New 1,3,4-Oxadiazole Derivatives of Pyridothiazine-1,1-Dioxide with Anti-Inflammatory Activity
出版年份 2020 全文链接
标题
New 1,3,4-Oxadiazole Derivatives of Pyridothiazine-1,1-Dioxide with Anti-Inflammatory Activity
作者
关键词
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出版物
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Volume 21, Issue 23, Pages 9122
出版商
MDPI AG
发表日期
2020-12-01
DOI
10.3390/ijms21239122
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Design, Synthesis, and Biological Evaluation of 2‐(2‐Bromo‐3‐nitrophenyl)‐5‐phenyl‐1,3,4‐oxadiazole Derivatives as Possible Anti‐Breast Cancer Agents
- (2020) Arjun H. Ananth et al. CHEMISTRY & BIODIVERSITY
- Diversity-oriented synthesis and antifungal activities of novel pimprinine derivative bearing a 1,3,4-oxadiazole-5-thioether moiety
- (2020) Zi-Long Song et al. MOLECULAR DIVERSITY
- Design, Synthesis and In Vitro Characterization of Novel Antimicrobial Agents Based on 6-Chloro-9H-carbazol Derivatives and 1,3,4-Oxadiazole Scaffolds
- (2020) Alexandra T. Bordei Telehoiu et al. MOLECULES
- Effect of Novel Pyrrolo[3,4-d]pyridazinone Derivatives on Lipopolysaccharide-Induced Neuroinflammation
- (2020) Karolina Wakulik et al. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
- Synthesis and anticancer evaluation of new lipophilic 1,2,4 and 1,3,4-oxadiazoles
- (2019) Wiliam Caneschi et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and evaluation of 1,3,4-oxadiazole derivatives for development as broad-spectrum antibiotics
- (2019) Cédric Tresse et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Design, synthesis and molecular docking of benzophenone conjugated with oxadiazole sulphur bridge pyrazole pharmacophores as anti inflammatory and analgesic agents
- (2019) Zabiulla et al. BIOORGANIC CHEMISTRY
- Synthesis, molecular modelling studies and ADME prediction of benzothiazole clubbed oxadiazole-Mannich bases, and evaluation of their anti-diabetic activity through in vivo model
- (2018) Rubina Bhutani et al. BIOORGANIC CHEMISTRY
- Synthesis, thymidine phosphorylase inhibitory and computational study of novel 1,3,4-oxadiazole-2-thione derivatives as potential anticancer agents
- (2018) Shalini Bajaj et al. COMPUTATIONAL BIOLOGY AND CHEMISTRY
- Hypoxia, oxidative stress and inflammation
- (2018) Trudy McGarry et al. FREE RADICAL BIOLOGY AND MEDICINE
- Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain
- (2018) Jatinder Kaur et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Anti-Cancer Activity of Derivatives of 1,3,4-Oxadiazole
- (2018) Teresa Glomb et al. MOLECULES
- S -substituted 3,5-dinitrophenyl 1,3,4-oxadiazole-2-thiols and tetrazole-5-thiols as highly efficient antitubercular agents
- (2017) Galina Karabanovich et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of Oxadiazole-Thiadiazole Hybrids and Their Anticandidal Activity
- (2017) Serkan Levent et al. MOLECULES
- Design, synthesis, evaluation and molecular modelling studies of some novel 5,6-diphenyl-1,2,4-triazin-3(2H)-ones bearing five-member heterocyclic moieties as potential COX-2 inhibitors: A hybrid pharmacophore approach
- (2016) Anupam G. Banerjee et al. BIOORGANIC CHEMISTRY
- Ultrasound- and Molecular Sieves-Assisted Synthesis, Molecular Docking and Antifungal Evaluation of 5-(4-(Benzyloxy)-substituted phenyl)-3-((phenylamino)methyl)-1,3,4-oxadiazole-2(3H)-thiones
- (2016) Urja Nimbalkar et al. MOLECULES
- Synthesis, characterization, evaluation and molecular dynamics studies of 5, 6–diphenyl–1,2,4–triazin–3(2 H )–one derivatives bearing 5–substituted 1,3,4–oxadiazole as potential anti–inflammatory and analgesic agents
- (2015) Anupam G. Banerjee et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Systematic study of constitutive cyclooxygenase-2 expression: Role of NF-κB and NFAT transcriptional pathways
- (2015) Nicholas S. Kirkby et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Design, synthesis, and pharmacological studies of some new Mannich bases and S-alkylated analogs of pyrazole integrated 1,3,4-oxadiazole
- (2015) Shivapura Viveka et al. RESEARCH ON CHEMICAL INTERMEDIATES
- 2,5-Diaryl-1,3,4-oxadiazoles as selective COX-2 inhibitors and anti-inflammatory agents
- (2015) Jagdeep Grover et al. RSC Advances
- Design and Synthesis of Benzimidazole Analogs Endowed with Oxadiazole as Selective COX-2 Inhibitor
- (2014) Ankita Rathore et al. ARCHIV DER PHARMAZIE
- Synthesis, pharmacological screening and in silico studies of new class of Diclofenac analogues as a promising anti-inflammatory agents
- (2014) Mahesh B. Palkar et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Design and synthesis of novel 2-phenyl-5-(1,3-diphenyl-1H-pyrazol-4-yl)-1,3,4-oxadiazoles as selective COX-2 inhibitors with potent anti-inflammatory activity
- (2014) Sumit Bansal et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Oxicams Bind in a Novel Mode to the Cyclooxygenase Active Site via a Two-water-mediated H-bonding Network
- (2014) Shu Xu et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Anti-Inflammatory, Analgesic Evaluation and Molecular Docking Studies of N-Phenyl Anthranilic Acid-Based 1,3,4-Oxadiazole Analogues
- (2013) Suman Bala et al. Journal of Chemistry
- Synthesis and anti-inflammatory activity of novel pyridazine and pyridazinone derivatives as non-ulcerogenic agents
- (2012) Makarem M. Saeed et al. ARCHIVES OF PHARMACAL RESEARCH
- Synthesis and Analgesic and Anti-inflammatory Activity of Ethyl (6-Substituted-3(2H)-pyridazinone-2-yl)acetate Derivatives
- (2012) Yasemin Dündar et al. ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
- Synthesis and biological evaluation of novel piperazine derivatives of flavone as potent anti-inflammatory and antimicrobial agent
- (2012) Girish D. Hatnapure et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Prostaglandins and Inflammation
- (2011) Emanuela Ricciotti et al. ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
- Synthesis, biological evaluation and molecular docking studies of stellatin derivatives as cyclooxygenase (COX-1, COX-2) inhibitors and anti-inflammatory agents
- (2011) Raju Gautam et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis of Novel Nalidixic Acid-Based 1,3,4-Thiadiazole and 1,3,4-Oxadiazole Derivatives as Potent Antibacterial Agents
- (2011) Nisha Aggarwal et al. Chemical Biology & Drug Design
- Oxadiazoles in Medicinal Chemistry
- (2011) Jonas Boström et al. JOURNAL OF MEDICINAL CHEMISTRY
- Preventive but Not Curative Efficacy of Celecoxib on Bladder Carcinogenesis in a Rat Model
- (2011) José Sereno et al. MEDIATORS OF INFLAMMATION
- Managing the adverse effects of nonsteroidal anti-inflammatory drugs
- (2011) Paola Patrignani et al. Expert Review of Clinical Pharmacology
- Anti-inflammatory, anti-proliferative and antioxidant profiles of selective cyclooxygenase-2 inhibition as chemoprevention for rat bladder carcinogenesis
- (2010) Belmiro Parada et al. CANCER BIOLOGY & THERAPY
- Synthesis and biological evaluation of some 1,3,4-oxadiazole derivatives
- (2010) K. Manjunatha et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Inflammation and cancer: interweaving microRNA, free radical, cytokine and p53 pathways
- (2009) A. J. Schetter et al. CARCINOGENESIS
- AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility
- (2009) Garrett M. Morris et al. JOURNAL OF COMPUTATIONAL CHEMISTRY
- Cyclooxygenase-2 Inhibitors, Nonsteroidal Anti-inflammatory Drugs, and Cardiovascular Risk
- (2008) Orly Vardeny et al. CARDIOLOGY CLINICS
- Aroylpropionic acid based 2,5-disubstituted-1,3,4-oxadiazoles: Synthesis and their anti-inflammatory and analgesic activities
- (2008) Mymoona Akhter et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Cancer-related inflammation
- (2008) Alberto Mantovani et al. NATURE
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- (2007) Shashikant V. Bhandari et al. BIOORGANIC & MEDICINAL CHEMISTRY
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