Efficient tritiation of the translocator protein (18 kDa) selective ligand DPA-714

Regioselective and Stereospecific Deuteration of Bioactive Aza Compounds by the Use of Ruthenium Nanoparticles

(2013) Grégory Pieters et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The potential of carbon-11 and fluorine-18 chemistry: illustration through the development of positron emission tomography radioligands targeting the translocator protein 18 kDa

(2013) Annelaure Damont et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Molecular Imaging of Microglial Activation in Amyotrophic Lateral Sclerosis

(2013) Philippe Corcia et al.   PLoS One

The translocator protein ligand [18F]DPA-714 images glioma and activated microglia in vivo

(2012) Alexandra Winkeler et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Tritium: a coming of age for drug discovery and development ADME studies

(2012) W. J. S. Lockley et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Reactive Astrocytes Overexpress TSPO and Are Detected by TSPO Positron Emission Tomography Imaging

(2012) S. Lavisse et al.   JOURNAL OF NEUROSCIENCE

[18F]DPA-714, [18F]PBR111 and [18F]FEDAA1106—Selective radioligands for imaging TSPO 18kDa with PET: Automated radiosynthesis on a TRACERLAb FX-FN synthesizer and quality controls

(2011) Bertrand Kuhnast et al.   APPLIED RADIATION AND ISOTOPES

Initial evaluation in healthy humans of [18F]DPA-714, a potential PET biomarker for neuroinflammation

(2011) Nicolas Arlicot et al.   NUCLEAR MEDICINE AND BIOLOGY

Translocator protein (18 kDa) (TSPO) as a therapeutic target for neurological and psychiatric disorders

(2010) Rainer Rupprecht et al.   NATURE REVIEWS DRUG DISCOVERY

Radiolabelled Molecules for Imaging the Translocator Protein (18 kDa) Using Positron Emission Tomography

(2009) Frederic Dolle et al.   CURRENT MEDICINAL CHEMISTRY

Simultaneous tritium labelling of two potent 5-HT4 ligands

(2009) Franck Sobrio et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Nuclear imaging of neuroinflammation: a comprehensive review of [11C]PK11195 challengers

(2008) Fabien Chauveau et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

Radiosynthesis of [18F]DPA‐714, a selective radioligand for imaging the translocator protein (18 kDa) with PET

(2008) Annelaure Damont et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS