Formal [4+2] Reaction between 1,3-Diynes and Pyrroles: Gold(I)-Catalyzed Indole Synthesis by Double Hydroarylation

Energy efficiency of heterogeneous catalytic microwave-assisted organic reactions

(2014) Hyejin Cho et al.   GREEN CHEMISTRY

Gold-Catalyzed Cascade Cyclization of (Azido)ynamides: An Efficient Strategy for the Construction of Indoloquinolines

(2014) Yusuke Tokimizu et al.   ORGANIC LETTERS

Synthesis of Indole Derivatives from 2-Alkynylanilines by Means of Gold Catalysis

(2013) Giorgio Abbiati et al.   ISRAEL JOURNAL OF CHEMISTRY

Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds

(2013) Hiroaki Ohno   ISRAEL JOURNAL OF CHEMISTRY

Discovery of 4-{4-[(3R)-3-Methylmorpholin-4-yl]-6-[1-(methylsulfonyl)cyclopropyl]pyrimidin-2-yl}-1H-indole (AZ20): A Potent and Selective Inhibitor of ATR Protein Kinase with Monotherapy in Vivo Antitumor Activity

(2013) Kevin M. Foote et al.   JOURNAL OF MEDICINAL CHEMISTRY

Simple indole alkaloids and those with a non-rearranged monoterpenoid unit

(2013) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

Consecutive Gold(I)-Catalyzed Cyclization Reactions of o-(Buta-1,3-diyn-1-yl-)-Substituted N-Aryl Ureas: A One-Pot Synthesis of Pyrimido[1,6-a]indol-1(2H)-ones and Related Systems

(2013) Phillip P. Sharp et al.   ORGANIC LETTERS

Gold(I)-Catalyzed Macrocyclization of 1,n-Enynes

(2013) Carla Obradors et al.   ORGANIC LETTERS

Synthesis of Pyrroles, Indoles, and Carbazoles through Transition-Metal-Catalyzed CH Functionalization

(2013) Naohiko Yoshikai et al.   Asian Journal of Organic Chemistry

Total Synthesis of (−)-Quinocarcin by Gold(I)-Catalyzed Regioselective Hydroamination

(2012) Hiroaki Chiba et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids

(2012) Arndt W. Schmidt et al.   CHEMICAL REVIEWS

Total Synthesis of (+)-trans-Trikentrin A

(2012) Iris R. M. Tébéka et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ruthenium-Catalyzed Functionalization of Pyrroles and Indoles with Propargyl Alcohols

(2012) Nora Thies et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fused Arene Ring Construction Around Pyrrole To Form 4,7-Disubstitued Indole

(2012) Elżbieta Nojman et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Gold(I)-Catalyzed Regioselective Inter-/Intramolecular Addition Cascade of Di- and Triynes for Direct Construction of Substituted Naphthalenes

(2012) Saori Naoe et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Hydrovinylation of Vinylindoles. A Facile Route to Cyclopenta[g]indole Natural Products (+)-cis-Trikentrin A and (+)-cis-Trikentrin B

(2012) Wang Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hybrid System of Metal/Brønsted Acid Relay Catalysis for the Intramolecular Double Hydroarylation and Cationic Cyclization of Diyne Diethers and Diamines

(2012) Juntae Mo et al.   ORGANIC LETTERS

Recent trends in the synthesis of carbazoles: an update

(2012) Joyeeta Roy et al.   TETRAHEDRON

Indole synthesis – something old, something new

(2012) Martyn Inman et al.   Chemical Science

A New One-Pot Synthesis of Polysubstituted Indoles from Pyrroles and β-Nitroacrylates

(2011) Alessandro Palmieri et al.   ADVANCED SYNTHESIS & CATALYSIS

Structure-based optimization of morpholino-triazines as PI3K and mTOR inhibitors

(2011) Anders Poulsen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Green chemistry: solvent- and metal-free Prins cyclization. Application to sequential reactions

(2011) Damien Clarisse et al.   CHEMICAL COMMUNICATIONS

Structure–Activity Relationships of Carboline and Carbazole Derivatives as a Novel Class of ATP-Competitive Kinesin Spindle Protein Inhibitors

(2011) Tomoki Takeuchi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Direct Synthesis of Fused Indoles by Gold-Catalyzed Cascade Cyclization of Diynes

(2011) Kimio Hirano et al.   JOURNAL OF ORGANIC CHEMISTRY

Gold(I)-Catalyzed Polycyclizations of Polyenyne-Type Anilines Based on Hydroamination and Consecutive Hydroarylation Cascade

(2011) Kimio Hirano et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent advances in indole syntheses: New routes for a classic target

(2011) Rubén Vicente   ORGANIC & BIOMOLECULAR CHEMISTRY

Gold-Catalyzed Three-Component Annulation: Efficient Synthesis of Highly Functionalized Dihydropyrazoles from Alkynes, Hydrazines, and Aldehydes or Ketones

(2011) Yamato Suzuki et al.   ORGANIC LETTERS

4,7-Diaryl indole-based fluorescent chemosensor for iodide ions

(2011) Krishnaswamy R. Rathikrishnan et al.   TETRAHEDRON

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Kinesin Spindle Protein (KSP) Inhibitors with 2,3-Fused Indole Scaffolds

(2010) Shinya Oishi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper catalysis in the construction of indole and benzo[b]furan rings

(2010) Sandro Cacchi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Access to 2,5-Diamidopyrroles and 2,5-Diamidofurans by Au(I)-Catalyzed Double Hydroamination or Hydration of 1,3-Diynes

(2010) Søren Kramer et al.   ORGANIC LETTERS

Highly Efficient and Regioselective Platinum(II)-Catalyzed Tandem Synthesis of Multiply Substituted Indolines and Tetrahydroquinolines

(2009) Xin-Yuan Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and adrenolytic activity of 1-(1H-indol-4-yloxy)-3-(2-(2-methoxy phenoxy)ethylamino)propan-2-ol analogs and its enantiomers. Part 2

(2009) Grażyna Groszek et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Homogeneous Catalytic Hydroamination of Alkynes and Allenes with Ammonia

(2008) Vincent Lavallo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent advances in syntheses of heterocycles and carbocycles via homogeneous gold catalysis. Part 1: Heteroatom addition and hydroarylation reactions of alkynes, allenes, and alkenes

(2008) Hong C. Shen   TETRAHEDRON