Highly N2-Selective Palladium-Catalyzed Arylation of 1,2,3-Triazoles

The First Large-Scale Synthesis of MK-4305: A Dual Orexin Receptor Antagonist for the Treatment of Sleep Disorder

(2011) Carl A. Baxter et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Novel pyrrole- and 1,2,3-triazole-based 2,3-oxidosqualene cyclase inhibitors

(2010) Takumi Watanabe et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia

(2010) Christopher D. Cox et al.   JOURNAL OF MEDICINAL CHEMISTRY

Aerobic Hydroxylation ofN-Borylenamine: Triethylborane-Mediated Hydroxyalkylation of α,β-Unsaturated Oxime Ether

(2009) Masafumi Ueda et al.   ORGANIC LETTERS

Bromo-DirectedN-2 Alkylation ofNH-1,2,3-Triazoles: Efficient Synthesis of Poly-Substituted 1,2,3-Triazoles

(2009) Xiao-jun Wang et al.   ORGANIC LETTERS

Highly RegioselectiveN-2 Arylation of 4,5-Dibromo-1,2,3-triazole: Efficient Synthesis of 2-Aryltriazoles

(2009) Xiao-jun Wang et al.   ORGANIC LETTERS

Conformational control in the regioselective synthesis of N-2-substituted-1,2,3-triazoles

(2008) Yunfeng Chen et al.   CHEMICAL COMMUNICATIONS

Efficient Synthesis of 2-Substituted-1,2,3-triazoles

(2008) Jarosław Kalisiak et al.   ORGANIC LETTERS

Efficient Synthesis ofN-2-Aryl-1,2,3-Triazole Fluorophores via Post-Triazole Arylation

(2008) Yuxiu Liu et al.   ORGANIC LETTERS