One-Pot Synthesis of (−)-Oseltamivir and Mechanistic Insights into the Organocatalyzed Michael Reaction

Pot Economy in the Synthesis of Prostaglandin A1and E1Methyl Esters

(2013) Yujiro Hayashi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stoichiometric Reactions of Enamines Derived from Diphenylprolinol Silyl Ethers with Nitro Olefins and Lessons for the Corresponding Organocatalytic Conversions - a Survey

(2013) Dieter Seebach et al.   HELVETICA CHIMICA ACTA

Organocatalytic Michael Reaction of Nitroenamine Derivatives with Aldehydes: Short and Efficient Asymmetric Synthesis of (−)-Oseltamivir

(2012) Jiang Weng et al.   ChemCatChem

EnantioselectiveMichaelAddition of the 2-(1-Ethylpropoxy)acetaldehyde toN-[(1Z)-2-Nitroethenyl]acetamide - Optimization of the Key Step in the Organocatalytic Oseltamivir Synthesis

(2012) Viktória Hajzer et al.   HELVETICA CHIMICA ACTA

Thiol-Free Synthesis of Oseltamivir and Its Analogues via Organocatalytic Michael Additions of Oxyacetaldehydes to 2-Acylaminonitroalkenes

(2012) Július Durmis et al.   SYNTHESIS-STUTTGART

One-Pot High-Yielding Synthesis of the DPP4-Selective Inhibitor ABT-341 by a Four-Component Coupling Mediated by a Diphenylprolinol Silyl Ether

(2011) Hayato Ishikawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Reactions Accelerate the Synthesis of Active Pharmaceutical Ingredients

(2011) Carine Vaxelaire et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of (-)-Oseltamivir by Using a Microreactor in the Curtius Rearrangement

(2011) Hayato Ishikawa et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalyzed Michael Addition of Aldehydes to Nitro Alkenes - Generally Accepted Mechanism Revisited and Revised

(2011) Krystyna Patora-Komisarska et al.   HELVETICA CHIMICA ACTA

Organocatalytic Michael Addition of Aldehydes to Protected 2-Amino-1-Nitroethenes: The Practical Syntheses of Oseltamivir (Tamiflu) and Substituted 3-Aminopyrrolidines

(2010) Shaolin Zhu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

High-Yielding Synthesis of the Anti-Influenza Neuraminidase Inhibitor (−)-Oseltamivir by Two “One-Pot” Sequences

(2010) Hayato Ishikawa et al.   CHEMISTRY-A EUROPEAN JOURNAL

High-Yielding Synthesis of the Anti-Influenza Neuramidase Inhibitor (−)-Oseltamivir by Three “One-Pot” Operations

(2009) Hayato Ishikawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structures of the Reactive Intermediates in Organocatalysis with Diarylprolinol Ethers

(2009) Uroš Grošelj et al.   HELVETICA CHIMICA ACTA

A Short and Practical Synthesis of Oseltamivir Phosphate (Tamiflu) from (−)-Shikimic Acid†

(2009) Liang-Deng Nie et al.   JOURNAL OF ORGANIC CHEMISTRY

Efficient Asymmetric Synthesis of Oseltamivir from d-Mannitol

(2009) Tadakatsu Mandai et al.   SYNLETT

A Concise Synthesis of (−)-Oseltamivir

(2008) Barry M. Trost et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Concise and Flexible Synthesis of the Potent Anti‐Influenza Agents Tamiflu and Tamiphosphor

(2008) Jiun‐Jie Shie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

New, Efficient Synthesis of Oseltamivir Phosphate (Tamiflu) via Enzymatic Desymmetrization of ameso-1,3-Cyclohexanedicarboxylic Acid Diester

(2008) Ulrich Zutter et al.   JOURNAL OF ORGANIC CHEMISTRY

Efficient Short Step Synthesis of Corey's Tamiflu Intermediate

(2008) Nsiama Tienabe Kipassa et al.   ORGANIC LETTERS

A chemoenzymatic synthesis of the anti-influenza agent Tamiflu®

(2008) Maria Matveenko et al.   TETRAHEDRON LETTERS