Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain
Published 2018 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain
Authors
Keywords
-
Journal
ChemMedChem
Volume -, Issue -, Pages -
Publisher
Wiley
Online
2018-08-07
DOI
10.1002/cmdc.201800397
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Neuropathic Pain: Delving into the Oxidative Origin and the Possible Implication of Transient Receptor Potential Channels
- (2018) Cristina Carrasco et al. Frontiers in Physiology
- First dual AK/GSK-3β inhibitors endowed with antioxidant properties as multifunctional, potential neuroprotective agents
- (2017) Simone Brogi et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474
- (2017) Annelot C. M. van Esbroeck et al. SCIENCE
- The FAAH inhibitor URB597 suppresses hippocampal maximal dentate afterdischarges and restores seizure-induced impairment of short and long-term synaptic plasticity
- (2017) Roberto Colangeli et al. Scientific Reports
- Discovery of novel Tetrahydrobenzo[ b ]thiophene and pyrrole based scaffolds as potent and selective CB2 receptor ligands: The structural elements controlling binding affinity, selectivity and functionality
- (2016) Noha A. Osman et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Donepezil-like multifunctional agents: Design, synthesis, molecular modeling and biological evaluation
- (2016) Ming-Yu Wu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer’s Disease Agents
- (2016) Serena Montanari et al. JOURNAL OF MEDICINAL CHEMISTRY
- Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain
- (2016) Margherita Brindisi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structural insights into HDAC6 tubulin deacetylation and its selective inhibition
- (2016) Yasuyuki Miyake et al. Nature Chemical Biology
- Harnessing the pyrroloquinoxaline scaffold for FAAH and MAGL interaction: definition of the structural determinants for enzyme inhibition
- (2016) Margherita Brindisi et al. RSC Advances
- A review of chronic pain impact on patients, their social environment and the health care system
- (2016) María Duenas et al. Journal of Pain Research
- Development of HuperTacrines as Non-Toxic, Cholinesterase Inhibitors for the Potential Treatment of Alzheimer’s Disease
- (2015) Mourad Chioua et al. MINI-REVIEWS IN MEDICINAL CHEMISTRY
- Endocannabinoid Modulation of Predator Stress-Induced Long-Term Anxiety in Rats
- (2015) James Lim et al. NEUROPSYCHOPHARMACOLOGY
- Targeting Dopamine D3 and Serotonin 5-HT1A and 5-HT2A Receptors for Developing Effective Antipsychotics: Synthesis, Biological Characterization, and Behavioral Studies
- (2014) Margherita Brindisi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Targeting the endogenous cannabinoid system to treat neuropathic pain
- (2014) Benjamin K. Lau et al. Frontiers in Pharmacology
- A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity
- (2013) Claudio Battilocchio et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Morphologic Features and Glial Activation in Rat Oxaliplatin-Dependent Neuropathic Pain
- (2013) Lorenzo Di Cesare Mannelli et al. JOURNAL OF PAIN
- Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation
- (2013) Stefania Butini et al. ACS Medicinal Chemistry Letters
- Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties
- (2012) Stefania Butini et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Discovery of Potent Inhibitors of Human and Mouse Fatty Acid Amide Hydrolases
- (2012) Stefania Butini et al. JOURNAL OF MEDICINAL CHEMISTRY
- Oxaliplatin-Induced Neuropathy: Oxidative Stress as Pathological Mechanism. Protective Effect of Silibinin
- (2012) Lorenzo Di Cesare Mannelli et al. JOURNAL OF PAIN
- New Insight into the Central Benzodiazepine Receptor–Ligand Interactions: Design, Synthesis, Biological Evaluation, and Molecular Modeling of 3-Substituted 6-Phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and Related Compounds
- (2011) Maurizio Anzini et al. JOURNAL OF MEDICINAL CHEMISTRY
- Fluoride-Mediated Capture of a Noncovalent Bound State of a Reversible Covalent Enzyme Inhibitor: X-ray Crystallographic Analysis of an Exceptionally Potent α-Ketoheterocycle Inhibitor of Fatty Acid Amide Hydrolase
- (2011) Mauro Mileni et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- The Interactions of the 5-HT3 Receptor with Quipazine-Like Arylpiperazine Ligands. The Journey Track at the End of the First Decade of the Third Millennium
- (2010) Andrea Cappelli et al. CURRENT TOPICS IN MEDICINAL CHEMISTRY
- Novel, Potent, and Selective Quinoxaline-Based 5-HT3Receptor Ligands. 1. Further Structure−Activity Relationships and Pharmacological Characterization
- (2009) Stefania Butini et al. JOURNAL OF MEDICINAL CHEMISTRY
- Specific Targeting of Peripheral Serotonin 5-HT3Receptors. Synthesis, Biological Investigation, and Structure−Activity Relationships
- (2009) Elena Morelli et al. JOURNAL OF MEDICINAL CHEMISTRY
- Tetrahydrolipstatin Analogues as Modulators of Endocannabinoid 2-Arachidonoylglycerol Metabolism
- (2008) Giorgio Ortar et al. JOURNAL OF MEDICINAL CHEMISTRY
- Discovery and Development of Fatty Acid Amide Hydrolase (FAAH) Inhibitors
- (2008) Mark Seierstad et al. JOURNAL OF MEDICINAL CHEMISTRY
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreFind the ideal target journal for your manuscript
Explore over 38,000 international journals covering a vast array of academic fields.
Search