Molecular imaging of σ receptors: synthesis and evaluation of the potent σ1 selective radioligand [18F]fluspidine

System-Dependent Outcomes during the Evaluation of Drug Candidates as Inhibitors of Cytochrome P450 (CYP) and Uridine Diphosphate Glucuronosyltransferase (UGT) Enzymes: Human Hepatocytes versus Liver Microsomes versus Recombinant Enzymes

(2010) Andrew Parkinson et al.   Drug Metabolism and Pharmacokinetics

Synthesis of spirocyclic σ1 receptor ligands as potential PET radiotracers, structure–affinity relationships and in vitro metabolic stability

(2009) Eva Große Maestrup et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and Pharmacological Evaluation of SNC80 Analogues with a Bridged Piperazine Ring

(2009) Ralph Holl et al.   ChemMedChem

Evaluation of Spirocyclic 3-(3-Fluoropropyl)-2-benzofurans as σ1Receptor Ligands for Neuroimaging with Positron Emission Tomography

(2009) Eva Große Maestrup et al.   JOURNAL OF MEDICINAL CHEMISTRY

When the Endogenous Hallucinogenic Trace Amine N,N-Dimethyltryptamine Meets the Sigma-1 Receptor

(2009) T.-P. Su et al.   Science Signaling

Low density of sigma1 receptors in early Alzheimer’s disease

(2008) Masahiro Mishina et al.   ANNALS OF NUCLEAR MEDICINE

Synthesis and pharmacological evaluation of bicyclic SNC80 analogues with separated benzhydryl moiety

(2008) Bettina Jung et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Novel 4-(4-Aryl)cyclohexyl-1-(2-pyridyl)piperazines as Δ8−Δ7Sterol Isomerase (Emopamil Binding Protein) Selective Ligands with Antiproliferative Activity

(2008) Francesco Berardi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Modulation of glutamatergic transmission by sulfated steroids: Role in fetal alcohol spectrum disorder

(2007) C. Fernando Valenzuela et al.   BRAIN RESEARCH REVIEWS