Syntheses, Receptor Bindings,in vitroandin vivoStabilities and Biodistributions of DOTA-Neurotensin(8-13) Derivatives Containingβ-Amino Acid Residues - A Lesson about the Importance of Animal Experiments

Improved Efficacy of Fosmidomycin against Plasmodium and Mycobacterium Species by Combination with the Cell-Penetrating Peptide Octaarginine

(2013) Christof Sparr et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

G-protein-coupled receptor structure, ligand binding and activation as studied by solid-state NMR spectroscopy

(2013) Xiaoyan Ding et al.   BIOCHEMICAL JOURNAL

Permeation through Phospholipid Bilayers, Skin-Cell Penetration, Plasma Stability, and CD Spectra ofα- andβ-Oligoproline Derivatives

(2013) Beata Kolesinska et al.   CHEMISTRY & BIODIVERSITY

Enantiomeric and Diastereoisomeric (Mixed)L/ D-Octaarginine Derivatives - A Simple Way of Modulating the Properties of Cell-Penetrating Peptides

(2013) Nirupam Purkayastha et al.   CHEMISTRY & BIODIVERSITY

Impact of the Proline Residue on Ligand Binding of Neurotensin Receptor 2 (NTS2)-Selective Peptide-Peptoid Hybrids

(2013) Cornelia Held et al.   ChemMedChem

Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand

(2012) Cornelia Held et al.   ChemMedChem

Structure of the agonist-bound neurotensin receptor

(2012) Jim F. White et al.   NATURE

Novel DOTA-Neurotensin Analogues for111In Scintigraphy and68Ga PET Imaging of Neurotensin Receptor-Positive Tumors

(2011) Faisal Alshoukr et al.   BIOCONJUGATE CHEMISTRY

On the Terminal Homologation of Physiologically Active Peptides as a Means of Increasing Stability in Human Serum - Neurotensin, Opiorphin, B27-KK10 Epitope, NPY

(2011) Dieter Seebach et al.   CHEMISTRY & BIODIVERSITY

On the Mechanism of Eukaryotic Cell Penetration by α- and β-Oligoarginines - Targeting Infected Erythro­cytes

(2011) Faustin Kamena et al.   CHEMISTRY & BIODIVERSITY

Discovery of Highly Potent and Neurotensin Receptor 2 Selective Neurotensin Mimetics

(2011) Jürgen Einsiedel et al.   JOURNAL OF MEDICINAL CHEMISTRY

Radical arylation of tyrosine and its application in the synthesis of a highly selective neurotensin receptor 2 ligand

(2011) Gerald Pratsch et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The role of neurotensin in physiologic and pathologic processes

(2011) W Conan Mustain et al.   Current Opinion in Endocrinology Diabetes and Obesity

Heterologous high yield expression and purification of neurotensin and its functional fragment in Escherichia coli

(2010) Satita Tapaneeyakorn et al.   PROTEIN EXPRESSION AND PURIFICATION

Synthesis of a 68Ga-Labeled Peptoid−Peptide Hybrid for Imaging of Neurotensin Receptor Expression in Vivo

(2010) Simone Maschauer et al.   ACS Medicinal Chemistry Letters

Labeling and Glycosylation of Peptides Using Click Chemistry: A General Approach to 18F-Glycopeptides as Effective Imaging Probes for Positron Emission Tomography

(2009) Simone Maschauer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Constitutive Dimerization of the G-Protein Coupled Receptor, Neurotensin Receptor 1, Reconstituted into Phospholipid Bilayers

(2009) Peter J. Harding et al.   BIOPHYSICAL JOURNAL

NMR-Solution Structures and Affinities for the Human Somatostatin G-Protein-Coupled Receptors hsst1–5 of CF3 Derivatives of Sandostatin® (Octreotide)

(2009) Dieter Seebach et al.   HELVETICA CHIMICA ACTA

The Replacement of His(4) in Angiotensin IV by Conformationally Constrained Residues Provides Highly Potent and Selective Analogues

(2009) Aneta Lukaszuk et al.   JOURNAL OF MEDICINAL CHEMISTRY

Ligands bind to Sortilin in the tunnel of a ten-bladed β-propeller domain

(2009) Esben M Quistgaard et al.   NATURE STRUCTURAL & MOLECULAR BIOLOGY

β-Peptidic Peptidomimetics

(2008) Dieter Seebach et al.   ACCOUNTS OF CHEMICAL RESEARCH

Peptide backbone modifications on the C-terminal hexapeptide of neurotensin

(2008) Jürgen Einsiedel et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

β-Homo-amino Acid Scan of Angiotensin IV

(2008) Aneta Lukaszuk et al.   JOURNAL OF MEDICINAL CHEMISTRY

Artificial Chemokines: Combining Chemistry and Molecular Biology for the Elucidation of Interleukin-8 Functionality

(2008) Ralf David et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Preparation of β²-Amino Acid Derivatives for β-Peptide Synthesis

(2008) Dieter Seebach et al.   SYNTHESIS-STUTTGART

The Synthesis and Chelation Chemistry of DOTA−Peptide Conjugates

(2007) Luis M. De León-Rodríguez et al.   BIOCONJUGATE CHEMISTRY