Rational Design of Resorcylic Acid Lactone Analogues as Covalent MNK1/2 Kinase Inhibitors by Tuning the Reactivity of an Enamide Michael Acceptor
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Title
Rational Design of Resorcylic Acid Lactone Analogues as Covalent MNK1/2 Kinase Inhibitors by Tuning the Reactivity of an Enamide Michael Acceptor
Authors
Keywords
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Journal
ChemMedChem
Volume 8, Issue 9, Pages 1483-1494
Publisher
Wiley
Online
2013-08-08
DOI
10.1002/cmdc.201300231
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