Transition-Metal-Catalyzed Selective Cyclization Strategy to 2-Substituted Benzofurans and Indoles en Route to the Oxa Analogues of Isocryptolepine

Chemoselective Catalytic Conjugate Addition of Alcohols over Amines

(2014) Shuhei Uesugi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Divergent Syntheses of Fused β-Naphthol and Indene Scaffolds by Rhodium-Catalyzed Direct and Decarbonylative Alkyne-Benzocyclobutenone Couplings

(2014) Peng-hao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-pot synthesis of 2-substituted benzo[b]furans via Pd–tetraphosphine catalyzed coupling of 2-halophenols with alkynes

(2014) Rong Zhou et al.   CHEMICAL COMMUNICATIONS

Facile Synthesis of 2-(Perfluoroalkyl)indoles through a Michael Addition/CuI-Catalyzed Annulation Process

(2014) Long Cao et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides

(2014) Mingjuan Su et al.   ORGANIC LETTERS

Intramolecular Larock Indole Synthesis: Preparation of 3,4-Fused Tricyclic Indoles and Total Synthesis of Fargesine

(2013) Dong Shan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Kinugasa Reaction: A Direct One-Pot Route to Highly Functionalized β-Lactams

(2013) Rama K. Khangarot et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Addition of Potassium Aryltrifluoroborates to Aliphatic Nitriles: Synthesis of Alkyl Aryl Ketones, Diketone Compounds, and 2-Arylbenzo[b]furans

(2013) Xingyong Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Electrophilicity: the “dark-side” of indole chemistry

(2013) Marco Bandini   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient Preparation of 4-Hydroxyquinolin-2(1H)-one Derivatives with Silver-Catalyzed Carbon Dioxide Incorporation and Intramolecular Rearrangement

(2013) Tomonobu Ishida et al.   ORGANIC LETTERS

Palladium-Catalyzed Reaction of Arylboronic Acids with Aliphatic Nitriles: Synthesis of Alkyl Aryl Ketones and 2-Arylbenzofurans

(2013) Miaochang Liu et al.   SYNTHESIS-STUTTGART

Recyclable [bmIm]OH promoted one-pot heterocyclization: synthesis of substituted benzofurans

(2013) I.R. Siddiqui et al.   TETRAHEDRON LETTERS

Catalytic Selective Synthesis

(2012) Jessada Mahatthananchai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles in Multicomponent Processes (MCPs)

(2012) Morteza Shiri   CHEMICAL REVIEWS

A Stereoselective Route to Aza-C-aryl Glycosides from Arynes and Chiral Nitrones

(2012) Rama Kanwar Khangarot et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A One-Pot, Copper-Catalyzed Cascade Route to 2-Indolyl-C-glycosides

(2012) Parthasarathi Subramanian et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Dehydrative C–H Alkylation and Alkenylation of Phenols with Alcohols: Expedient Synthesis for Substituted Phenols and Benzofurans

(2012) Dong-Hwan Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Efficient Copper-Catalyzed Three-Component Synthesis of 3-C-Linked Glycosyl Iminocoumarins

(2012) Krishna Kaliappan et al.   SYNTHESIS-STUTTGART

DFT studies of unique stereoelectronic effects of substituents on divergent reaction pathways of methylenecyclobutanone radical cations

(2012) Yusuke Kano et al.   TETRAHEDRON

Palladium-catalyzed cross-couplings of functionalized 2-bromobenzofurans for atom-economic synthesis of 2-arylbenzofurans using triarylbismuth reagents

(2012) Maddali L.N. Rao et al.   TETRAHEDRON LETTERS

Domino Sonogashira Coupling/Cyclization Reaction Catalyzed by Copper and ppb Levels of Palladium: A Concise Route to Indoles and Benzo[b]furans

(2011) Ruiping Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

The Pictet-Spengler Reaction in Nature and in Organic Chemistry

(2011) Joachim Stöckigt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and antimalarial evaluation of novel isocryptolepine derivatives

(2011) Louise R. Whittell et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions

(2011) Sandro Cacchi et al.   CHEMICAL REVIEWS

Sequential and One-Pot Reactions of Phenols with Bromoalkynes for the Synthesis of (Z)-2-Bromovinyl Phenyl Ethers and Benzo[b]furans

(2011) Shihua Wang et al.   ORGANIC LETTERS

An efficient new route towards biologically active isocryptolepine and γ-carboline derivatives using an intramolecular thermal electrocyclization strategy

(2011) Dattatray G. Hingane et al.   TETRAHEDRON LETTERS

To Protonate or Alkylate? Stereoselective Brønsted Acid Catalysis of CC Bond Formation Using Diazoalkanes

(2010) Jeffrey N. Johnston et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

A Flexible Synthesis of Indoles from ortho-Substituted Anilines: A Direct Synthesis of Isocryptolepine

(2010) George Kraus et al.   SYNTHESIS-STUTTGART

Domino synthesis of 2-arylbenzo[b]furans by copper(II)-catalyzed coupling of o-iodophenols and aryl acetylenes

(2010) E.A. Jaseer et al.   TETRAHEDRON

Domino rhodium(I)-catalysed reactions for the efficient synthesis of substituted benzofurans and indoles

(2010) Alistair Boyer et al.   TETRAHEDRON

A direct synthesis of neocryptolepine and isocryptolepine

(2010) George A. Kraus et al.   TETRAHEDRON LETTERS

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Facile and Expeditious Synthesis of Cryptosanguinolentines

(2009) Dalip Kumar et al.   CHEMISTRY LETTERS

Construction of Nitrogen Heterocycles Bearing an Aminomethyl Group by Copper-Catalyzed Domino Three-Component Coupling−Cyclization

(2009) Yusuke Ohta et al.   JOURNAL OF ORGANIC CHEMISTRY

Domino Approach to Benzofurans by the Sequential Sonogashira/Hydroalkoxylation Couplings Catalyzed by New N-Heterocyclic-Carbene-Palladium Complexes

(2009) Alessandro Zanardi et al.   ORGANOMETALLICS

‘Click’ Chemistry on Sugar-Derived Alkynes: A Tandem ‘Click-Click’ Approach to Bistriazoles

(2009) Krishna Kaliappan et al.   SYNLETT

New Route to the Synthesis of the Isocryptolepine Alkaloid and Its Related Skeletons Using a Modified Pictet-Spengler Reaction

(2008) Piyush K. Agarwal et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Development of a one-pot sequential Sonogashira coupling for the synthesis of benzofurans

(2008) Márton Csékei et al.   TETRAHEDRON