Rapid Assembly of Functionalised Spirocyclic Indolines by Palladium-Catalysed Dearomatising Diallylation of Indoles with Allyl Acetate

Rings in Drugs

(2014) Richard D. Taylor et al.   JOURNAL OF MEDICINAL CHEMISTRY

Direct Imine Acylation for Molecular Diversity in Heterocyclic Synthesis

(2014) William P. Unsworth et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium(II)-Catalyzed Efficient C-3 Functionalization of Indoles with Benzylic and Allylic Alcohols under Co-Catalyst, Acid, Base, Additive and External Ligand-Free Conditions

(2013) Debjit Das et al.   ADVANCED SYNTHESIS & CATALYSIS

A Highly Enantioselective Catalytic Mannich Reaction of Indolenines with Ketones

(2013) Dao-Juan Cheng et al.   ADVANCED SYNTHESIS & CATALYSIS

A Rapid Route to Aminocyclopropanes via Carbamatoorganozinc Carbenoids

(2013) Shingo Ishikawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Hydrogen-Bond-Promoted Palladium Catalysis: Allylic Alkylation of Indoles with Unsymmetrical 1,3-Disubstituted Allyl Acetates Using Chiral Bis(sulfoxide) Phosphine Ligands

(2013) Le Du et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

2-(Aryl-sulfonyl)oxetanes as designer 3-dimensional fragments for fragment screening: synthesis and strategies for functionalisation

(2013) Kate F. Morgan et al.   CHEMICAL COMMUNICATIONS

Isocyanide-Based Multicomponent Reactions: Catalyst-Free Stereoselective Construction of Polycyclic Spiroindolines

(2013) Xiang Wang et al.   ORGANIC LETTERS

Palladium Catalyzed Decarboxylative Rearrangement of N-Alloc Indoles

(2013) Jun Chen et al.   ORGANIC LETTERS

Trianion Synthon Approach to Spirocyclic Heterocycles

(2013) Matthew A. Perry et al.   ORGANIC LETTERS

Palladium-Catalyzed Decarboxylative Allylation and Benzylation of N-Alloc and N-Cbz Indoles

(2013) Thomas D. Montgomery et al.   ORGANIC LETTERS

Cation-directed enantioselective synthesis of quaternary-substituted indolenines

(2013) Meiling Li et al.   Chemical Science

Catalytic Diastereo- and Enantioselective Annulations between Transient Nitrosoalkenes and Indoles

(2012) Yu Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries

(2012) Jason T. Lowe et al.   JOURNAL OF ORGANIC CHEMISTRY

Controlled Rearrangement of Lactam-Tethered Allenols with Brominating Reagents: A Combined Experimental and Theoretical Study on α- versus β-Keto Lactam Formation

(2011) Benito Alcaide et al.   CHEMISTRY-A EUROPEAN JOURNAL

Preparation and Synthetic Applications of Azetidines

(2011) F. G. West et al.   HETEROCYCLES

Palladium-Catalyzed C3-Benzylation of Indoles

(2011) Ye Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rapid synthesis of highly functionalised α-amino amides and medium ring lactones using multicomponent reactions of amino alcohols and isocyanides

(2011) Martin Bachman et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Highly Enantioselective Pd-Catalyzed Allylic Alkylation of Indoles Using Sulfur-MOP Ligand

(2011) Takashi Hoshi et al.   ORGANIC LETTERS

Strategies for the synthesis of 2,3-dihydrobenzofurans

(2011) Tom D. Sheppard   JOURNAL OF CHEMICAL RESEARCH

Oxetanes as Versatile Elements in Drug Discovery and Synthesis

(2010) Johannes A. Burkhard et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Alstiphyllanines E–H, picraline and ajmaline-type alkaloids from Alstonia macrophylla inhibiting sodium glucose cotransporter

(2010) Hiroko Arai et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Role of zinc in the development and treatment of mood disorders

(2010) Elise C Cope et al.   CURRENT OPINION IN CLINICAL NUTRITION AND METABOLIC CARE

Diverse Strategies for the Synthesis of the Indoline Scaffold

(2010) Dianyu Liu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Arylcyclopropanes: Properties, Synthesis and Use in Medicinal Chemistry

(2010) Alexandre Gagnon et al.   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Isocyanide based multicomponent reactions of oxazolidines and related systems

(2010) Robert W. Waller et al.   TETRAHEDRON

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

(2009) Frank Lovering et al.   JOURNAL OF MEDICINAL CHEMISTRY

Alstiphyllanines A−D, Indole Alkaloids fromAlstonia macrophylla

(2009) Yusuke Hirasawa et al.   JOURNAL OF NATURAL PRODUCTS

Recent Progress in the Synthesis of 2,3-Dihydrobenzofurans

(2009) Ferruccio Bertolini et al.   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Coupling Isocyanide-Based Multicomponent Reactions with Aliphatic or Acyl Nucleophilic Substitution Processes

(2009) Luca Banfi et al.   SYNLETT

Spirocyclic Oxetanes: Synthesis and Properties

(2008) Georg Wuitschik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel Syntheses of Azetidines and Azetidinones

(2008) Alberto Brandi et al.   CHEMICAL REVIEWS

Multiple Multicomponent Macrocyclizations Including Bifunctional Building Blocks (MiBs) Based on Staudinger and Passerini Three-Component Reactions

(2008) Fredy Leon et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed β-Allylation of 2,3-Disubstituted Indoles

(2008) Natsuko Kagawa et al.   ORGANIC LETTERS

Palladium-catalyzed selective activation of allyl alcohols as allyl cations, allyl anions, and zwitterionic trimethylenemethanes

(2008) Yoshinao Tamaru et al.   PURE AND APPLIED CHEMISTRY

Synthesis of unusually strained spiroheterocyclic ring systems and their exploits in synthesis

(2008) Richard J. Duffy et al.   TETRAHEDRON

Beyond the Ugi reaction: less conventional interactions between isocyanides and iminium species

(2008) Laurent El Kaim et al.   TETRAHEDRON