Highly Enantioselective Ring-Opening Reactions of Aziridines with Indole and Its Application in the Building of C3-Halogenated Pyrroloindolines

Chiral magnesium(ii)-catalyzed asymmetric ring-opening of meso-aziridines with primary alcohols

(2014) Jun Li et al.   CHEMICAL COMMUNICATIONS

Design of a Combinational Magnesium Catalyst for the Stereocontrolled Cross Reaction of Enones

(2014) Dongxu Yang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Desymmetrization of meso-Aziridines with TMSNCS Using Metal Salts of Novel Chiral Imidazoline–Phosphoric Acid Catalysts

(2014) Shuichi Nakamura et al.   ORGANIC LETTERS

Complex Bioactive Alkaloid-Type Polycycles through Efficient Catalytic Asymmetric Multicomponent Aza-Diels-Alder Reaction of Indoles with Oxetane as Directing Group

(2013) Zhilong Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral-at-Metal Octahedral Iridium Catalyst for the Asymmetric Construction of an All-Carbon Quaternary Stereocenter

(2013) Liang-An Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Site-Specific and Highly Enantioselective γ-Functionalization of Linear α,β-Unsaturated Ketones: Bifunctional Catalytic Strategy

(2013) Dongxu Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Synthesis of Mixed 3,3′-Bisindoles and Their Evaluation as Wnt Signaling Inhibitors

(2013) Takayoshi Arai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (−)-Chimonanthine

(2013) Weiqing Xie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of Indotertine A and Drimentines A, F, and G

(2013) Yu Sun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Palladium(II) Phosphate Catalyzed Three-Component Reactions of Pyrrole, Diazoesters, and Imines

(2013) Dan Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Friedel-Crafts Alkylation/N-Hemiacetalization Cascade Reaction with Indoles

(2013) Hong-Gang Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Hydrogen-Bond-Promoted Palladium Catalysis: Allylic Alkylation of Indoles with Unsymmetrical 1,3-Disubstituted Allyl Acetates Using Chiral Bis(sulfoxide) Phosphine Ligands

(2013) Le Du et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Enantioselective Ring-Opening Reaction ofmeso-Aziridines with α-Isothiocyanato Imides

(2013) Yi-Ming Cao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Lewis Acid Catalyzed SN2-Type Ring Opening of N-Activated Aziridines with Electron-Rich Arenes/Heteroarenes

(2013) Manas K. Ghorai et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent Developments in the Catalytic, Asymmetric Construction of Pyrroloindolines Bearing All-Carbon Quaternary Stereocenters

(2013) Lindsay M. Repka et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Highly Enantioselective Cyclopentannulation of Indoles with Donor–Acceptor Cyclopropanes

(2013) Hu Xiong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Functionalization of Indoles and Pyrroles via an in Situ-Formed Spiro Intermediate

(2013) Chun-Xiang Zhuo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Enantioselective Construction of Trifluoromethylated All-Carbon Quaternary Stereocenters via Nickel-Catalyzed Friedel–Crafts Alkylation Reaction

(2013) Jian-Rong Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Construction of Vicinal All-Carbon Quaternary Stereocenters by Catalytic Asymmetric Alkylation Reaction of 3-Bromooxindoles with 3-Substituted Indoles: Total Synthesis of (+)-Perophoramidine

(2013) Hailong Zhang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Novel Lewis Acid Catalyzed [3 + 3]-Annulation Strategy for the Syntheses of Tetrahydro-β-Carbolines and Tetrahydroisoquinolines

(2013) Shaoyin Wang et al.   ORGANIC LETTERS

Highly Enantioselective Synthesis of Tetrahydrocarbolines via Iridium-Catalyzed Intramolecular Friedel–Crafts Type Allylic Alkylation Reactions

(2013) Qing-Long Xu et al.   ORGANIC LETTERS

Asymmetric Synthesis of Indole Homo-Michael Adducts via Dynamic Kinetic Friedel–Crafts Alkylation with Cyclopropanes

