Identification of novel cell-impermeant fluorescent substrates for testing the function and drug interaction of Organic Anion-Transporting Polypeptides, OATP1B1/1B3 and 2B1
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Title
Identification of novel cell-impermeant fluorescent substrates for testing the function and drug interaction of Organic Anion-Transporting Polypeptides, OATP1B1/1B3 and 2B1
Authors
Keywords
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Journal
Scientific Reports
Volume 8, Issue 1, Pages -
Publisher
Springer Nature
Online
2018-02-02
DOI
10.1038/s41598-018-20815-1
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Note: Only part of the references are listed.- Intestinal Drug Interactions Mediated by OATPs: A Systematic Review of Preclinical and Clinical Findings
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- (2015) Kazuya Maeda BIOLOGICAL & PHARMACEUTICAL BULLETIN
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- (2014) Bo Gao et al. PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY
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- (2012) Péter Tátrai et al. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
- Clinical significance of organic anion transporting polypeptides (OATPs) in drug disposition: their roles in hepatic clearance and intestinal absorption
- (2012) Yoshihisa Shitara et al. BIOPHARMACEUTICS & DRUG DISPOSITION
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- Reliable transgene-independent method for determining Sleeping Beauty transposon copy numbers
- (2011) Orsolya Kolacsek et al. Mobile DNA
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- (2010) Dallas Bednarczyk ANALYTICAL BIOCHEMISTRY
- Membrane transporters in drug development
- (2010) NATURE REVIEWS DRUG DISCOVERY
- Near-infrared fluorescent nanoprobes for cancer molecular imaging: status and challenges
- (2010) Xiaoxiao He et al. TRENDS IN MOLECULAR MEDICINE
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- (2010) P. Annaert et al. XENOBIOTICA
- Mechanisms of pH-gradient driven transport mediated by organic anion polypeptide transporters
- (2009) Simone Leuthold et al. AMERICAN JOURNAL OF PHYSIOLOGY-CELL PHYSIOLOGY
- Human Skeletal Muscle Drug Transporters Determine Local Exposure and Toxicity of Statins
- (2009) Michael J. Knauer et al. CIRCULATION RESEARCH
- The International Transporter Consortium: A Collaborative Group of Scientists From Academia, Industry, and the FDA
- (2009) S-M Huang et al. CLINICAL PHARMACOLOGY & THERAPEUTICS
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