Iodine-Mediated Oxidation of Ynamides: A Facile Access toN-Monosubstituted α-Ketoamides and α-Ketoimides

Regio-, and Stereoselective Iodobromination of Ynamides for Synthesis of (E)-1-Bromo-2-iodoenamides

(2014) Masataka Ide et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Studies on copper(i)-catalyzed highly regio- and stereo-selective hydroboration of alkynamides

(2014) Guangke He et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition metal-free oxidation of ynamides for synthesis of α-keto-imides

(2014) Takuya Chikugo et al.   TETRAHEDRON

Intramolecular Paternò–Büchi reaction of atropisomeric α-oxoamides in solution and in the solid-state

(2013) Ramya Raghunathan et al.   CHEMICAL COMMUNICATIONS

Organocatalytic asymmetric multicomponent cascade reaction via 1,3-proton shift and [3+2] cycloaddition: an efficient strategy for the synthesis of oxindole derivatives

(2013) Li Tian et al.   CHEMICAL COMMUNICATIONS

A novel approach for the one-pot preparation of α-ketoamides by anodic oxidation

(2013) Zhenlei Zhang et al.   CHEMICAL COMMUNICATIONS

Synthesis of Oxindoles through the Gold-Catalyzed Oxidation ofN-Arylynamides

(2013) Liu-Qing Yang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iodine/Water-Mediated Oxidation ofo-Alkynylaroyl Compounds and Application of the Products of Oxidation in the Synthesis of Nitrogen Heterocycles

(2013) Karuppusamy Sakthivel et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper(I)-Catalyzed Highly Regio- and Stereoselective Boron Addition-Protonolysis of Alkynamides to give Alkenamides

(2013) Guangke He et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

α-Diketone Formation Accompanied by Oxidation of Sulfur Functional Group by the Reaction of o-Alkynylarenesulfoxide with Iodine

(2013) Shoji Matsumoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Pyrrolo(spiro-[2.3′]-oxindole)-spiro-[4.3″]-oxindole via 1,3-Dipolar Cycloaddition of Azomethine Ylides with 3-Acetonylideneoxindole

(2013) Jun-An Xiao et al.   JOURNAL OF ORGANIC CHEMISTRY

Generation of Rhodium(I) Carbenes from Ynamides and Their Reactions with Alkynes and Alkenes

(2013) Renhe Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective synthesis of 3-hydroxy oxindoles by ytterbium-catalysed decarboxylative addition of β-ketoacids to isatins

(2013) Zhiqiang Duan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Palladium-Catalyzed sp2 and sp3 C–H Bond Activation and Addition to Isatin toward 3-Hydroxy-2-oxindoles

(2013) Gang-Wei Wang et al.   ORGANIC LETTERS

Synthesis of 3-Aza-bicyclo[3.1.0]hexan-2-one Derivatives via Gold-Catalyzed Oxidative Cyclopropanation of N-Allylynamides

(2013) Kai-Bing Wang et al.   ORGANIC LETTERS

Preparation of Phosphonooxymethyl Prodrugs of HIV-1 Attachment Inhibitors

(2013) David K. Leahy et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Iodine in Modern Oxidation Catalysis

(2013) Boris Nachtsheim et al.   SYNTHESIS-STUTTGART

A novel synthesis of diverse 2-amino-5-hydroxy-4H-chromene derivatives with a spirooxindole nucleus by Ca(OH)2-mediated three-component reactions of substituted resorcinols with isatins and malononitrile

(2013) Ji Hyang Park et al.   TETRAHEDRON

Carbon–carbon bond formation via benzoyl umpolung attained by photoinduced electron-transfer with benzimidazolines

(2013) Tomohito Igarashi et al.   TETRAHEDRON LETTERS

Discovery of di-indolinone as a novel scaffold for protein tyrosine phosphatase 1B inhibitors

(2012) Hou-ling Dai et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Gold-catalyzed synthesis of substituted 2-aminofurans via formal [4+1]-cycloadditions on 3-en-1-ynamides

(2012) Ramesh B. Dateer et al.   CHEMICAL COMMUNICATIONS

nBu4NI-catalyzed direct synthesis of α-ketoamides from aryl methyl ketones with dialkylformamides in water using TBHP as oxidant

(2012) Wen-Peng Mai et al.   CHEMICAL COMMUNICATIONS

NIS-Catalyzed Reactions: Amidation of Acetophenones and Oxidative Amination of Propiophenones

(2012) Manjunath Lamani et al.   CHEMISTRY-A EUROPEAN JOURNAL

Gold(I)-Catalyzed Aminohalogenation of FluorinatedN′-Aryl-N-Propargyl Amidines for the Synthesis of Imidazole Derivatives under Mild Conditions

(2012) Shan Li et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Spiro[indoline-3,2′-quinoline] Derivatives through a Four-Component Reaction

(2012) Jing Sun et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Cinchona Alkaloid Catalyzed Regio- and Enantioselective Allylic Amination of Morita-Baylis-Hillman Carbonates with Isatins

(2012) Mei-Xin Zhao et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

TBHP/I2-promoted oxidative coupling of acetophenones with amines at room temperature under metal-free and solvent-free conditions for the synthesis of α-ketoamides

(2012) Xiaobin Zhang et al.   GREEN CHEMISTRY

Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment 6. Preclinical and Human Pharmacokinetic Profiling of BMS-663749, a Phosphonooxymethyl Prodrug of the HIV-1 Attachment Inhibitor 2-(4-Benzoyl-1-piperazinyl)-1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxoethanone (BMS-488043)

(2012) John F. Kadow et al.   JOURNAL OF MEDICINAL CHEMISTRY

Evaluation of Synthetic FK506 Analogues as Ligands for the FK506-Binding Proteins 51 and 52

(2012) Ranganath Gopalakrishnan et al.   JOURNAL OF MEDICINAL CHEMISTRY

α-Oxo-γ-Butyrolactam, N-Containing Pronucleophile in Organocatalytic One-Pot Assembly of Butyrolactam-Fused Indoloquinolizidines

(2012) Hai-Liang Zhu et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Aerobic Oxidative Cross-Dehydrogenative Coupling of Amine and α-Carbonyl Aldehyde: A Practical and Efficient Approach to α-Ketoamides with Wide Substrate Scope

(2012) Chun Zhang et al.   ORGANIC LETTERS

Direct Catalytic Enantioselective Vinylogous Aldol Reaction of α-Branched Enals with Isatins

(2012) Carlo Cassani et al.   ORGANIC LETTERS

Selenium dioxide-mediated synthesis of α-ketoamides from arylglyoxals and secondary amines

(2012) Arthur Y. Shaw et al.   TETRAHEDRON LETTERS

Highly Efficient Assembly of 3-Hydroxy Oxindole Scaffold via a Catalytic Decarboxylative [1,2]-Addition Strategy

(2012) Qiao Ren et al.   ACS Catalysis

Synthesis of 2,6′-Dioxo-1′,5′,6′,7′-tetrahydrospiro[indoline-3,4′-pyrazolo[3,4-b]pyridine]-5′-carbonitriles via a One-Pot, Three-Component Reaction in Water

(2012) Abbas Rahmati et al.   ACS Combinatorial Science

Palladium complexes grafted onto mesoporous silica catalysed the double carbonylation of aryl iodides with amines to give α-ketoamides

(2012) Marie Genelot et al.   Catalysis Science & Technology

Copper-Catalyzed Aerobic Oxidative Coupling of Aryl Acetaldehydes with Anilines Leading to α-Ketoamides

(2011) Chun Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Gold-Catalyzed Oxidative Cyclization of 1,5-Enynes Using External Oxidants

(2011) Dhananjayan Vasu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Neighbouring Formyl Group Assisted Oxidation of o-Alkynylarenecarbaldehydes by an Iodine/Water System

(2011) Karuppusamy Sakthivel et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Gold- and Iodine-Mediated Internal Oxygen Transfer of Nitrone- and Sulfoxide-Functionalized Alkynes

(2011) Dan Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Gold-Catalyzed 1,2-Difunctionalizations of Aminoalkynes Using Only N- and O-Containing Oxidants

(2011) Anupam Mukherjee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Gold-Catalyzed Synthesis of Benzil Derivatives and α-Keto Imides via Oxidation of Alkynes

(2011) Cheng-Fu Xu et al.   ORGANIC LETTERS

Practical synthesis of amides from alkynyl bromides, amines, and water

(2011) Zheng-Wang Chen et al.   TETRAHEDRON

Fine tuning of receptor polarity for the development of selective naked eye anion receptor

(2011) Jin Joo Park et al.   TETRAHEDRON LETTERS

Total Synthesis of Complestatin (Chloropeptin II)

(2010) Zhihui Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Three-Component Coupling Reactions of Silyl Glyoxylates, Vinyl Grignard Reagent, and Nitroalkenes: An Efficient, Highly Diastereoselective Approach to Nitrocyclopentanols

(2010) Gregory R. Boyce et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ynamides: Versatile Tools in Organic Synthesis

(2010) Gwilherm Evano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Inhibition of monoamine oxidase by selected C5- and C6-substituted isatin analogues

(2010) Clarina I. Manley-King et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Site-specific introduction of gold-carbenoids by intermolecular oxidation of ynamides or ynol ethers

(2010) Paul W. Davies et al.   CHEMICAL COMMUNICATIONS

Ynamides: A Modern Functional Group for the New Millennium

(2010) Kyle A. DeKorver et al.   CHEMICAL REVIEWS

Synthesis and in vitro antimycobacterial activity of 8-OCH3 ciprofloxacin methylene and ethylene isatin derivatives

(2010) Lian-Shun Feng et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A stereoselective intramolecular cyclopropanation via a de novo class of push–pull carbenes derived from DMDO-epoxidations of chiral ynamides

(2010) Hongyan Li et al.   NEW JOURNAL OF CHEMISTRY

Highly Enantioselective Pictet-Spengler Reactions with α-Ketoamide-Derived Ketimines: Access to an Unusual Class of Quaternary α-Amino Amides

(2009) Farhan R. Bou-Hamdan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Retinoid receptor subtype-selective modulators through synthetic modifications of RARγ agonists

(2009) Susana Álvarez et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Alkyne activation with Brønsted acids, iodine, or gold complexes, and its fate leading to synthetic application

(2009) Yoshinori Yamamoto et al.   CHEMICAL COMMUNICATIONS

QSAR study of isatin analogues as in vitro anti-cancer agents

(2009) Razieh Sabet et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cr(III)(salen)Cl Catalyzed Enantioselective Intramolecular Addition of Tertiary Enamides to Ketones: A General Access to Enantioenriched 1H-Pyrrol-2(3H)-one Derivatives Bearing a Hydroxylated Quaternary Carbon Atom

(2009) Luo Yang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Synthesis of SM-130686 Based on the Development of Asymmetric Cu(I)F Catalysis To Access 2-Oxindoles Containing a Tetrasubstituted Carbon

(2009) Daisuke Tomita et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dioxygen Activation under Ambient Conditions: Cu-Catalyzed Oxidative Amidation−Diketonization of Terminal Alkynes Leading to α-Ketoamides

(2009) Chun Zhang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Molecular Iodine-Mediated Cyclization of Tethered Heteroatom-Containing Alkenyl or Alkynyl Systems

(2009) Malose Jack Mphahlele   MOLECULES

Palladium-catalysed selective aminocarbonylation of 1′,4-diiodostyrene

(2009) Antal Szilágyi et al.   TETRAHEDRON

Synthesis of Diastereomers of Complestatin and Chloropeptin I: Substrate-Dependent Atropstereoselectivity of the Intramolecular Suzuki–Miyaura Reaction

(2008) Yanxing Jia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Microwave-assisted efficient oxidation of internal alkynes to 1,2-diaryldiketones with DMSO/I2

(2008) Min Chen et al.   JOURNAL OF CHEMICAL SCIENCES

Design and Synthesis of a Novel Series ofN-Alkyl Isatin Acylhydrazone Derivatives that Act as Selective Cannabinoid Receptor 2 Agonists for the Treatment of Neuropathic Pain

(2008) Philippe Diaz et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of α-Keto-Imides via Oxidation of Ynamides

(2008) Ziyad F. Al-Rashid et al.   JOURNAL OF ORGANIC CHEMISTRY

Amide Synthesis from Alcohols and Amines by the Extrusion of Dihydrogen

(2008) Lars Ulrik Nordstrøm et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Reactive Intermediates from DMDO Oxidation of Ynamides. Trapping of a de novo Chiral Push−Pull Carbene via Cyclopropanation

(2008) Ziyad F. Al-Rashid et al.   ORGANIC LETTERS

Synthesis of Functionalized Oxazolones by a Sequence of Cu(II)- and Au(I)-Catalyzed Transformations

(2008) Florin M. Istrate et al.   ORGANIC LETTERS

Palladium-catalysed aminocarbonylation of iodoarenes and iodoalkenes with aminophosphonate as N-nucleophile

(2008) Attila Takács et al.   TETRAHEDRON