(2013) Steven M. Wales et al.   ORGANIC LETTERS

Organocatalytic Michael Addition of Indoles to Isatylidene-3-acetaldehydes: Application to the Formal Total Synthesis of (−)-Chimonanthine

(2013) Renrong Liu et al.   ORGANIC LETTERS

Enantioselective fluoride ring opening of aziridines enabled by cooperative Lewis acid catalysis

(2013) Julia A. Kalow et al.   TETRAHEDRON

Enantioselective Synthesis and Stereoselective Ring Opening ofN-Acylaziridines

(2012) Jennifer Cockrell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Diastereo- and Enantioselective Synthesis of α-Alkyl Norstatine Derivatives: Catalytic Asymmetric Mannich Reactions of 5H-Oxazol-4-ones

(2012) Depeng Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Dearomatization Reactions

(2012) Chun-Xiang Zhuo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The highly enantioselective addition of indoles and pyrroles to isatins-derived N-Boc ketimines catalyzed by chiral phosphoric acids

(2012) Jingchao Feng et al.   CHEMICAL COMMUNICATIONS

Double Axially Chiral Bisphosphorylimides Catalyzed Highly Enantioselective and Efficient Friedel-Crafts Reaction of Indoles with Imines

(2012) Kun Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of β-Fluoroamines by Lewis Base Catalyzed Hydrofluorination of Aziridines

(2012) Julia A. Kalow et al.   JOURNAL OF ORGANIC CHEMISTRY

Cinchona Alkaloid Amides/Dialkylzinc Catalyzed Enantioselective Desymmetrization of Aziridines with Phosphites

(2012) Masashi Hayashi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Asymmetric Ring Openings of Meso and Terminal Aziridines with Halides Mediated by Chiral 1,2,3-Triazolium Silicates

(2012) Kohsuke Ohmatsu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Synthesis of Tryptophan Derivatives by a Tandem Friedel–Crafts Conjugate Addition/Asymmetric Protonation Reaction

(2012) Madeleine E. Kieffer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Thiourea-catalysed ring opening of episulfonium ions with indole derivatives by means of stabilizing non-covalent interactions

(2012) Song Lin et al.   Nature Chemistry

Highly enantioselective trapping of zwitterionic intermediates by imines

(2012) Huang Qiu et al.   Nature Chemistry

Synthesis of tryptophans by Lewis acid promoted ring-opening of aziridine-2-carboxylates: optimization of protecting group and Lewis acid

(2012) Ilaria Tirotta et al.   TETRAHEDRON LETTERS

Total Synthesis of Indoline Alkaloids: A Cyclopropanation Strategy

(2011) Dan Zhang et al.   ACCOUNTS OF CHEMICAL RESEARCH

Asymmetric Binary Acid Catalysis: A Regioselectivity Switch between Enantioselective 1,2- and 1,4-Addition through Different Counteranions of InIII

(2011) Jian Lv et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of (+)-Gliocladin C Enabled by Visible-Light Photoredox Catalysis

(2011) Laura Furst et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploiting the Electrophilic Properties of Indole Intermediates: New Options in Designing Asymmetric Reactions

(2011) Charles C. J. Loh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalyzed Enantioselective Fluorocyclizations

(2011) Oscar Lozano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Ring-Opening ofmeso-Aziridines with Malonates under Heterodinuclear Rare Earth Metal Schiff Base Catalysis

(2011) Yingjie Xu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifunctional 3,3′-Ph2-BINOL-Mg Catalyzed Direct Asymmetric Vinylogous Michael Addition of α,β-Unsaturated γ-Butyrolactam

(2011) Li Lin et al.   ORGANIC LETTERS

Pd-Catalyzed Asymmetric Allylic Alkylation of Indoles and Pyrroles by Chiral Alkene-Phosphine Ligands

