A combination of docking and cheminformatics approaches for the identification of inhibitors against 4′ phosphopantetheinyl transferase of Mycobacterium tuberculosis

The Ecstasy and Agony of Assay Interference Compounds

(2017) Courtney Aldrich et al.   ACS Medicinal Chemistry Letters

Virtual Screening, pharmacophore development and structure based similarity search to identify inhibitors against IdeR, a transcription factor of Mycobacterium tuberculosis

(2017) Akshay Rohilla et al.   Scientific Reports

Mass spectral determination of phosphopantetheinylation specificity for carrier proteins in Mycobacterium tuberculosis

(2016) James Jung et al.   FEBS Open Bio

AcpM, the Meromycolate Extension Acyl Carrier Protein of Mycobacterium tuberculosis, Is Activated by the 4′-Phosphopantetheinyl Transferase PptT, a Potential Target of the Multistep Mycolic Acid Biosynthesis

(2015) Oren Zimhony et al.   BIOCHEMISTRY

Structure, Biochemistry, and Inhibition of Essential 4′-Phosphopantetheinyl Transferases from Two Species of Mycobacteria

(2014) Christopher R. Vickery et al.   ACS Chemical Biology

Crystal structure of the essential Mycobacterium tuberculosis phosphopantetheinyl transferase PptT, solved as a fusion protein with maltose binding protein

(2014) James Jung et al.   JOURNAL OF STRUCTURAL BIOLOGY

Fluorescent techniques for discovery and characterization of phosphopantetheinyl transferase inhibitors

(2013) Nicolas M Kosa et al.   JOURNAL OF ANTIBIOTICS

4′-Phosphopantetheinyl Transferase PptT, a New Drug Target Required for Mycobacterium tuberculosis Growth and Persistence In Vivo

(2013) Cécile Leblanc et al.   PLoS Pathogens

Rapid and flexible biochemical assays for evaluating 4′-phosphopantetheinyl transferase activity

(2011) Jeremy G. Owen et al.   BIOCHEMICAL JOURNAL

A strategy to discover inhibitors of Bacillus subtilis surfactin-type phosphopantetheinyl transferase

(2009) Adam Yasgar et al.   Molecular BioSystems