Convenient and Reliable Routes Towards 2-Aminothiazoles: Palladium-CatalyzedversusCopper-Catalyzed Aminations of Halothiazoles

Synthesis of Internal Alkynes through the Pd-Catalyzed Coupling of Heteroaryl Halides with Terminal Alkynes

(2013) Linhua Lu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Preparation, antibacterial evaluation and preliminary structure–activity relationship (SAR) study of benzothiazol- and benzoxazol-2-amine derivatives

(2012) Liang Ouyang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of phenothiazines via ligand-free CuI-catalyzed cascade C–S and C–N coupling of aryl ortho-dihalides and ortho-aminobenzenethiols

(2012) Chuan Dai et al.   CHEMICAL COMMUNICATIONS

Palladium Catalyzed Coupling of Tosylhydrazones with Aryl and Heteroaryl Halides in the Absence of External Ligands: Synthesis of Substituted Olefins

(2012) Devi Prasan Ojha et al.   JOURNAL OF ORGANIC CHEMISTRY

High-valent organometallic copper and palladium in catalysis

(2012) Amanda J. Hickman et al.   NATURE

Palladium-Catalyzed N-Arylation of 2-Aminothiazoles

(2012) Meredeth A. McGowan et al.   ORGANIC LETTERS

Copper-Catalyzed Sequential Ullmann N-Arylation and Aerobic Oxidative C–H Amination: A Convenient Route to Indolo[1,2-c]quinazoline Derivatives

(2012) Peng Sang et al.   ORGANIC LETTERS

Copper-catalyzed oxidative C‒H, N‒H coupling of azoles and thiophenes

(2012) Shinobu Mitsuda et al.   TETRAHEDRON

Novel Solid-Phase Parallel Synthesis of N-Substituted-2-aminobenzo [d]thiazole Derivatives via Cyclization Reactions of 2-Iodophenyl Thiourea Intermediate Resin

(2012) Seul-Gi Kim et al.   ACS Combinatorial Science

A one-pot strategy for the synthesis of 2-aminobenzothiazole in water by copper catalysis

(2012) Nilufa Khatun et al.   RSC Advances

Synthesis of 2-Aminobenzothiazoles via Copper(I)-Catalyzed Cross-Coupling with Part-Per-Million Catalyst Loadings

(2011) Ya-Lei Sun et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of 5-arylated N-arylthiazole-2-amines as potential skeletal muscle cell differentiation promoters

(2011) Michael Schnürch et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Direct N-alkylation of amino-azoles with alcohols catalyzed by an iridium complex/base system

(2011) Feng Li et al.   CHEMICAL COMMUNICATIONS

Synthesis of Diheteroarylamine Ligands by Palladium-Catalyzed Mono- and Diamination of Dichlorohetero­arenes with Heteroarenamines

(2011) Daniel Samson et al.   HELVETICA CHIMICA ACTA

Direct, Metal-Free Amination of Heterocyclic Amides/Ureas with NH-Heterocycles and N-Substituted Anilines in POCl3

(2011) Xiaohu Deng et al.   JOURNAL OF ORGANIC CHEMISTRY

A Protocol to 2-Aminobenzimidazoles via Copper-Catalyzed Cascade Addition and Cyclization ofo-Haloanilines and Carbodiimides

(2011) Fei Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Merrifield resin supported phenanthroline–Cu(I): a highly efficient and recyclable catalyst for the synthesis of 2-aminobenzothiazoles via the reaction of 2-haloanilines with isothiocyanates

(2011) Jin Yang et al.   TETRAHEDRON

Domino Condensation/S-Arylation/Heterocyclization Reactions: Copper-Catalyzed Three-Component Synthesis of 2-N-Substituted Benzothiazoles

(2010) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 2-aminobenzothiazole via FeCl3-catalyzed tandem reaction of 2-iodoaniline with isothiocyanate in water

(2010) Qiuping Ding et al.   GREEN CHEMISTRY

An economically and environmentally sustainable synthesis of 2-aminobenzothiazoles and 2-aminobenzoxazoles promoted by water

(2010) Xinying Zhang et al.   GREEN CHEMISTRY

Metal-Free Synthesis of 2-Substituted (N, O, C) Benzothiazoles via an Intramolecular C−S Bond Formation

(2010) Enguang Feng et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Copper-Catalyzed Annulation of 2-Formylazoles witho-Aminoiodoarenes

(2010) Jonathan T. Reeves et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition-Metal-FreeO-,S-, andN-Arylation of Alcohols, Thiols, Amides, Amines, and Related Heterocycles†

(2010) Rafael Cano et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemospecific and ligand free CuI catalysed heterogeneous N-arylation of amines with diheteroaryl halides at room temperature

(2010) Sanjeev K. Verma et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Aza-Fused Polycyclic Quinolines through Copper-Catalyzed Cascade Reactions

(2010) Qian Cai et al.   ORGANIC LETTERS

Domino N−H/C−H Bond Activation: Copper-Catalyzed Synthesis of Nitrogen-Bridgehead Heterocycles Using Azoles and 1,4-Dihalo-1,3-dienes

(2010) Qian Liao et al.   ORGANIC LETTERS

An efficient copper(II)-catalyzed synthesis of benzothiazoles through intramolecular coupling-cyclization of N-(2-chlorophenyl)benzothioamides

(2010) E.A. Jaseer et al.   TETRAHEDRON LETTERS

Iron-Catalyzed Tandem Reactions of 2-Halobenzenamines with Isothiocyanates Leading to 2-Aminobenzothiazoles

(2009) Jing-Wen Qiu et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of 2-fluoroalkylbenzimidazoles via copper(i)-catalyzed tandem reactions

(2009) Jiangtao Zhu et al.   CHEMICAL COMMUNICATIONS

A General Palladium-Catalyzed Amination of Aryl Halides with Ammonia

(2009) Thomas Schulz et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ligand-Free Iron/Copper-Cocatalyzed Amination of Aryl Iodides

(2009) Xiao-Feng Wu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis ofN-Substituted-2-Aminobenzothiazoles by Ligand-Free Copper(I)-Catalyzed Cross-Coupling Reaction of 2-Haloanilines with Isothiocyanates

(2009) Guodong Shen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Ligand-free iron/copper cocatalyzed N-arylations of aryl halides with amines under microwave irradiation

(2009) Diliang Guo et al.   GREEN CHEMISTRY

Synthesis of 2-Aminobenzothiazole via Copper(I)-Catalyzed Tandem Reaction of 2-Iodobenzenamine with Isothiocyanate

(2009) Qiuping Ding et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Highly Functional Group Tolerance in Copper-CatalyzedN-Arylation of Nitrogen-Containing Heterocycles under Mild Conditions

(2009) Liangbo Zhu et al.   JOURNAL OF ORGANIC CHEMISTRY

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

(2009) Prasenjit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Cascade Addition/Cyclization: An Efficient and Versatile Synthesis ofN-Substituted 2-Heterobenzimidazoles

(2009) Xin Lv et al.   JOURNAL OF ORGANIC CHEMISTRY

An Efficient Process for Pd-Catalyzed C−N Cross-Coupling Reactions of Aryl Iodides: Insight Into Controlling Factors

(2009) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Efficient One-Pot Copper-Catalyzed Approach to Isoquinolin-1(2H)-one Derivatives

(2009) Feng Wang et al.   ORGANIC LETTERS

Nucleophilic Capture of the Imino-Quinone Methide Type Intermediates Generated from 2-Aminothiazol-5-yl Carbinols

(2009) Mark G. Saulnier et al.   ORGANIC LETTERS

A straightforward copper-free palladium methodology for the selective alkynylation of a wide variety of S-, O-, and N-based mono- and diheterocyclic bromides and chlorides

(2009) Samer Saleh et al.   TETRAHEDRON

Copper-catalyzed tandem reactions of 2-halobenzenamines with isothiocyanates under ligand- and base-free conditions

(2009) Yan-Jin Guo et al.   TETRAHEDRON LETTERS

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Simple and Efficient Approach to Quinazolinones under Mild Copper-Catalyzed Conditions

(2008) Xiaowei Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides

(2008) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Reactive, General and Long-Lived Catalysts for Palladium-Catalyzed Amination of Heteroaryl and Aryl Chlorides, Bromides, and Iodides: Scope and Structure–Activity Relationships

(2008) Qilong Shen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Carbon–heteroatom bond formation catalysed by organometallic complexes

(2008) John F. Hartwig   NATURE

Synthesis of Indolines via a Domino Cu-Catalyzed Amidation/Cyclization Reaction

(2008) Ana Minatti et al.   ORGANIC LETTERS

Assembly of Isoquinolines via CuI-Catalyzed Coupling of β-Keto Esters and 2-Halobenzylamines

(2008) Bao Wang et al.   ORGANIC LETTERS

Unexpected Formation of Benzothiazoles in the Synthesis of New Heterocycles: Benzo-1,2,4-dithiazines

(2008) Dagmar Fajkusova et al.   SYNTHESIS-STUTTGART

Novel azolyl-(phenylmethyl)]aryl/heteroarylamines: Potent CYP26 inhibitors and enhancers of all-trans retinoic acid activity in neuroblastoma cells

(2007) Mohamed Sayed Gomaa et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of N-benzothiazol-2-yl-amides by a copper-catalyzed intramolecular cyclization process

(2007) Junke Wang et al.   TETRAHEDRON LETTERS