(2011) Ziping Cao et al.   ORGANIC LETTERS

Zinc-Mediated Asymmetric Additions of Dialkylphosphine Oxides to α,β-Unsaturated Ketones andN-Sulfinylimines

(2010) Depeng Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Construction of Spiroindolenines by Ir-Catalyzed Allylic Alkylation Reactions

(2010) Qing-Feng Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Acyl Phosphonates: Good Hydrogen Bond Acceptors and Ester/Amide Equivalents in Asymmetric Organocatalysis

(2010) Hao Jiang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Scalable Total Syntheses ofN-Linked Tryptamine Dimers by Direct Indole−Aniline Coupling: Psychotrimine and Kapakahines B and F

(2010) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Asymmetric Hydrophosphinylation of α,β-UnsaturatedN-Acylpyrroles: Application of Dialkyl Phosphine Oxides in Enantioselective Synthesis of Chiral Phosphine Oxides or Phosphines

(2010) Depeng Zhao et al.   ORGANIC LETTERS

Enantioselective Gold-Catalyzed Allylic Alkylation of Indoles with Alcohols: An Efficient Route to Functionalized Tetrahydrocarbazoles

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Titanium Binolate Catalyzed Aminolysis ofmeso Aziridines: A Highly Enantioselective and Direct Access to 1,2-Diamines

(2009) Saravanan Peruncheralathan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Friedel-Crafts Reactions in Water Using a DNA-Based Catalyst

(2009) Arnold J. Boersma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Regio- and Enantioselective N-Allylation of Indoles

(2009) Levi M. Stanley et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Enantioselective Friedel-Crafts Alkylation of 4,7-Dihydroindoles with Enones Catalyzed by Primary-Secondary Diamines

(2009) Liang Hong et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective Brønsted Acid-CatalyzedN-Acyliminium Cyclization Cascades

(2009) Michael E. Muratore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Practical Asymmetric Conjugate Alkynylation of Meldrum’s Acid-Derived Acceptors: Access to Chiral β-Alkynyl Acids

(2009) Sheng Cui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Enantioselective Friedel−Crafts Alkylation of 4,7-Dihydroindoles with α,β-Unsaturated Aldehydes: An Easy Access to 2-Substituted Indoles

(2009) Liang Hong et al.   ORGANIC LETTERS

Chiral zinc(II) and copper(II)-catalyzed asymmetric ring-opening reactions of meso-epoxides with aniline and indole derivatives

(2009) Masaya Kokubo et al.   TETRAHEDRON

Efficient chirality switching in the asymmetric addition of indole to N-tosylarylimines in the presence of axially chiral cyclometalated bidentate N-heterocyclic carbene palladium(II) complexes

(2009) Zhen Liu et al.   TETRAHEDRON-ASYMMETRY

Chiral Phosphoric Acid Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with Nitroalkenes: Cooperative Effect of 3 Å Molecular Sieves

(2008) Junji Itoh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Aluminum-Catalyzed Asymmetric Alkylations of Pyridyl-Substituted Alkynyl Ketones with Dialkylzinc Reagents

(2008) Donna K. Friel et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Expeditious Synthesis of C(3)−N(1′) Heterodimeric Indolines

(2008) Vinson R. Espejo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Friedel−Crafts Alkylation of Pyrroles with Nitroalkenes Using a Dinuclear Zinc Catalyst

(2008) Barry M. Trost et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ir-Catalyzed Regio- and Enantioselective Friedel–Crafts-Type Allylic Alkylation of Indoles

(2008) Wen-Bo Liu et al.   ORGANIC LETTERS

Synthesis of potent BCRP inhibitor—Ko143

(2008) Yuexian Li et al.   TETRAHEDRON LETTERS

Asymmetric Brønsted Acid Catalysis: Enantioselective Nucleophilic Substitutions and 1,4-Additions

(2007) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION