2-Aroylindoles from o-bromochalcones via Cu(i)-catalyzed SNAr with an azide and intramolecular nitrene C–H insertion

Synthesis of pseudo-indoxyl derivatives via sequential Cu-catalyzed SNAr and Smalley cyclization

(2013) Yogesh Goriya et al.   CHEMICAL COMMUNICATIONS

Recyclable copper catalyzed nitrogenation of biphenyl halides: a direct approach to carbazoles

(2013) Yang Ou et al.   CHEMICAL COMMUNICATIONS

Palladium-catalyzed decarboxylative C2-acylation of indoles with α-oxocarboxylic acids

(2013) Changduo Pan et al.   CHEMICAL COMMUNICATIONS

Iodine-mediated intramolecular amination of ketones: the synthesis of 2-acylindoles and 2-acylindolines by tuning N-protecting groups

(2013) Wen-Chao Gao et al.   CHEMICAL COMMUNICATIONS

Evaluation of viability of halogen⋯O2N interactions: Insight from crystal packing in a series of isomeric halo and nitro substituted triaryl compounds with modular positioning of halogen and NO2 groups

(2013) C. V. Ramana et al.   CRYSTENGCOMM

Biomedical Importance of Indoles

(2013) Nagendra Kaushik et al.   MOLECULES

Simple indole alkaloids and those with a non-rearranged monoterpenoid unit

(2013) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

Cu(OTf)2-Catalyzed Synthesis of 2,3-Disubstituted Indoles and 2,4,5-Trisubstituted Pyrroles from α-Diazoketones

(2013) B. V. Subba Reddy et al.   ORGANIC LETTERS

Design, synthesis and antiproliferative activity of indole analogues of indanocine

(2013) Gemma A. Tunbridge et al.   MedChemComm

Synthesis of Indoles through Highly Efficient Cascade Reactions of Sulfur Ylides and N-(ortho-Chloromethyl)aryl Amides

(2012) Qing-Qing Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium-catalyzed oxidative C2-acylation of indoles with aryl and alkyl aldehydes

(2012) Bing Zhou et al.   CHEMICAL COMMUNICATIONS

Progress in palladium-based catalytic systems for the sustainable synthesis of annulated heterocycles: a focus on indole backbones

(2012) Mélanie Platon et al.   CHEMICAL SOCIETY REVIEWS

Indole synthesis – something old, something new

(2012) Martyn Inman et al.   Chemical Science

Synthesis, antimicrobial, antimycobacterial and structure–activity relationship of substituted pyrazolo-, isoxazolo-, pyrimido- and mercaptopyrimidocyclohepta[b]indoles

(2011) Ezhumalai Yamuna et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of conolidine, a potent non-opioid analgesic for tonic and persistent pain

(2011) Michael A. Tarselli et al.   Nature Chemistry

Consecutive Condensation, C–N and N–N Bond Formations: A Copper- Catalyzed One-Pot Three-Component Synthesis of 2H-Indazole

(2011) Manian Rajesh Kumar et al.   ORGANIC LETTERS

One-pot aromatic amination based on carbon–nitrogen coupling reaction between aryl halides and azido compounds

(2011) Toshihide Maejima et al.   TETRAHEDRON

CuI-catalyzed photochemical or thermal reactions of 3-(2-azidobenzylidene)lactams. Application to the synthesis of fused indoles

(2010) Zongjun Shi et al.   CHEMICAL COMMUNICATIONS

Copper catalysis in the construction of indole and benzo[b]furan rings

(2010) Sandro Cacchi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The [Cu]-catalyzed SNAR reactions: direct amination of electron deficient aryl halides with sodium azide and the synthesis of arylthioethers under Cu(II)–ascorbate redox system

(2010) Yogesh Goriya et al.   TETRAHEDRON

Molecular and biochemical pharmacology of the histamine H4 receptor

(2009) Rob Leurs et al.   BRITISH JOURNAL OF PHARMACOLOGY

Microwave-assisted Cadogan reaction for the synthesis of 2-aryl-2H-indazoles, 2-aryl-1H-benzimidazoles, 2-carbonylindoles, carbazole, and phenazine

(2009) Evelyn Cuevas Creencia et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Palladium-Catalyzed Domino C,N-Coupling/Carbonylation/Suzuki Coupling Reaction: An Efficient Synthesis of 2-Aroyl-/Heteroaroylindoles

(2009) Martin Arthuis et al.   ORGANIC LETTERS

Dirhodium(II)-Catalyzed Intramolecular CH Amination of Aryl Azides

(2008) Meihua Shen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Evaluation of a chemical library of small-molecule Dishevelled antagonists that suppress tumor growth by down-regulating T-cell factor–mediated transcription

(2008) Liang You et al.   MOLECULAR CANCER THERAPEUTICS