan Thangaraj et al.   JOURNAL OF ORGANIC CHEMISTRY

A Tandem Reaction of Benzyne with Functionalized Benzylidenephthalan To Afford Phenanthro[10,1-bc]furan

(2014) Hai Xiao Siyang et al.   JOURNAL OF ORGANIC CHEMISTRY

Tandem [4 + 2]/[2 + 2] Cycloaddition Reactions Involving Indene or Benzofurans and Arynes

(2014) Sachin Suresh Bhojgude et al.   ORGANIC LETTERS

Efficient Synthesis of 9-Aryldihydrophenanthrenes by a Cascade Reaction Involving Arynes and Styrenes

(2014) Sachin Suresh Bhojgude et al.   ORGANIC LETTERS

One-pot synthesis of α-fluoro-β-amino acid and indole spiro-derivatives via CN bond cleavage/formation

(2014) Chen-Yu Tang et al.   TETRAHEDRON LETTERS

Direct Assembly of Benzo[a]carbazole-5-carboxylates via a Diels-Alder Reaction with Arynes and 3-Alkenylindoles

(2014) Yuan Tao et al.   Asian Journal of Organic Chemistry

Visible-Light Sensitization of Vinyl Azides by Transition-Metal Photocatalysis

(2013) Elliot P. Farney et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Regioselective Assembly of Di- or Trisubstituted Pyridines from Arynes, Isocyanides, and 3-Bromo- or 3-Acetoxypropynes

(2013) Feng Sha et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Dibromoisobenzofuran as a Formal Equivalent of Didehydroisobenzofuran: Reactive Platform for Expeditious Assembly of Polycycles

(2013) Hiroshi Haneda et al.   ORGANIC LETTERS

Pd-catalyzed assembly of phenanthridines from aryl ketone O-acetyloximes and arynes through C–H bond activation

(2013) Chen-Yu Tang et al.   TETRAHEDRON LETTERS

A Closer Look at Aryne Chemistry: Details that Remain Mysterious

(2013) Chunrui Wu et al.   Asian Journal of Organic Chemistry

Arynes in Transition-Metal-Free Multicomponent Coupling Reactions

(2012) Sachin Suresh Bhojgude et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Arynes and Cyclohexyne in Natural Product Synthesis

(2012) Christian M. Gampe et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Comprehensive History of Arynes in Natural Product Total Synthesis

(2012) Pamela M. Tadross et al.   CHEMICAL REVIEWS

Recent advances in transition-metal-free carbon–carbon and carbon–heteroatom bond-forming reactions using arynes

(2012) Anup Bhunia et al.   CHEMICAL SOCIETY REVIEWS

Chemo- and Regioselective Assembly of Polysubstituted Pyridines and Isoquinolines from Isocyanides, Arynes, and Terminal Alkynes

(2012) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

Use of benzynes for the synthesis of heterocycles

(2012) Anton V. Dubrovskiy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Construction of Naphtho-Fused Oxindoles via the Aryne Diels–Alder Reaction with Methyleneindolinones

(2012) Jian Li et al.   ORGANIC LETTERS

A Practical and General Diels–Alder Reaction of Pentafulvenes with Arynes

(2012) Sachin Suresh Bhojgude et al.   ORGANIC LETTERS

Aryne Insertion Reactions into Carbon-Carbon σ-Bonds

(2012) Hiroto Yoshida et al.   SYNLETT

Overturning Indolyne Regioselectivities and Synthesis of Indolactam V

(2011) Sarah M. Bronner et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Preparation and Regioselective Diels-Alder Reactions of Borylbenzynes: Synthesis of Functionalized Arylboronates

(2010) Takashi Ikawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Domino Diels-Alder Cycloadditions of Arynes: New Approach to Elusive Perylene Derivatives

(2010) Alejandro Criado et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Multicomponent Reaction of Arynes, Isocyanides, and Terminal Alkynes: Highly Chemo- and Regioselective Synthesis of Polysubstituted Pyridines and Isoquinolines

(2009) Feng Sha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enamide-Benzyne-[2 + 2] Cycloaddition: Stereoselective Tandem [2 + 2]−Pericyclic Ring-Opening−IntramolecularN-Tethered [4 + 2] Cycloadditions

(2009) John B. Feltenberger et al.   ORGANIC LETTERS

Duocarmycin-based prodrugs for cancer prodrug monotherapy

(2008) Lutz F. Tietze et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A Concise Total Synthesis of (−)-Quinocarcin via Aryne Annulation

(2008) Kevin M. Allan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Multicomponent reactions of pyridines, α-bromo carbonyl compounds and silylaryl triflates as aryne precursors: a facile one-pot synthesis of pyrido[2,1-a]isoindoles

(2008) Xian Huang et al.   TETRAHEDRON LETTERS