An organocatalytic asymmetric Mannich reaction of pyrazoleamides with cyclic trifluoromethyl ketimines: enantioselective access to dihydroquinazolinone skeletons

Organocatalytic asymmetric Michael addition of pyrazoleamides to β -phthalimidonitroethene

(2017) Yuan Luo et al.   TETRAHEDRON

Organocatalytic asymmetric [3+2] cycloaddition of N-2,2,2-trifluoroethylisatin ketimines with 3-alkenyl-5-arylfuran-2(3H)-ones

(2016) Zhen-Hua Wang et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Asymmetric Arylation of Trifluoromethylated/Perfluoroalkylated 2-Quinazolinones with High Enantioselectivity

(2016) Bo Zhou et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective direct vinylogous aldol-cyclization cascade reaction between β,γ-unsaturated amides and o-quinones

(2016) Yu Jiang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Organocatalytic asymmetric addition of alcohols to cyclic trifluoromethyl ketimines: highly enantioselective synthesis of chiral N,O-ketals

(2016) Ding Zhou et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective Vinylogous Michael/Cyclization Cascade Reaction of Acyclic β,γ-Unsaturated Amides with Isatylidene Malononitriles: Asymmetric Construction of Spirocyclic Oxindoles

(2015) Tian-Ze Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Organocatalytic enantio- and diastereoselective synthesis of highly substituted δ-lactones via a Michael-cyclization cascade

(2015) Santosh Agrawal et al.   CHEMICAL COMMUNICATIONS

3-Pyrrolyl-oxindoles as efficient nucleophiles for organocatalytic asymmetric synthesis of structurally diverse 3,3′-disubstituted oxindole derivatives

(2015) Bao-Dong Cui et al.   CHEMICAL COMMUNICATIONS

Diastereo- and enantioselective direct vinylogous Michael addition of γ-substituted butenolides to 2-enoylpyridines catalyzed by chiral bifunctional amine-squaramides

(2015) Zhen-Hua Wang et al.   CHEMICAL COMMUNICATIONS

Organocatalytic asymmetric Michael addition of 3-substituted oxindoles to α,β-unsaturated acyl phosphonates for the synthesis of 3,3′-disubstituted oxindoles with chiral squaramides

(2015) Lin Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A Quinine-Squaramide Catalyzed Enantioselective Aza-Friedel–Crafts Reaction of Cyclic Trifluoromethyl Ketimines with Naphthols and Electron-Rich Phenols

(2015) Ding Zhou et al.   ORGANIC LETTERS

Direct enantioselective vinylogous aldol–cyclization cascade reaction of allyl pyrazoleamides with isatins: asymmetric construction of spirocyclic oxindole–dihydropyranones

(2014) Tian-Ze Li et al.   CHEMICAL COMMUNICATIONS

Organocatalyzed Enantioselective Mannich Reaction of Pyrazoleamides with Isatin-Derived Ketimines

(2014) Tian-Ze Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Cinchona Alkaloid Squaramide/AgOAc Cooperatively Catalyzed Diastereo- and Enantioselective Mannich/Cyclization Cascade Reaction of Isocyanoacetates and Cyclic Trifluoromethyl Ketimines

(2014) Mei-Xin Zhao et al.   ORGANIC LETTERS

Chiral Phosphoric Acid-Catalyzed Asymmetric Aza-Friedel-Crafts Reaction of Indoles with CyclicN-Acylketimines: Enantioselective Synthesis of Trifluoromethyldihydroquinazolines

(2013) Ke-Feng Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Hydrogen-Bond-Directed Enantioselective Decarboxylative Mannich Reaction of β-Ketoacids with Ketimines: Application to the Synthesis of Anti-HIV Drug DPC 083

(2013) Hai-Na Yuan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Decarboxylative Mannich Reaction of Malonic Acid Half Oxyesters with Cyclic Trifluoromethyl Ketimines: Synthesis of β-Amino Esters and Anti-HIV Drug DPC 083

(2013) Hai-Na Yuan et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Highly Regio- and Diastereoselective Phosphane-Catalyzed [3+2] Annulation of Morita-Baylis-Hillman Carbonates with CyclicN-Acyl Ketimines

(2013) Li-Jun Yang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Bisphosphine-Triggered One-Pot Sequential [3 + 2]/[3 + 2] Annulation of Allenoates with Cyclic Ketimines

(2013) Li-Jun Yang et al.   ORGANIC LETTERS

Rationally Designed Amide Donors for Organocatalytic Asymmetric Michael Reactions

(2012) Bin Tan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly enantioselective organocatalytic Strecker reaction of cyclic N-acyl trifluoromethylketimines: synthesis of anti-HIV drug DPC 083

(2012) Fa-Guang Zhang et al.   CHEMICAL COMMUNICATIONS

Quinine-thiourea catalyzed enantioselective hydrophosphonylation of trifluoromethyl 2(1H)-quinazolinones

(2012) Hexin Xie et al.   CHEMICAL COMMUNICATIONS

Bifunctional Cinchona Alkaloid Thiourea Catalyzed Highly Efficient, Enantioselective Aza-Henry Reaction of Cyclic Trifluoromethyl Ketimines: Synthesis of Anti-HIV Drug DPC 083

(2011) Hexin Xie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stereoelectronic properties of spiroquinazolinones in differential PDE7 inhibitory activity

(2008) Pankaj R. Daga et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY