Synthesis of 10-Methylacridin-9(10H)-ones through Cu-Catalyzed Intramolecular Oxidative C(sp2)-H Amination of 2-(Methylamino)benzophenones

Overcoming the “Oxidant Problem”: Strategies to Use O2 as the Oxidant in Organometallic C–H Oxidation Reactions Catalyzed by Pd (and Cu)

(2012) Alison N. Campbell et al.   ACCOUNTS OF CHEMICAL RESEARCH

Palladium-Catalyzed Oxidation of Unsaturated Hydrocarbons Using Molecular Oxygen

(2012) Wanqing Wu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Palladium-catalyzed allylic C–H amination of alkenes with N-fluorodibenzenesulfonimide: water plays an important role

(2012) Tao Xiong et al.   CHEMICAL COMMUNICATIONS

Ruthenium(iv) porphyrin catalyzed phosphoramidation of aldehydes with phosphoryl azides as a nitrene source

(2012) Wenbo Xiao et al.   CHEMICAL COMMUNICATIONS

Copper-catalyzed intramolecular direct amination of sp2 C–H bonds for the synthesis of N-aryl acridones

(2012) Wang Zhou et al.   CHEMICAL COMMUNICATIONS

Recent advances in transition-metal catalyzed reactions using molecular oxygen as the oxidant

(2012) Zhuangzhi Shi et al.   CHEMICAL SOCIETY REVIEWS

Recent advances in copper-catalyzed dehydrogenative functionalization via a single electron transfer (SET) process

(2012) Chun Zhang et al.   CHEMICAL SOCIETY REVIEWS

[Ru(TPP)CO]-Catalysed Intramolecular Benzylic CH Bond Amination, Affording Phenanthridine and Dihydrophenanthridine Derivatives

(2012) Daniela Intrieri et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Catalyzed Intramolecular Oxidative CH Functionalization and CN Formation of 2-Aminobenzophenones: Unusual Pseudo-1,2-Shift of the Substituent on the Aryl Ring

(2012) Pang-Chi Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Formation of Acridones by Ethylene Extrusion in the Reaction of Arynes with β-Lactams and Dihydroquinolinones

(2012) Yuesi Fang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(II) Triflate Catalyzed Amination and Aziridination of 2-Alkyl Substituted 1,3-Dicarbonyl Compounds

(2012) Thi My Uyen Ton et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Aerobic [3+2]-Annulation of N-Alkenyl Amidines

(2012) Yi-Feng Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

CuI-Mediated Sequential Iodination/Cycloetherification of o-Arylphenols: Synthesis of 2- or 4-Iododibenzofurans and Mechanistic Studies

(2012) Jiaji Zhao et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of Purine-Fused Polycyclics

(2012) Gui-Rong Qu et al.   ORGANIC LETTERS

Total Synthesis of (−)-Kaitocephalin Based on a Rh-Catalyzed C–H Amination

(2012) Keisuke Takahashi et al.   ORGANIC LETTERS

Insight into Mechanistic Features of Ruthenium(II)–Pybox-Catalyzed C–H Amination

(2012) Djamaladdin G. Musaev et al.   ORGANOMETALLICS

Synthesis of novel heme-interacting acridone derivatives to prevent free heme-mediated protein oxidation and degradation

(2011) Chinmay Pal et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Observation and Mechanistic Study of Facile CO Bond Formation between a Well-Defined Aryl-Copper(III) Complex and Oxygen Nucleophiles

(2011) Lauren M. Huffman et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Fluorinated Benzophenones, Xanthones, Acridones, and Thioxanthones by Iterative Nucleophilic Aromatic Substitution

(2011) Zachary R. Woydziak et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Direct Oxidative C–H Amination of Benzoxazoles with Formamides or Secondary Amines under Mild Conditions

(2011) Yaming Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed C−H Aminations of Anilides withN-Fluorobenzenesulfonimide

(2011) Kai Sun et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mechanistic Understanding of the Unexpected Meta Selectivity in Copper-Catalyzed Anilide C–H Bond Arylation

(2011) Bo Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Journey Under the Sea: The Quest for Marine Anti-Cancer Alkaloids

(2011) Rita Tohme et al.   MOLECULES

Palladium-Catalyzed Oxidative C–H Bond Coupling of Steered Acetanilides and Aldehydes: A Facile Access toortho-Acylacetanilides

(2011) Yinuo Wu et al.   ORGANIC LETTERS

Ruthenium-Catalyzed γ-Carbolinium Ion Formation from Aryl Azides; Synthesis of Dimebolin

(2011) Huijun Dong et al.   ORGANIC LETTERS

Palladium-/Copper-Catalyzed Regioselective Amination and Chloroamination of Indoles

(2011) Xue-Yuan Liu et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed Intermolecular Direct Amination of Aromatic C–H Bonds with N-Chloroamines

(2011) Ka-Ho Ng et al.   ORGANIC LETTERS

Rhodium-Catalyzed C–H Amination. An Enabling Method for Chemical Synthesis

(2011) J. Du Bois   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Palladium-Catalyzed Aerobic Dehydrogenative Cross-Coupling of Polyfluoroarenes with Thiophenes: Facile Access to Polyfluoroarene–Thiophene Structure

(2011) Chun-Yang He et al.   ORGANOMETALLICS

Remote amide-directed palladium-catalyzed benzylic C–H amination with N-fluorobenzenesulfonimide

(2010) Tao Xiong et al.   CHEMICAL COMMUNICATIONS

Synthesis of New Acridone Derivatives, Inhibitors of NS3 Helicase, Which Efficiently and Specifically Inhibit Subgenomic HCV Replication

(2010) Anna Stankiewicz-Drogoń et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Direct Intramolecular C−H Amination Reaction Cocatalyzed by Copper(II) and Iron(III) as Part of an Efficient Route for the Synthesis of Pyrido[1,2-a]benzimidazoles fromN-Aryl-2-aminopyridines

(2010) Honggen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A New Entry of Amination Reagents for Heteroaromatic C−H Bonds: Copper-Catalyzed Direct Amination of Azoles with Chloroamines at Room Temperature

(2010) Tsuyoshi Kawano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Scope and Mechanism of Allylic C−H Amination of Terminal Alkenes by the Palladium/PhI(OPiv)2Catalyst System: Insights into the Effect of Naphthoquinone

(2010) Guoyin Yin et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Room Temperature Palladium-Catalyzed Decarboxylativeortho-Acylation of Acetanilides with α-Oxocarboxylic Acids

(2010) Ping Fang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Oxidative Amination of Benzoxazoles via C−H and C−N Bond Activation: A New Strategy for Using Tertiary Amines as Nitrogen Group Sources

(2010) Shengmei Guo et al.   ORGANIC LETTERS

Pd(II)-catalyzed synthesis of indoles from α-aryloxime O-pentafluorobenzoates via intramolecular aromatic C–H amination

(2010) Shunsuke Chiba et al.   TETRAHEDRON

Search for MDR modulators: Design, syntheses and evaluations of N-substituted acridones for interactions with p-glycoprotein and Mg2+

(2009) Palwinder Singh et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Catalytic C–H amination: recent progress and future directions

(2009) Florence Collet et al.   CHEMICAL COMMUNICATIONS

Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor

(2009) Giuseppe Manfroni et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Mediated Amidation of Heterocyclic and Aromatic C−H Bonds

(2009) Qiu Wang et al.   ORGANIC LETTERS

Direct Amination of Azoles via Catalytic C−H, N−H Coupling

(2009) Daiki Monguchi et al.   ORGANIC LETTERS

Insertion of Benzene Rings into the Amide Bond: One-Step Synthesis of Acridines and Acridones from Aryl Amides

(2009) Didier G. Pintori et al.   ORGANIC LETTERS

Total synthesis of (±)-megistophylline I

(2009) Yuko Nishihama et al.   TETRAHEDRON LETTERS

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Copper-Catalyzed Aerobic Oxidative Amidation of Terminal Alkynes:  Efficient Synthesis of Ynamides

(2008) Tetsuya Hamada et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic C–H functionalization by metal carbenoid and nitrenoid insertion

(2008) Huw M. L. Davies et al.   NATURE

Stereoselective Rhodium-Catalyzed Imination of Sulfides

(2008) Florence Collet et al.   ORGANIC LETTERS

A mechanistic analysis of the Rh-catalyzed intramolecular C–H amination reaction

(2008) Kristin Williams Fiori et al.   TETRAHEDRON