Access to 2-substituted-2H-indazoles via a copper-catalyzed regioselective cross-coupling reaction

Rh(III)-Catalyzed [4 + 1]-Annulation of Azoxy Compounds with Alkynes: A Regioselective Approach to 2H-Indazoles

(2017) Zhen Long et al.   ORGANIC LETTERS

Copper-Catalyzed Arylation with Diaryliodonium Salts

(2017) Martín Fañanás-Mastral   SYNTHESIS-STUTTGART

Iodine-catalyzed aerobic oxidation of o-alkylazoarenes to 2H-indazoles

(2017) Xiangli Yi et al.   TETRAHEDRON

A mild and regioselective Ullmann reaction of indazoles with aryliodides in water

(2017) Xiao Ding et al.   TETRAHEDRON

Copper-mediated annulation of 2-(1-arylvinyl) anilines and aryl nitrosos towards 2,3-diaryl-2H-indazoles

(2017) Weiming Hu et al.   Organic Chemistry Frontiers

Synthesis of 2H-IndazolesviaTandem Palladium-Catalyzed Deacylative Cross-Coupling and Denitrogenative Cyclization of 2-Iodoazoarenes and 2-Iodoaryltriazenes with Acyldiazoacetates in One-Pot

(2016) Woo-Soon Yong et al.   ADVANCED SYNTHESIS & CATALYSIS

Substrate-Controlled Transformation of Azobenzenes to Indazoles and Indoles via Rh(III)-Catalysis

(2016) Shangjun Cai et al.   JOURNAL OF ORGANIC CHEMISTRY

I2-Mediated 2H-indazole synthesis via halogen-bond-assisted benzyl C–H functionalization

(2016) Xiangli Yi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Organophosphorus-mediated N–N bond formation: facile access to 3-amino-2H-indazoles

(2016) Hassen Bel Abed et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

BF3·OEt2 mediated metal-free one-pot sequential multiple annulation cascade (SMAC) synthesis of complex and diverse tetrahydroisoquinoline fused hybrid molecules

(2016) Anand H. Shinde et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Access to 3-Acyl-(2H)-indazoles via Rh(III)-Catalyzed C–H Addition and Cyclization of Azobenzenes with α-Keto Aldehydes

(2016) Taejoo Jeong et al.   ORGANIC LETTERS

Functionalization of indazoles by means of transition metal-catalyzed cross-coupling reactions

(2016) Saïd El Kazzouli et al.   TETRAHEDRON

Synthesis of indazole motifs and their medicinal importance: An overview

(2015) Digambar D. Gaikwad et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rhenium-Catalyzed [4 + 1] Annulation of Azobenzenes and Aldehydes via Isolable Cyclic Rhenium(I) Complexes

(2015) Xiaoyu Geng et al.   ORGANIC LETTERS

Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor

(2015) Zining Wu et al.   ACS Combinatorial Science

Copper-Catalyzed Arylation of Nitrogen Heterocycles from Anilines under Ligand-Free Conditions

(2014) Dounia Toummini et al.   CHEMISTRY-A EUROPEAN JOURNAL

Davis–Beirut Reaction: Route to Thiazolo-, Thiazino-, and Thiazepino-2H-indazoles

(2014) Kelli M. Farber et al.   JOURNAL OF ORGANIC CHEMISTRY

Cobalt(III)-Catalyzed Synthesis of Indazoles and Furans by C–H Bond Functionalization/Addition/Cyclization Cascades

(2014) Joshua R. Hummel et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective Synthesis of 2H-Indazoles Using a Mild, One-Pot Condensation–Cadogan Reductive Cyclization

(2014) Nathan E. Genung et al.   ORGANIC LETTERS

Multiple functional therapeutic effects of the estrogen receptor β agonist indazole-Cl in a mouse model of multiple sclerosis

(2014) Spencer M. Moore et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Ligand-Free Copper(I) Oxide Nanoparticle Catalyzed Three-Component ­Synthesis of 2H-Indazole Derivatives from 2-Halobenzaldehydes, Amines and Sodium Azide in Polyethylene Glycol as a Green Solvent

(2014) Hashem Sharghi et al.   SYNLETT

A facile synthesis of 2H-indazoles under neat conditions and further transformation into aza-γ-carboline alkaloid analogues in a tandem one-pot fashion

(2014) Shinde Vidyacharan et al.   RSC Advances

Rhodium(III)-Catalyzed Indazole Synthesis by C–H Bond Functionalization and Cyclative Capture

(2013) Yajing Lian et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The poly(ADP-ribose) polymerase inhibitor niraparib (MK4827) in BRCA mutation carriers and patients with sporadic cancer: a phase 1 dose-escalation trial

(2013) Shahneen K Sandhu et al.   LANCET ONCOLOGY

Direct Access to Acylated Azobenzenes via Pd-Catalyzed C–H Functionalization and Further Transformation into an Indazole Backbone

(2013) Hongji Li et al.   ORGANIC LETTERS

Process Development of C–N Cross-Coupling and Enantioselective Biocatalytic Reactions for the Asymmetric Synthesis of Niraparib

(2013) Cheol K. Chung et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Ligand-free Cu2O-catalyzed cross coupling of nitrogen heterocycles with iodopyridines

(2013) Yong-Chua Teo et al.   TETRAHEDRON

CuO nanoparticle catalysed synthesis of 2H-indazoles under ligand free conditions

(2013) Nilufa Khatun et al.   RSC Advances

A general and efficient aldehyde decarbonylation reaction by using a palladium catalyst

(2012) Atanu Modak et al.   CHEMICAL COMMUNICATIONS

Pazopanib for metastatic soft-tissue sarcoma (PALETTE): a randomised, double-blind, placebo-controlled phase 3 trial

(2012) Winette TA van der Graaf et al.   LANCET

The Davis-Beirut Reaction: A Novel Entry into 2H-indazoles and Indazolones. Recent Biological Activity of Indazoles

(2012) Makhluf J. Haddadin et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

An efficient synthesis of 2H-indazoles via reductive cyclization of 2-nitrobenzylamines induced by low-valent titanium reagent

(2012) Fang Sun et al.   TETRAHEDRON

A general and efficient approach to 2H-indazoles and 1H-pyrazoles through copper-catalyzed intramolecular N–N bond formation under mild conditions

(2011) Jiantao Hu et al.   CHEMICAL COMMUNICATIONS

Synthesis of 2H-Indazoles by the [3 + 2] Dipolar Cycloaddition of Sydnones with Arynes

(2011) Yuesi Fang et al.   JOURNAL OF ORGANIC CHEMISTRY

Indazole: a medicinally important heterocyclic moiety

(2011) Ananda Thangadurai et al.   MEDICINAL CHEMISTRY RESEARCH

The Davis–Beirut Reaction:N1,N2-Disubstituted-1H-Indazolones via 1,6-Electrophilic Addition to 3-Alkoxy-2H-Indazoles

(2011) Wayne E. Conrad et al.   ORGANIC LETTERS

Consecutive Condensation, C–N and N–N Bond Formations: A Copper- Catalyzed One-Pot Three-Component Synthesis of 2H-Indazole

(2011) Manian Rajesh Kumar et al.   ORGANIC LETTERS

Regiospecific Reductive Elimination from Diaryliodonium Salts

(2010) Bijia Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pazopanib in Locally Advanced or Metastatic Renal Cell Carcinoma: Results of a Randomized Phase III Trial

(2010) Cora N. Sternberg et al.   JOURNAL OF CLINICAL ONCOLOGY

Synthesis of 2H-Indazoles by the [3 + 2] Cycloaddition of Arynes and Sydnones

(2010) Chunrui Wu et al.   ORGANIC LETTERS

Mild, base-free copper-catalyzed N-arylations of heterocycles using potassium aryltrifluoroborates in water under air

(2010) Nicolas Joubert et al.   TETRAHEDRON LETTERS

Diaryliodonium Salts: A Journey from Obscurity to Fame

(2009) Eleanor���A. Merritt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Safety, Pharmacokinetics, and Pharmacodynamics of Single Doses of LXR-623, a Novel Liver X-Receptor Agonist, in Healthy Participants

(2009) Arie Katz et al.   JOURNAL OF CLINICAL PHARMACOLOGY

Selective Synthesis of 1-Functionalized-alkyl-1H-indazoles§

(2009) Kevin W. Hunt et al.   ORGANIC LETTERS

Preparation of Polyfunctional Indazoles and Heteroarylazo Compounds Using Highly Functionalized Zinc Reagents

(2009) Benjamin Haag et al.   ORGANIC LETTERS