Highly Regioselective Assembly of Di- or Trisubstituted Pyridines from Arynes, Isocyanides, and 3-Bromo- or 3-Acetoxypropynes

Coupling of enamides with alkynes or arynes for synthesis of substituted pyridines and isoquinolines via amide activation

(2012) Mi-Na Zhao et al.   CHEMICAL COMMUNICATIONS

A “one-pot” multicomponent approach to polysubstituted 4-aminopyridines

(2012) Jiaan Shao et al.   CHEMICAL COMMUNICATIONS

Chemo- and Regioselective Assembly of Polysubstituted Pyridines and Isoquinolines from Isocyanides, Arynes, and Terminal Alkynes

(2012) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

Use of benzynes for the synthesis of heterocycles

(2012) Anton V. Dubrovskiy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

DPTA-catalyzed one-pot regioselective synthesis of polysubstituted pyridines and 1,4-dihydropyridines

(2012) Jianjun Li et al.   TETRAHEDRON

Synthesis of polysubstituted pyridines under combined microwave and ultrasound irradiation: K2CO3-promoted tandem addition/cyclization/hydrogen shift process

(2012) Huangdi Feng et al.   TETRAHEDRON LETTERS

Oppolzer-Type Intramolecular Diels–Alder Cycloadditions via Isomerizations of Allenamides

(2011) John B. Feltenberger et al.   ORGANIC LETTERS

Tandem One-Pot Synthesis of Polysubstituted Pyridines Using the Blaise Reaction Intermediate and 1,3-Enynes

(2011) Yu Sung Chun et al.   ORGANIC LETTERS

Synthesis of Acridines by the [4 + 2] Annulation of Arynes and 2-Aminoaryl Ketones

(2010) Donald C. Rogness et al.   JOURNAL OF ORGANIC CHEMISTRY

A New Strategy for the Synthesis of Poly-Substituted 3-H, 3-Fluoro, or 3-Trifluoromethyl Pyridines via the Tandem C−F Bond Cleavage Protocol

(2010) Zixian Chen et al.   ORGANIC LETTERS

Synthesis of 2-Azaanthracenes via a Sequential Sonogashira Coupling/Alkynyl Imine−Allenyl Imine Isomerization/Aza-Diels−Alder/Elimination−Aromatization Reaction

(2010) Jian Cao et al.   ORGANIC LETTERS

C−H Bond Functionalization via Hydride Transfer: Direct Coupling of Unactivated Alkynes and sp3C−H Bonds Catalyzed by Platinum Tetraiodide

(2009) Paul A. Vadola et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Insertion of Benzene Rings into the Amide Bond: One-Step Synthesis of Acridines and Acridones from Aryl Amides

(2009) Didier G. Pintori et al.   ORGANIC LETTERS

Regioselective synthesis of polysubstituted pyridines via hetero-Diels–Alder reaction of isotellurazoles with acetylenic dienophiles

(2009) Kazuaki Shimada et al.   TETRAHEDRON LETTERS

Metal-free Michael addition initiated multicomponent oxidative cyclodehydration route to polysubstituted pyridines from 1,3-dicarbonyls

(2008) Frédéric Liéby-Muller et al.   CHEMICAL COMMUNICATIONS

Orthogonal Synthesis of Indolines and Isoquinolines via Aryne Annulation

(2008) Christopher D. Gilmore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY